Commercial Route Research and Development for SGLT2 Inhibitor Candidate Ertugliflozin
Bowles, Paul, Brenek, Steven J, Caron, Stéphane, Do, Nga M, Drexler, Michele T, Duan, Shengquan, Dubé, Pascal, Hansen, Eric C, Jones, Brian P, Jones, Kris N, Ljubicic, Tomislav A, Makowski, Teresa W, Mustakis, Jason, Nelson, Jade D, Olivier, Mark, Peng, Zhihui, Perfect, Hahdi H, Place, David W, Ragan, John A, Salisbury, John J, Stanchina, Corey L, Vanderplas, Brian C, Webster, Mark E, Weekly, R. Matt
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
A Robust, Streamlined Approach to Bosutinib Monohydrate
Withbroe, Gregory J, Seadeek, Chris, Girard, Kevin P, Guinness, Steven M, Vanderplas, Brian C, Vaidyanathan, Rajappa
Published in Organic process research & development (15.03.2013)
Published in Organic process research & development (15.03.2013)
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Journal Article
Synthesis of Filibuvir. Part II. Second-Generation Synthesis of a 6,6-Disubstituted 2H‑Pyranone via Dieckmann Cyclization of a β‑Acetoxy Ester
Peng, Zhihui, Ragan, John A, Colon-Cruz, Roberto, Conway, Brian G, Cordi, Eric M, Leeman, Kyle, Letendre, Leo J, Ping, Li-Jen, Sieser, Janice E, Singer, Robert A, Sluggett, Gregory W, Strohmeyer, Holly, Vanderplas, Brian C, Blunt, Jon, Mawby, Nicola, Meldrum, Kevin, Taylor, Stuart
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
Development of a Practical and Efficient Synthesis of Chloromethyl 2-Ethoxy-2-methylpropanoate
Ragan, John A, Ide, Nathan D, Cai, Weiling, Cawley, James J, Colon-Cruz, Roberto, Kumar, Rajesh, Peng, Zhihui, Vanderplas, Brian C
Published in Organic process research & development (19.11.2010)
Published in Organic process research & development (19.11.2010)
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Journal Article
LARGE SCALE, GREEN SYNTHESIS OF A GENERATION-1 MELAMINE (TRIAZINE) DENDRIMER
Chouai, Abdellatif, Venditto, Vincent J, Simanek, Eric E, Vanderplas, Brian C, Ragan, John A
Published in Organic syntheses (01.01.2009)
Published in Organic syntheses (01.01.2009)
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Journal Article
Development of a Practical and Efficient Synthesis of CP-945,598-01, a CB1 Antagonist for the Treatment of Obesity
Ragan, John A, Bourassa, Dennis E, Blunt, Jon, Breen, Darragh, Busch, Frank R, Cordi, Eric M, Damon, David B, Do, Nga, Engtrakul, Alanya, Lynch, Denis, McDermott, Ruth E, Mongillo, Joseph A, O’Sullivan, Maria M, Rose, Peter R, Vanderplas, Brian C
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Journal Article
Safe Execution of a Large-Scale Ozonolysis: Preparation of the Bisulfite Adduct of 2-Hydroxyindan-2-carboxaldehyde and Its Utility in a Reductive Amination
Ragan, John A, am Ende, David J, Brenek, Steven J, Eisenbeis, Shane A, Singer, Robert A, Tickner, Derek L, Teixeira, John J, Vanderplas, Brian C, Weston, Neil
Published in Organic process research & development (01.03.2003)
Published in Organic process research & development (01.03.2003)
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Journal Article
Process Research and Scale-up of the κ-Opioid Receptor Agonist CJ-15,161 Drug Candidate
Brian M. Andresen, Brian C. Vanderplas, John L. Tucker, Janice E. Sieser, Maxime Riou, Teresa M. Makowski, Joel M. Hawkins, Melina Girardin, Arun Ghosh, Kristina Dupont-Gaudet, Nga M. Do, Keith M. DeVries, Michel Couturier, Stéphane Caron, Timothy J.N. Watson
Published in Chimia (01.01.2006)
Published in Chimia (01.01.2006)
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Journal Article
Oxidation of carbamate-protected alkylhydrazines to the corresponding hydrazones under Swern conditions
