Rapid and Selective Cleavage of Amide Groups at Neutral pH: Applications from Hyaluronic Acid to Small Molecules
Jing, Jing, Bankefors, Johan, Bonneaud, Céline, Sawen, Elin, Gerfaud, Thibaud, Westin, Jonatan, El‐Bazbouz, Ghizlane, Kandelin, Lina, Rousseau, Antoine, Olsson, Johan, Karlsson, Anders, Nord, Lars, Bouix‐Peter, Claire, Helander Kenne, Anne, Boiteau, Jean‐Guy, Tomas, Loic, Hennequin, Laurent, Harris, Craig S.
Published in European journal of organic chemistry (22.06.2018)
Published in European journal of organic chemistry (22.06.2018)
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Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis
Ouvry, Gilles, Atrux‐Tallau, Nicolas, Bihl, Franck, Bondu, Aline, Bouix‐Peter, Claire, Carlavan, Isabelle, Christin, Olivier, Cuadrado, Marie‐Josée, Defoin‐Platel, Claire, Deret, Sophie, Duvert, Denis, Feret, Christophe, Forissier, Mathieu, Fournier, Jean‐François, Froude, David, Hacini‐Rachinel, Fériel, Harris, Craig Steven, Hervouet, Catherine, Huguet, Hélène, Lafitte, Guillaume, Luzy, Anne‐Pascale, Musicki, Branislav, Orfila, Danielle, Ozello, Benjamin, Pascau, Coralie, Pascau, Jonathan, Parnet, Véronique, Peluchon, Guillaume, Pierre, Romain, Piwnica, David, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent François
Published in ChemMedChem (20.02.2018)
Published in ChemMedChem (20.02.2018)
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Rational design of a JAK1-selective siRNA inhibitor for the modulation of autoimmunity in the skin
Tang, Qi, Fakih, Hassan H., Zain UI Abideen, Mohammad, Hildebrand, Samuel R., Afshari, Khashayar, Gross, Katherine Y., Sousa, Jacquelyn, Maebius, Allison S., Bartholdy, Christina, Søgaard, Pia Pernille, Jackerott, Malene, Hariharan, Vignesh, Summers, Ashley, Fan, Xueli, Okamura, Ken, Monopoli, Kathryn R., Cooper, David A., Echeverria, Dimas, Bramato, Brianna, McHugh, Nicholas, Furgal, Raymond C., Dresser, Karen, Winter, Sarah J., Biscans, Annabelle, Chuprin, Jane, Haddadi, Nazgol-Sadat, Sherman, Shany, Yıldız-Altay, Ümmügülsüm, Rashighi, Mehdi, Richmond, Jillian M., Bouix-Peter, Claire, Blanchard, Carine, Clauss, Adam, Alterman, Julia F., Khvorova, Anastasia, Harris, John E.
Published in Nature communications (04.11.2023)
Published in Nature communications (04.11.2023)
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Multispecies-targeting siRNAs for the modulation of JAK1 in the skin
Tang, Qi, Gross, Katherine Y., Fakih, Hassan H., Jackson, Samuel O., Zain U.I. Abideen, Mohammad, Monopoli, Kathryn R., Blanchard, Carine, Bouix-Peter, Claire, Portal, Thibaud, Harris, John E., Khvorova, Anastasia, Alterman, Julia F.
Published in Molecular therapy. Nucleic acids (12.03.2024)
Published in Molecular therapy. Nucleic acids (12.03.2024)
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Novel library synthesis of 3,4-disubstituted pyridin-2(1 H )-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperature
Pierre, Romain, Brethon, Anne, Jacques, Sylvain A, Blond, Aurélie, Chambon, Sandrine, Talano, Sandrine, Raffin, Catherine, Musicki, Branislav, Bouix-Peter, Claire, Tomas, Loic, Ouvry, Gilles, Morgentin, Rémy, Hennequin, Laurent F, Harris, Craig S
Published in Beilstein journal of organic chemistry (2021)
Published in Beilstein journal of organic chemistry (2021)
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CHIMIE, DERMO-COSMETIQUE ET BEAUTE
Andre, Patrice, Aubry, Jean-Marie, Berteina-Raboin, Sabine, Bouix-Peter, Claire, Bino, Sandra Del, Humbert, Philippe, Leclaire, Jacques, Marrot, Laurent, Masson, Christophe, Pelisson, Isabelle, Piccerelle, Philippe, Walter, Philippe, Dinh-Audouin, Minh-Thu, Olivier, Daniele, Rigny, Paul
Year of Publication 03.01.2017
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Year of Publication 03.01.2017
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Sugar-Derived Aziridines: Functionalization via Lithiation of the Aziridine Ring
Bisseret, Philippe, Bouix-Peter, Claire, Jacques, Olivier, Henriot, Stéphanie, Eustache, Jacques
Published in Organic letters (21.10.1999)
Published in Organic letters (21.10.1999)
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Discovery of a novel series of selective macrocyclic PKCTheta inhibitors
Crosignani, Stefano, Campos, Sebastien, Bouix-Peter, Claire, Harris, Craig, Talbot, Eric, Hu, Haiyang, Wang, Shun, Maclean, John, Zanelli, Ugo, Taylor, Simon, Foote, Kevin, Hacini-Rachinel, Feriel, Nicodeme, Edwige, Julia, Valerie
Published in Bioorganic & medicinal chemistry letters (01.03.2024)
Published in Bioorganic & medicinal chemistry letters (01.03.2024)
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Intrinsic Property Forecast Index (iPFI) as a Rule of Thumb for Medicinal Chemists to Remove a Phototoxicity Liability
Fournier, Jean-François, Bouix-Peter, Claire, Duvert, Denis, Luzy, Anne-Pascale, Ouvry, Gilles
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
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Structure-based design of Trifarotene (CD5789), a potent and selective RARγ agonist for the treatment of acne
Thoreau, Etienne, Arlabosse, Jean-Marie, Bouix-Peter, Claire, Chambon, Sandrine, Chantalat, Laurent, Daver, Sébastien, Dumais, Laurence, Duvert, Gwenaëlle, Feret, Angélique, Ouvry, Gilles, Pascau, Jonathan, Raffin, Catherine, Rodeville, Nicolas, Soulet, Catherine, Tabet, Samuel, Talano, Sandrine, Portal, Thibaud
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
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Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists
Ouvry, Gilles, Bouix-Peter, Claire, Ciesielski, Fabrice, Chantalat, Laurent, Christin, Olivier, Comino, Catherine, Duvert, Denis, Feret, Christophe, Harris, Craig S., Lamy, Laurent, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Pascau, Jonathan, Parnet, Véronique, Perrin, Agnès, Pierre, Romain, Polge, Gaëlle, Raffin, Catherine, Rival, Yves, Taquet, Nathalie, Thoreau, Etienne, Hennequin, Laurent F.
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
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Route scouting and optimization of a potent sulfoximine-based inverse agonist of RORγt
Lafitte, Guillaume, Parnet, Veronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Musicki, Branislav, Tomas, Loic, Bouix-Peter, Claire, Ouvry, Gilles, Daver, Sebastien, Arlabosse, Jean-Marie, Boiteau, Jean-Guy, Gerfaud, Thibaud, Harris, Craig S.
Published in Tetrahedron (04.10.2018)
Published in Tetrahedron (04.10.2018)
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