알파-1-항트립신 결핍증(AATD) 치료를 위한 알파-1-항트립신 조절제로서의 피롤로[2,3-F]인다졸 유도체 및 2,4,5,10-테트라아자트리시클로[7.3.0.03,7]도데카-1,3,5,8,11-펜타엔 유도체
BRODNEY MICHAEL AARON, HALL AMY B, FIMOGNARI JR. ROBERT FRANCIS, ZAKY MARIAM, NUHANT PHILIPPE MARCEL, JONES PETER, COTTRELL KEVIN MICHAEL, FANNING LEV T. D, HURLEY DENNIS JAMES, KESAVAN SARATHY, JOHNSON JR. MAC ARTHUR, GARCIA BARRANTES PEDRO MANUEL, XU JINWANG, TAPLEY TIMOTHY LEWIS, BOYD MICHAEL JOHN, THOMSON STEPHEN A, SWETT REBECCA JANE, DAMAGNEZ VERONIQUE, BOUCHER DIANE MARIE, MAXWELL JOHN PATRICK, GIROUX SIMON, GREY JR. RONALD LEE
Year of Publication 09.12.2022
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Year of Publication 09.12.2022
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알파-1-항트립신 결핍증(AATD)의 치료를 위한 알파-1-항트립신 조절제로서의 인돌 유도체
HALL AMY B, FIMOGNARI JR. ROBERT FRANCIS, TANG QING, HURLEY DENNIS JAMES, JOHNSON JR. MAC ARTHUR, BANDARAGE UPUL KEERTHI, TAPLEY TIMOTHY LEWIS, BOYD MICHAEL JOHN, ZHANG HU, DAMAGNEZ VERONIQUE, CLARK MICHAEL PHILIP, DEININGER DAVID D, MAXWELL JOHN PATRICK, BRODNEY MICHAEL AARON, NUHANT PHILIPPE MARCEL, ZAKY MARIAM, RONKIN STEVEN M, JONES PETER, COTTRELL KEVIN MICHAEL, COLLIER PHILIP NOEL, WAAL NATHAN D, FLEMING GABRIELLE SIMONE, MAXWELL BRAD, FANNING LEV T.D, ALLEN EMILY ELIZABETH, DENG HONGBO, WANG JIAN, THOMSON STEPHEN A, SWETT REBECCA JANE, BOUCHER DIANE MARIE, GIROUX SIMON
Year of Publication 14.12.2022
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Year of Publication 14.12.2022
Patent
PYRROLO[2,3-F]INDAZOLE AND 2,4,5,10-TETRAZATRICYCLO[7.3.0.03,7]DODECA-1,3(7),5,8,11-PENTAENE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, BOYD, Michael John, ZAKY, Mariam, GARCIA BARRANTES, Pedro Manuel, GREY, Jr., Ronald Lee, HURLEY, Dennis James, BOUCHER, Diane Marie, FIMOGNARI, Jr., Robert Francis, FANNING, Lev T.D, MAXWELL, John Patrick, XU, Jinwang, DAMAGNEZ, Veronique, KESAVAN, Sarathy, JOHNSON, Jr., Mac Arthur, JONES, Peter, TAPLEY, Timothy Lewis, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, NUHANT, Philippe Marcel
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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7- OR 8-HYDROXY-ISOQUINOLINE AND 7- OR 8-HYDROXY-QUINOLINE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, SENTER, Timothy J, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, CLARK, Michael Philip, FANNING, Lev T.D, MAXWELL, John Patrick, DAMAGNEZ, Veronique, STONE, Steven David, JOHNSON, Jr., Mac Arthur, JONES, Peter, TAPLEY, Timothy Lewis, DENINNO, Michael Paul, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, GALE-DAY, Zachary, TANG, Qing
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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PYRANO[4,3-B]INDOLE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, CLARK, Michael Philip, FANNING, Lev T.D, MAXWELL, John Patrick, JOHNSON, JR., Mac Arthur, DAMAGNEZ, Veronique, KESAVAN, Sarathy, JONES, Peter, TAPLEY, Timothy Lewis, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, WAAL, Nathan D, COLLIER, Philip Noel, TANG, Qing
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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PYRANO[4,3-B]L NDOLE DERIVATIVES AS ALPHA-1 -ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1 -ANTITRYPSIN DEFICIENCY (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, CLARK, Michael Philip, FANNING, Lev T.D, MAXWELL, John Patrick, JOHNSON, JR., Mac Arthur, DAMAGNEZ, Veronique, KESAVAN, Sarathy, JONES, Peter, TAPLEY, Timothy Lewis, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, WAAL, Nathan D, COLLIER, Philip Noel, TANG, Qing
Year of Publication 08.02.2023
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Year of Publication 08.02.2023
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7- OR 8-HYDROXY-ISOQUINOLINE AND 7- OR 8-HYDROXY-QUINOLINE DERIVATIVES AS ALPHA-1 -ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1 -ANTITRYPSIN DEFICIENCY (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, SENTER, Timothy J, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, CLARK, Michael Philip, FANNING, Lev T.D, MAXWELL, John Patrick, JOHNSON, JR., Mac Arthur, DAMAGNEZ, Veronique, STONE, Steven David, JONES, Peter, TAPLEY, Timothy Lewis, DENINNO, Michael Paul, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, GALE-DAY, Zachary, TANG, Qing