Dupont, Joseph, Bemish, R.J, McCarthy, Keith E, Payne, Emily R, Pollard, Ernest B, Ripin, David H.B, Vanderplas, Brian C, Watrous, Richard M
Published in Tetrahedron letters (19.02.2001)
Published in Tetrahedron letters (19.02.2001)
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Journal Article
Synthesis of an optically active octahydro-2H-pyrido[1,2-a]pyrazine based CNS agent
Urban, Frank J, Breitenbach, Ralph, Murtiashaw, Charles W, Vanderplas, Brian C
Published in Tetrahedron: asymmetry (01.02.1995)
Published in Tetrahedron: asymmetry (01.02.1995)
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Journal Article
Development of two synthetic routes to CE-178,253, a CB1 antagonist for the treatment of obesity
Brandt, Thomas A., Caron, Stephane, Damon, David B., DiBrino, Joseph, Ghosh, Arun, Griffith, David A., Kedia, Sandeep, Ragan, John A., Rose, Peter R., Vanderplas, Brian C., Wei, Lulin
Published in Tetrahedron (18.04.2009)
Published in Tetrahedron (18.04.2009)
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Journal Article
Synthesis of Filibuvir. Part II. Second-Generation Synthesis of a 6,6-Disubstituted 2 H -Pyranone via Dieckmann Cyclization of a β-Acetoxy Ester
Peng, Zhihui, Ragan, John A., Colon-Cruz, Roberto, Conway, Brian G., Cordi, Eric M., Leeman, Kyle, Letendre, Leo J., Ping, Li-Jen, Sieser, Janice E., Singer, Robert A., Sluggett, Gregory W., Strohmeyer, Holly, Vanderplas, Brian C., Blunt, Jon, Mawby, Nicola, Meldrum, Kevin, Taylor, Stuart
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
Development of two synthetic routes to CE-178,253, a CB1 antagonist for the treatment of obesity: Recent Advances in Synthetic Methodology: Development and Applications
BRANDT, Thomas A, CARON, Stéphane, LULIN WEI, DAMON, David B, DIBRINO, Joseph, GHOSH, Arun, GRIFFITH, David A, KEDIA, Sandeep, RAGAN, John A, ROSE, Peter R, VANDERPLAS, Brian C
Published in Tetrahedron (2009)
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Published in Tetrahedron (2009)
Journal Article
Development of a Practical and Efficient Synthesis of CP-945,598-01, a CB 1 Antagonist for the Treatment of Obesity
Ragan, John A., Bourassa, Dennis E., Blunt, Jon, Breen, Darragh, Busch, Frank R., Cordi, Eric M., Damon, David B., Do, Nga, Engtrakul, Alanya, Lynch, Denis, McDermott, Ruth E., Mongillo, Joseph A., O’Sullivan, Maria M., Rose, Peter R., Vanderplas, Brian C.
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Journal Article
Efficient synthesis of the κ-opioid receptor agonist CJ-15,161: four stereospecific inversions at a single aziridinium stereogenic center
Couturier, Michel, Tucker, John L., Andresen, Brian M., DeVries, Keith M., Vanderplas, Brian C., Ito, Fumitaka
Published in Tetrahedron: asymmetry (14.11.2003)
Published in Tetrahedron: asymmetry (14.11.2003)
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Journal Article
The preparation of β-substituted amines from mixtures of epoxide opening products via a common aziridinium ion intermediate
Anderson, Shelby R., Ayers, Joshua T., DeVries, Keith M., Fumitaka Ito, Mendenhall, Debra, Vanderplas, Brian C.
Published in Tetrahedron: asymmetry (16.07.1999)
Published in Tetrahedron: asymmetry (16.07.1999)
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Journal Article
Corrigendum to “Oxidation of carbamate-protected alkylhydrazines to the corresponding hydrazones under Swern conditions”: [Tetrahedron Letters 42 (2001) 1453–1454]
Dupont, Joseph, Bemish, R.J., McCarthy, Keith E., Payne, Emily R., Pollard, Ernest B., Ripin, David H.B., Vanderplas, Brian C., Watrous, Richard M.
Published in Tetrahedron letters (01.08.2001)
Published in Tetrahedron letters (01.08.2001)
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