Acylideneoxoindoles: A new class of reversible inhibitors of human transglutaminase 2
Klöck, Cornelius, Jin, Xi, Choi, Kihang, Khosla, Chaitan, Madrid, Peter B., Spencer, Andrew, Raimundo, Brian C., Boardman, Paul, Lanza, Guido, Griffin, John H.
Published in Bioorganic & medicinal chemistry letters (01.05.2011)
Published in Bioorganic & medicinal chemistry letters (01.05.2011)
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Discovery of a Potent Small Molecule IL-2 Inhibitor through Fragment Assembly
Braisted, Andrew C, Oslob, Johan D, Delano, Warren L, Hyde, Jennifer, McDowell, Robert S, Waal, Nathan, Yu, Chul, Arkin, Michelle R, Raimundo, Brian C
Published in Journal of the American Chemical Society (02.04.2003)
Published in Journal of the American Chemical Society (02.04.2003)
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Identification of new inhibitors of protein kinase R guided by statistical modeling
Bryk, Ruslana, Wu, Kangyun, Raimundo, Brian C, Boardman, Paul E, Chao, Ping, Conn, Graeme L, Anderson, Eric, Cole, James L, Duffy, Nigel P, Nathan, Carl, Griffin, John H
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
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Integrating Fragment Assembly and Biophysical Methods in the Chemical Advancement of Small-Molecule Antagonists of IL-2: An Approach for Inhibiting Protein−Protein Interactions
Raimundo, Brian C, Oslob, Johan D, Braisted, Andrew C, Hyde, Jennifer, McDowell, Robert S, Randal, Mike, Waal, Nathan D, Wilkinson, Jennifer, Yu, Chul H, Arkin, Michelle R
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Tethering identifies fragment that yields potent inhibitors of human caspase-1
Fahr, Bruce T., O’Brien, Tom, Pham, Phuongly, Waal, Nathan D., Baskaran, Subramanian, Raimundo, Brian C., Lam, Joni W., Sopko, Michelle M., Purkey, Hans E., Romanowski, Michael J.
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Identification of nonpeptidic small-molecule inhibitors of interleukin-2
Waal, Nathan D., Yang, Wenjin, Oslob, Johan D., Arkin, Michelle R., Hyde, Jennifer, Lu, Wanli, McDowell, Robert S., Yu, Chul H., Raimundo, Brian C.
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
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Structural analysis of caspase-1 inhibitors derived from Tethering
Fahr, Bruce T., Sopko, Michelle M., Lam, Joni W., O'Brien, Tom, Waal, Nathan D., Pham, Phuongly, Purkey, Hans E., Raimundo, Brian C., Romanowski, Michael J.
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2005)
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2005)
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Acylidene oxoindoles: A new class of reversible inhibitors of human transglutaminase 2
Klöck, Cornelius, Jin, Xi, Choi, Kihang, Khosla, Chaitan, Madrid, Peter B., Spencer, Andrew, Raimundo, Brian C., Boardman, Paul, Lanza, Guido, Griffin, John H.
Published in Bioorganic & medicinal chemistry letters (16.12.2010)
Published in Bioorganic & medicinal chemistry letters (16.12.2010)
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