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Identification of new inhibitors of protein kinase R guided by statistical modeling
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Integrating Fragment Assembly and Biophysical Methods in the Chemical Advancement of Small-Molecule Antagonists of IL-2: An Approach for Inhibiting Protein−Protein Interactions
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Published in Journal of medicinal chemistry (03.06.2004)
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Tethering identifies fragment that yields potent inhibitors of human caspase-1
Fahr, Bruce T., O’Brien, Tom, Pham, Phuongly, Waal, Nathan D., Baskaran, Subramanian, Raimundo, Brian C., Lam, Joni W., Sopko, Michelle M., Purkey, Hans E., Romanowski, Michael J.
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Identification of nonpeptidic small-molecule inhibitors of interleukin-2
Waal, Nathan D., Yang, Wenjin, Oslob, Johan D., Arkin, Michelle R., Hyde, Jennifer, Lu, Wanli, McDowell, Robert S., Yu, Chul H., Raimundo, Brian C.
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
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Structural analysis of caspase-1 inhibitors derived from Tethering
Fahr, Bruce T., Sopko, Michelle M., Lam, Joni W., O'Brien, Tom, Waal, Nathan D., Pham, Phuongly, Purkey, Hans E., Raimundo, Brian C., Romanowski, Michael J.
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2005)
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2005)
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Acylidene oxoindoles: A new class of reversible inhibitors of human transglutaminase 2
Klöck, Cornelius, Jin, Xi, Choi, Kihang, Khosla, Chaitan, Madrid, Peter B., Spencer, Andrew, Raimundo, Brian C., Boardman, Paul, Lanza, Guido, Griffin, John H.
Published in Bioorganic & medicinal chemistry letters (16.12.2010)
Published in Bioorganic & medicinal chemistry letters (16.12.2010)
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Substituted pyrimidines for inhibiting Raf kinase activity
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Year of Publication 20.03.2018
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Year of Publication 20.03.2018
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Year of Publication 08.06.2017
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Year of Publication 08.06.2017
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Compounds useful as Raf kinase inhibitors
JONES JOHN HOWARD, TANAKA HIROKO, POWELL NOEL, KUMARAVEL GNANASAMBANDAM, WYNN THOMAS, GUAN BING, XIN ZHILI, COSSROW JENNIFER, PENG HAIRUO, VESSELS JEFFREY, LUGOVSKOY ALEXEY, RAIMUNDO BRIAN C
Year of Publication 12.08.2014
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Year of Publication 12.08.2014
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COMPOUNDS USEFUL AS RAF KINASE INHIBITORS
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Year of Publication 25.02.2015
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COMPOUNDS USEFUL AS RAF KINASE INHIBITORS
JONES JOHN HOWARD, TANAKA HIROKO, POWELL NOEL, WYNN THOMAS, GUAN BING, XIN ZHILI, COSSROW JENNIFER, LUGOVSKOY ALEXEY, KUMARAVEL GNANASAMBANDAM, LANE BENJAMIN, FRANKLIN LLOYD, CHEN WEIRONG, PENG HAIRUO, VESSELS JEFFREY, LITTKE ADAM, RAIMUNDO BRIAN C
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Year of Publication 14.03.2013
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Compounds useful as Raf kinase inhibitors
JONES JOHN HOWARD, TANAKA HIROKO, POWELL NOEL, WYNN THOMAS, GUAN BING, XIN ZHILI, COSSROW JENNIFER, LUGOVSKOY ALEXEY, KUMARAVEL GNANASAMBANDAM, LANE BENJAMIN, FRANKLIN LLOYD, CHEN WEIRONG, PENG HAIRUO, VESSELS JEFFREY, LITTKE ADAM, RAIMUNDO BRIAN C
Year of Publication 23.10.2012
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Year of Publication 23.10.2012
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Compounds useful as Raf kinase inhibitors
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Year of Publication 23.10.2012
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Year of Publication 23.10.2012
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Heterocyclic compounds useful as RAF kinase inhibitors
JONES JOHN HOWARD, ISHCHENKO ALEXEY, TANAKA HIROKO, POWELL NOEL, WYNN THOMAS, GUAN BING, XIN ZHILI, COSSROW JENNIFER, LUGOVSKOY ALEXEY, KUMARAVEL GNANASAMBANDAM, PENG HAIRUO, VESSELS JEFFREY, RAIMUNDO BRIAN C
Year of Publication 28.06.2011
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Year of Publication 28.06.2011
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Heterocyclic compounds useful as RAF kinase inhibitors
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Year of Publication 28.06.2011
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Year of Publication 28.06.2011
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