Synthesis and evaluation of 5-HT2A and 5-HT2C receptor binding affinities of novel pyrimidine derivatives
BOZSING, Daniel, SIMONEK, Ildiko, SIMIG, Gyula, JAKOCZI, Ivan, GACSALYI, Istvan, LEVAY, György, TIHANYI, Karoly, SCHMIDT, Eva
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
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Journal Article
Effects of EGIS-7625, a selective and competitive 5-HT2B receptor antagonist
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Published in Cardiovascular drugs and therapy (01.09.2003)
Published in Cardiovascular drugs and therapy (01.09.2003)
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Process for the preparation of quetiapine and intermediates therefore
KRASZNAI GYORGY, RAKOCZY GYORGYNE, KOVANYINE LAX GYORGYI, NAGY KALMAN, TOMPE PETER, VERECZKEYNE DONATH GYORGYI, BOZSING DANIEL, SIMIG GYULA
Year of Publication 08.02.2010
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Year of Publication 08.02.2010
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Quinazoline derivatives, process for the preparation thereof and pharmaceutical compositions comprising the same
Molnarne dr. Samu Erika, dr. Volk Balazs, dr. Bozsing Daniel, dr. Megyeri Katalin, Antoni Ferenc, dr. Kertesz Szabolcs, dr. Poszavacz Laszlo, dr. Barkoczy Jozsef, dr. Gacsalyi Istvan
Year of Publication 28.03.2017
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Year of Publication 28.03.2017
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Synthesis and Evaluation of 5‐HT 2A and 5‐HT 2C Receptor Binding Affinities of Novel Pyrimidine Derivatives
Bozsing, Daniel, Simonek, Ildiko, Simig, Gyula, Jakoczi, Ivan, Gacsalyi, Istvan, Levay, Gyoergy, Tihanyi, Karoly, Schmidt, Eva
Published in ChemInform (25.02.2003)
Published in ChemInform (25.02.2003)
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Quinazoline derivatives, process for the preparation thereof and pharmaceutical compositions comprising the same
MEGYERI KATALIN, BARKOCZY JOZSEF, GACSALYI ISTVAN, VOLK BALAZS, KERTESZ SZABOLCS, BOZSING DANIEL, MOLNARNE SAMU ERIKA, POSZAVACZ LASZLO, ANTONI FERENC
Year of Publication 29.12.2014
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Year of Publication 29.12.2014
Patent
NOVEL PIPERAZINYL ALKYLTHIO PYRIMIDINYL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH ACTIVE INGREDIENTS AND PROCESS FOR PRODUCING THE ACTIVE INGREDIENTS
TIHANYI KAROLY DR, NEMETH GABOR, GACSALYI ISTVAN, LEVAY GYOERGY DR, WELLMANN JANOS DR, RATZNE SIMONEK ILDIKO DR, EGYED ANDRAS DR, POSZAVACZ LASZLO, BOZSING DANIEL DR, JAKOCZI IVAN, SIMIG GYULA DR
Year of Publication 30.05.2011
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Year of Publication 30.05.2011
Patent
Piperazinylalkylthiopyrimidine derivatives, pharmaceutical compositions containing the same, and a process for their preparation
EGYED ANDRAS, NEMETH GABOR, WELLMAN JANOS, RATZNE SIMONEK ILDIKO, GACSALYI ISTVAN, TIHANYI KAROLY, LEVAY GYORGY, BOZSING DANIEL, SIMIG GYULA, POSZAVACZ LASZLO, JAKOCZI IVAN
Year of Publication 07.06.2007
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Year of Publication 07.06.2007
Patent
A PROCESS FOR THE PREPARATION OF QUETIAPINE AND INTERMEDIATES THEREOF
GYOERGYI VERECZKEYNE DONATH, GYULA SIMIG, KALMAN NAGY, GYOERGYI KOVANYINE LAX, GYOERGYNE RAKOCZY, PETER TOEMPE, DANIEL BOZSING, GYOERGY KRASZNAI
Year of Publication 31.08.2005
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Year of Publication 31.08.2005
Patent
METHOD OF SYNTHESIS OF 3-ETHYL-5-METHYL-2-(2-AMINOETHOXYMETHYL)- 4-(2-CHLOROPHENYL)-6-METHYL-1,4-DIHYDRO-3,5-PYRIDINE DICARBO-XYLATE AND BENZENESULFOACID SALT, and their intermediates
KRASZNAI GYORGY, BLASKO GABOR, NAGY KALMAN, VERECZKEY GYORGYI DONATH, TOMPE PETER, BOZSING DANIEL, SIMIG GYULA, NEMETH NORBERT, KOVANYI GYORGYI LAX, NEMET GABOR
Year of Publication 31.08.2006
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Year of Publication 31.08.2006
Patent
Ethyl 4-(2-chloroetoxy) acetoacetate, ethyl 4-(2-iodoetoxy) acetoacetate, ethyl 4-(2-chloroetoxy)-2-(2-chlorobenzylidene) acetoacetate and ethyl 4-(2-iodoetoxy)-2-(2-chlorobenzolidene) acetoacetate
KRASZNAI GYORGY, BLASKO GABOR, NAGY KALMAN, VERECZKEY GYORGYI DONATH, TOMPE PETER, BOZSING DANIEL, SIMIG GYULA, NEMETH NORBERT, KOVANYI GYORGYI LAX, NEMET GABOR
Year of Publication 31.08.2006
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Year of Publication 31.08.2006
Patent
A PROCESS FOR THE PREPARATION OF QUETIAPINE AND INTERMEDIATES THEREFOR
KRASZNAI GYORGY, RAKOCZY GYORGYNE, KOVANYINE LAX GYORGYI, NAGY KALMAN, TOMPE PETER, VERECZKEYNE DONATH GYORGYI, BOZSING DANIEL, SIMIG GYULA
Year of Publication 17.05.2004
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Year of Publication 17.05.2004
Patent