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Published in Journal of the American Chemical Society (18.03.1998)
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Matched and mixed cap derivatives in the tetracyclic indole class of HCV NS5A inhibitors
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Published in Bioorganic & medicinal chemistry letters (15.03.2010)
Published in Bioorganic & medicinal chemistry letters (15.03.2010)
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2-(2-Aminothiazol-4-yl)pyrrolidine-based tartrate diamides as potent, selective and orally bioavailable TACE inhibitors
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Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Biaryl substituted hydantoin compounds as TACE inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Rosner, Kristin E., Guo, Zhuyan, Orth, Peter, Shipps, Gerald W., Belanger, David B., Chan, Tin Yau, Curran, Patrick J., Dai, Chaoyang, Deng, Yongqi, Girijavallabhan, Vinay M., Hong, Liwu, Lavey, Brian J., Lee, Joe F., Li, Dansu, Liu, Zhidan, Popovici-Muller, Janeta, Ting, Pauline C., Vaccaro, Henry, Wang, Li, Wang, Tong, Yu, Wensheng, Zhou, Guowei, Niu, Xiaoda, Sun, Jing, Kozlowski, Joseph A., Lundell, Daniel J., Madison, Vincent, McKittrick, Brian, Piwinski, John J., Shih, Neng -Yang, Arshad Siddiqui, M., Strickland, Corey O.
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Discovery of novel spirocyclopropyl hydroxamate and carboxylate compounds as TACE inhibitors
Guo, Zhuyan, Orth, Peter, Wong, Shing-Chun, Lavey, Brian J., Shih, Neng-Yang, Niu, Xiaoda, Lundell, Daniel J., Madison, Vincent, Kozlowski, Joseph A.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Novel TNF-α converting enzyme (TACE) inhibitors as potential treatment for inflammatory diseases
Girijavallabhan, Vinay M., Chen, Lei, Dai, Chaoyang, Feltz, Robert J., Firmansjah, Luke, Li, Dansu, Kim, Seong Heon, Kozlowski, Joseph A., Lavey, Brian J., Kosinski, Aneta, Piwinski, John J., Popovici-Muller, Janeta, Rizvi, Razia, Rosner, Kristin E., Shankar, Banderpalle B., Shih, Neng-Yang, Siddiqui, M. Arshad, Tong, Ling, Wong, Michael K.C., Yang, De-yi, Yang, Liping, Yu, Wensheng, Zhou, Guowei, Guo, Zhuyan, Orth, Peter, Madison, Vincent, Bian, Hong, Lundell, Daniel, Niu, Xiaoda, Shah, Himanshu, Sun, Jing, Umland, Shelby
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
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Labelling and biological evaluation of [11 C]methoxy-Sch225336: a radioligand for the cannabinoid-type 2 receptor
Evens, Nele, Bosier, Barbara, Lavey, Brian J, Kozlowski, Joseph A, Vermaelen, Peter, Baudemprez, Luc, Busson, Roger, Lambert, Didier M, Van Laere, Koen, Verbruggen, Alfons M, Bormans, Guy M
Published in Nuclear medicine and biology (01.10.2008)
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Structure and activity relationships of tartrate-based TACE inhibitors
Li, Dansu, Popovici-Muller, Janeta, Belanger, David B., Caldwell, John, Dai, Chaoyang, David, Maria, Girijavallabhan, Vinay M., Lavey, Brian J., Lee, Joe F., Liu, Zhidan, Mazzola, Rob, Rizvi, Razia, Rosner, Kristin E., Shankar, Bandarpalle, Spitler, Jim, Ting, Pauline C., Vaccaro, Henry, Yu, Wensheng, Zhou, Guowei, Zhu, Zhaoning, Niu, Xiaoda, Sun, Jing, Guo, Zhuyan, Orth, Peter, Chen, Shiying, Kozlowski, Joseph A., Lundell, Daniel J., Madison, Vincent, McKittrick, Brian, Piwinski, John J., Shih, Neng-Yang, Shipps, Gerald W., Siddiqui, M. Arshad, Strickland, Corey O.
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
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Triaryl bis-sulfones as a new class of cannabinoid CB2 receptor inhibitors: identification of a lead and initial SAR studies
Lavey, Brian J., Kozlowski, Joseph A., Hipkin, R. William, Gonsiorek, Waldemar, Lundell, Daniel J., Piwinski, John J., Narula, Satwant, Lunn, Charles A.
