Discovery of Potent and Selective Dipeptidyl Peptidase IV Inhibitors Derived from β-Aminoamides Bearing Subsituted Triazolopiperazines
Kim, Dooseop, Kowalchick, Jennifer E, Brockunier, Linda L, Parmee, Emma R, Eiermann, George J, Fisher, Michael H, He, Huaibing, Leiting, Barbara, Lyons, Kathryn, Scapin, Giovanna, Patel, Sangita B, Petrov, Aleksandr, Pryor, KellyAnn D, Roy, Ranabir Sinha, Wu, Joseph K, Zhang, Xiaoping, Wyvratt, Matthew J, Zhang, Bei B, Zhu, Lan, Thornberry, Nancy A, Weber, Ann E
Published in Journal of medicinal chemistry (14.02.2008)
Published in Journal of medicinal chemistry (14.02.2008)
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Human β3-Adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides
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Published in Bioorganic & medicinal chemistry letters (01.09.2000)
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Design and evaluation of novel tetracyclic benzofurans as palm site allosteric inhibitors of HCV NS5B polymerase
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Asymmetric Synthesis of the Volatile Anesthetic 1,2,2,2-Tetrafluoroethyl Chlorofluoromethyl Ether Using a Stereospecific Decarboxylation of Unusual Stereochemical Outcome
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Human β 3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides
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HRUZA ALAN, GAO YING DUO, MONINGKA REMOND, MERTZ ERIC, LIU WEIGUO, ALI AMJAD, EDMONDSON SCOTT D, NEELAMKAVIL SANTHOSH F, SO SUNG SAU, SUN WANYING, BROCKUNIER LINDA L
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Heterocyclic acetamide and benzamide derivatives as potent and selective β3-adrenergic receptor agonists with improved rodent pharmacokinetic profiles
GOBLE, Stephen D, LIPING WANG, HURLEY, Amanda, HRENIUK, Donna, PARMEE, Emma, ROBBINS, Michael, SALITURO, Gino, SANFIZ, Anthony, STRECKFUSS, Eric, WATKINS, Eloisa, WEBER, Ann E, STRUTHERS, Mary, LULU HOWELL, K, EDMONDSON, Scott D, BANSAL, Alka, BERGER, Richard, BROCKUNIER, Linda, DISALVO, Jerry, FEIGHNER, Scott, HARPER, Bart, JIAFANG HE
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Year of Publication 16.01.2017
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Year of Publication 21.10.2015
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Year of Publication 21.10.2015
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Heterocyclic acetamide and benzamide derivatives as potent and selective b sub(3)-adrenergic receptor agonists with improved rodent pharmacokinetic profiles
Goble, Stephen D, Wang, Liping, Howell, KLulu, Bansal, Alka, Berger, Richard, Brockunier, Linda, DiSalvo, Jerry, Feighner, Scott, Harper, Bart, He, Jiafang, Hurley, Amanda, Hreniuk, Donna, Parmee, Emma, Robbins, Michael, Salituro, Gino, Sanfiz, Anthony, Streckfuss, Eric, Watkins, Eloisa, Weber, Ann E, Struthers, Mary, Edmondson, Scott D
Published in Bioorganic & medicinal chemistry letters (15.03.2010)
Published in Bioorganic & medicinal chemistry letters (15.03.2010)
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Heterocyclic acetamide and benzamide derivatives as potent and selective β 3-adrenergic receptor agonists with improved rodent pharmacokinetic profiles
Goble, Stephen D., Wang, Liping, Howell, K. Lulu, Bansal, Alka, Berger, Richard, Brockunier, Linda, DiSalvo, Jerry, Feighner, Scott, Harper, Bart, He, Jiafang, Hurley, Amanda, Hreniuk, Donna, Parmee, Emma, Robbins, Michael, Salituro, Gino, Sanfiz, Anthony, Streckfuss, Eric, Watkins, Eloisa, Weber, Ann E., Struthers, Mary, Edmondson, Scott D.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Discovery of Potent and Selective Dipeptidyl Peptidase IV Inhibitors Derived from [beta]-Aminoamides Bearing Subsituted Triazolopiperazines
Kim, Dooseop, Kowalchick, Jennifer E., Brockunier, Linda L., Parmee, Emma R., Eiermann, George J., Fisher, Michael H., He, Huaibing, Leiting, Barbara, Lyons, Kathryn, Scapin, Giovanna, Patel, Sangita B., Petrov, Aleksandr, Pryor, KellyAnn D., Roy, Ranabir Sinha, Wu, Joseph K., Zhang, Xiaoping, Wyvratt, Matthew J., Zhang, Bei B., Zhu, Lan, Thornberry, Nancy A., Weber, Ann E.
Published in Journal of medicinal chemistry (30.06.2008)
Published in Journal of medicinal chemistry (30.06.2008)
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