Isolation and structure of an intrastrand cross-link adduct of mitomycin C and DNA
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Published in Biochemistry (Easton) (31.03.1992)
Published in Biochemistry (Easton) (31.03.1992)
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IV. Discovery of CXCR3 antagonists substituted with heterocycles as amide surrogates: improved PK, hERG and metabolic profiles
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Published in Bioorganic & medicinal chemistry letters (15.11.2010)
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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Discovery of 2-aminoimidazopyridine adenosine A2A receptor antagonists
McGuinness, Brian F., Cole, Andrew G., Dong, Guizhen, Brescia, Marc-Raleigh, Shao, Yuefei, Henderson, Ian, Rokosz, Laura L., Stauffer, Tara M., Mannava, Neelima, Kimble, Earl F., Hicks, Catherine, White, Nicole, Wines, Pamela G., Quadros, Elizabeth
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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Synthesis and SAR studies of trisubstituted purinones as potent and selective adenosine A2A receptor antagonists
Shao, Yuefei, Cole, Andrew G, Brescia, Marc-Raleigh, Qin, Lan-Ying, Duo, Jingqi, Stauffer, Tara M, Rokosz, Laura L, McGuinness, Brian F, Henderson, Ian
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
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III. Identification of novel CXCR3 chemokine receptor antagonists with a pyrazinyl–piperazinyl–piperidine scaffold
Kim, Seong Heon, Anilkumar, Gopinadhan N., Zawacki, Lisa Guise, Zeng, Qingbei, Yang, De-Yi, Shao, Yuefei, Dong, Guizhen, Xu, Xiaolian, Yu, Wensheng, Jiang, Yueheng, Jenh, Chung-Her, Hall, James W., Carroll, Carolyn DiIanni, Hobbs, Doug W., Baldwin, John J., McGuinness, Brian F., Rosenblum, Stuart B., Kozlowski, Joseph A., Shankar, Bandarpalle B., Shih, Neng-Yang
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
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Novel CXCR3 antagonists with a piperazinyl-piperidine core
McGuinness, Brian F., Carroll, Carolyn DiIanni, Zawacki, Lisa Guise, Dong, Guizhen, Yang, Cangming, Hobbs, Doug W., Jacob-Samuel, Biji, Hall, James W., Jenh, Chung-Her, Kozlowski, Joseph A., Anilkumar, Gopinadhan N., Rosenblum, Stuart B.
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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II. SAR studies of pyridyl–piperazinyl-piperidine derivatives as CXCR3 chemokine antagonists
Shao, Yuefei, Anilkumar, Gopinadhan N., Carroll, Carolyn DiIanni, Dong, Guizhen, Hall, James W., Hobbs, Doug W., Jiang, Yueheng, Jenh, Chung-Her, Kim, Seong Heon, Kozlowski, Joseph A., McGuinness, Brian F., Rosenblum, Stuart B., Schulman, Inna, Shih, Neng-Yang, Shu, Youheng, Wong, Michael K.C., Yu, Wensheng, Zawacki, Lisa Guise, Zeng, Qingbei
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
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Discovery of novel quinolinone adenosine A2B antagonists
MCGUINNESS, Brian F, HO, Koc-Kan, ROGERS, W. Lynn, WEBB, Maria, JUXING YIN, YAN JIANG, TAILONG LI, HAO YAN, KONGHUA JING, SHENGTING ZHANG, KANAK KANTI MAJUMDAR, SRIVASTAVA, Vikash, STAUFFER, Tara M, SAHA, Samiran, ROKOSZ, Laura L, MANNAVA, Neelima, KULTGEN, Steven G, SAIONZ, Kurt, KLON, Anthony, WEIQING CHEN, DESAI, Hema
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
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Small molecule biaryl FSH receptor agonists. Part 1: Lead discovery via encoded combinatorial synthesis
Guo, Tao, Adang, Anton E.P., Dolle, Roland E., Dong, Guizhen, Fitzpatrick, Dan, Geng, Peng, Ho, Koc-Kan, Kultgen, Steven G., Liu, Ruiyan, McDonald, Edward, McGuinness, Brian F., Saionz, Kurt W., Valenzano, Kenneth J., van Straten, Nicole C.R., Xie, Dan, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (05.04.2004)
Published in Bioorganic & medicinal chemistry letters (05.04.2004)
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Year of Publication 26.07.2018
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Year of Publication 26.07.2018
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HETEROCYCLE AMINES AND USES THEREOF
PICKENS JASON C, PEDRAM BIJAN, JEFFREY J LETOURNEAU, ANDREW G COLE, QI LIN, HO KOC-KAN, ROSEN DAVID, SHEN YIXING, DAVID DILLER, BRIAN F MCGUINNESS, CORNELIS A VAN OEVEREN
Year of Publication 19.01.2017
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Year of Publication 19.01.2017
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Isolation and characterization of a major adduct between mitomycin C and DNA
Tomasz, Maria, Lipman, Roselyn, McGuinness, Brian F, Nakanishi, Koji
Published in Journal of the American Chemical Society (01.08.1988)
Published in Journal of the American Chemical Society (01.08.1988)
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Reductive alkylation of DNA by mitomycin A, a mitomycin with high redox potential
McGuinness, Brian F, Lipman, Roselyn, Goldstein, Jeffrey, Nakanishi, Koji, Tomasz, Maria
Published in Biochemistry (Easton) (02.07.1991)
Published in Biochemistry (Easton) (02.07.1991)
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Discovery of novel quinolinone adenosine A sub(2B) antagonists
McGuinness, Brian F, Ho, Koc-Kan, Stauffer, Tara M, Rokosz, Laura L, Mannava, Neelima, Kultgen, Steven G, Saionz, Kurt, Klon, Anthony, Chen, Weiqing, Desai, Hema, Rogers, WLynn, Webb, Maria, Yin, Juxing, Jiang, Yan, Li, Tailong, Yan, Hao, Jing, Konghua, Zhang, Shengting, Majumdar, Kanak Kanti, Srivastava, Vikash, Saha, Samiran
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
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Synthesis and SAR studies of trisubstituted purinones as potent and selective adenosine A 2A receptor antagonists
Shao, Yuefei, Cole, Andrew G., Brescia, Marc-Raleigh, Qin, Lan-Ying, Duo, Jingqi, Stauffer, Tara M., Rokosz, Laura L., McGuinness, Brian F., Henderson, Ian
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Discovery of novel quinolinone adenosine A 2B antagonists
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Published in Bioorganic & medicinal chemistry letters (2010)
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Sting agonists for treating bladder cancer and solid tumors
Gallagher, Grant, Diller, David J, McGuinness, Brian F, McQueney, Michael S, Nazan Eraslan, Rukiye, Schieven, Gary, Kaelin, David E, Trama, Jason, Metzger, Axel
Year of Publication 30.01.2024
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Year of Publication 30.01.2024
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