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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Non-aromatic A-ring replacement in the triaryl bis-sulfone CB2 receptor inhibitors
Gilbert, Eric J., Zhou, Guowei, Wong, Michael K.C., Tong, Ling, Shankar, Bandarpalle B., Huang, Chunli, Kelly, Joseph, Lavey, Brian J., McCombie, Stuart W., Chen, Lei, Rizvi, Razia, Dong, Youhao, Shu, Youheng, Kozlowski, Joseph A., Shih, Neng-Yang, Hipkin, R. William, Gonsiorek, Waldemar, Malikzay, Asra, Lunn, Charles A., Favreau, Len, Lundell, Daniel J.
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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The discovery of novel tartrate-based TNF-a converting enzyme (TACE) inhibitors
Rosner, Kristin E, Guo, Zhuyan, Orth, Peter, Shipps, Gerald W, Belanger, David B, Chan, Tin Yau, Curran, Patrick J, Dai, Chaoyang, Deng, Yongqi, Girijavallabhan, Vinay M, Hong, Liwu, Lavey, Brian J, Lee, Joe F, Li, Dansu, Liu, Zhidan, Popovici-Muller, Janeta, Ting, Pauline C, Vaccaro, Henry, Wang, Li, Wang, Tong, Yu, Wensheng, Zhou, Guowei, Niu, Xiaoda, Sun, Jing, Kozlowski, Joseph A, Lundell, Daniel J, Madison, Vincent, McKittrick, Brian, Piwinski, John J, Shih, Neng-Yang, Siddiqui, MArshad, Strickland, Corey O
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Published in Bioorganic & medicinal chemistry letters (17.09.2010)
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Triaryl bis-sulfones as cannabinoid-2 receptor ligands: SAR studies
Shankar, Bandarpalle B., Lavey, Brian J., Zhou, Guowei, Spitler, James A., Tong, Ling, Rizvi, Razia, Yang, De-Yi, Wolin, Ronald, Kozlowski, Joseph A., Shih, Neng-Yang, Wu, Jie, Hipkin, R. William, Gonsiorek, Waldemar, Lunn, Charles A.
Published in Bioorganic & medicinal chemistry letters (15.10.2005)
Published in Bioorganic & medicinal chemistry letters (15.10.2005)
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Optimization of triaryl bis-sulfones as cannabinoid-2 receptor ligands
Lavey, Brian J., Kozlowski, Joseph A., Shankar, Bandarpalle B., Spitler, James M., Zhou, Guowei, Yang, De-Yi, Shu, Youheng, Wong, Michael K.C., Wong, Shing-Chun, Shih, Neng-Yang, Wu, Jie, McCombie, Stuart W., Rizvi, Razia, Wolin, Ronald L., Lunn, Charles A.
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
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Alkyl substituted aminal derivatives of HCV NS5A inhibitor MK-8742
Yu, Wensheng, Coburn, Craig A., Nair, Anilkumar G., Wong, Michael, Tong, Ling, Dwyer, Michael P., Hu, Bin, Zhong, Bin, Hao, Jinglai, Yang, De-Yi, Selyutin, Oleg, Jiang, Yueheng, Rosenblum, Stuart B., Kim, Seong Heon, Lavey, Brian J., Zhou, Guowei, Rizvi, Razia, Shankar, Bandarpalle B., Zeng, Qingbei, Chen, Lei, Agrawal, Sony, Carr, Donna, Rokosz, Laura, Liu, Rong, Curry, Stephanie, McMonagle, Patricia, Ingravallo, Paul, Lahser, Fred, Asante-Appiah, Ernest, Nomeir, Amin, Kozlowski, Joseph A.
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
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Syntheses of 9.beta.-(Hydroxymethyl)-4,4,10.beta.-trimethyl- trans-decal-3.beta.-ol
Lavey, Brian J, Westkaemper, John G, Spencer, Thomas A
Published in Journal of organic chemistry (01.09.1994)
Published in Journal of organic chemistry (01.09.1994)
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Selective benzylic lithiation of N-boc-2-phenylpiperidine and pyrrolidine: expedient synthesis of a 2,2-disubstituted piperidine NK1 antagonist
Xiao, D, Lavey, BJ, Palani, A, Wang, C, Aslanian, RG, Kozlowski, JA, Shih, NY, McPhail, AT, Randolph, GP, Lachowicz, JE, Duffy, RA
Published in Tetrahedron letters (31.10.2005)
Published in Tetrahedron letters (31.10.2005)
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Selective benzylic lithiation of N-Boc-2-phenylpiperidine and pyrrolidine: expedient synthesis of a 2,2-disubstituted piperidine NK 1 antagonist
Xiao, Dong, Lavey, Brian J., Palani, Anandan, Wang, Cheng, Aslanian, Robert G., Kozlowski, Joseph A., Shih, Neng-Yang, McPhail, Andrew T., Randolph, Gerard P., Lachowicz, Jean E., Duffy, Ruth A.
Published in Tetrahedron letters (2005)
Published in Tetrahedron letters (2005)
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