Year of Publication 08.02.2023
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Year of Publication 08.02.2023
Patent
1H-PYRAZOLO[4,3-G]ISOQUINOLINE AND 1H-PYRAZOLO[4,3-G]QUINOLINE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD)
ZHANG, Hu, HALL, Amy B, COTTRELL, Kevin Michael, GARCIA BARRANTES, Pedro Manuel, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, FANNING, Lev T.D, MAXWELL, John Patrick, XU, Jinwang, DAMAGNEZ, Veronique, KARNS, Alexander S, BANDARAGE, Upul Keerthi, JOHNSON, Jr., Mac Arthur, TAPLEY, Timothy Lewis, DENINNO, Michael Paul, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, GALE-DAY, Zachary, ALLEN, Emily Elizabeth, NUHANT, Philippe Marcel, LIAO, Yusheng, TANG, Qing
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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MODULATORS OF ALPHA-1 ANTITRYPSIN
MESSERSMITH, David, HALL, Amy B, COTTRELL, Kevin Michael, BOYD, Michael John, FLEMING, Gabrielle Simone, FANNING, Lev T.D, RONKIN, Steven M, WANG, Jian, MORRIS, Mark A, KESAVAN, Sarathy, JONES, Peter, SWETT, Rebecca Jane, NUHANT, Philippe Marcel, WAAL, Nathan D, COLLIER, Philip Noel, BRODNEY, Michael Aaron, HURLEY, Dennis James, BOUCHER, Diane Marie, CLARK, Michael Philip, MAXWELL, John Patrick, XU, Jinwang, DAMAGNEZ, Veronique, BANDARAGE, Upul Keerthi, JOHNSON, Jr., Mac Arthur, DENG, Hongbo, TAPLEY, Timothy Lewis, THOMSON, Stephen A, GIROUX, Simon, TANG, Qing, DANIEL, Kevin Brett
Year of Publication 26.10.2023
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Year of Publication 26.10.2023
Patent
7- or 8-hydroxy-isoquinoline and 7- or 8-hydroxy-quinoline derivatives as alpha-1 -antitrypsin modulators for treating alpha-1 -antitrypsin deficiency (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, SENTER, Timothy J, JOHNSON, JR, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, CLARK, Michael Philip, FANNING, Lev T.D, MAXWELL, John Patrick, DAMAGNEZ, Veronique, STONE, Steven David, JONES, Peter, TAPLEY, Timothy Lewis, DENINNO, Michael Paul, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, GALE-DAY, Zachary, TANG, Qing
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent
Pyrano(4,3-b)l ndole derivatives as alpha-1 -antitrypsin modulators for treating alpha-1 -antitrypsin deficiency (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, JOHNSON, JR, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, CLARK, Michael Philip, FANNING, Lev T.D, MAXWELL, John Patrick, DAMAGNEZ, Veronique, KESAVAN, Sarathy, JONES, Peter, TAPLEY, Timothy Lewis, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, WAAL, Nathan D, COLLIER, Philip Noel, TANG, Qing
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent
Pyrrolo(2,3-f)indazole and 2,4,5,10-tetrazatricyclo(7.3.0.03,7)dodeca-1,3(7),5,8,11-pentaene derivatives as alpha-1-antitrypsin modulators for treating alpha-1-antitrypsin deficiency (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, BOYD, Michael John, ZAKY, Mariam, GARCIA BARRANTES, Pedro Manuel, GREY Jr., Ronald Lee, HURLEY, Dennis James, BOUCHER, Diane Marie, MAXWELL, John Patrick, XU, Jinwang, DAMAGNEZ, Veronique, KESAVAN, Sarathy, JONES, Peter, TAPLEY, Timothy Lewis, JOHNSON, Jr, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, FANNING, Lev T. D, NUHANT, Philippe Marcel, FIMOGNARI Jr., Robert Francis
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
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1 H-PYRAZOLO[4,3-G]ISOQUINOLINE AND 1 H-PYRAZOLO[4,3-G]QUINOLINE DERIVATIVES AS ALPHA-1 -ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1 -ANTITRYPSIN DEFICIENCY (AATD)
ZHANG, Hu, HALL, Amy B, COTTRELL, Kevin Michael, GARCIA BARRANTES, Pedro Manuel, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, FANNING, Lev T.D, MAXWELL, John Patrick, XU, Jinwang, JOHNSON, JR., Mac Arthur, DAMAGNEZ, Veronique, KARNS, Alexander S, BANDARAGE, Upul Keerthi, TAPLEY, Timothy Lewis, DENINNO, Michael Paul, THOMSON, Stephen A, SWETT, Rebecca Jane, GIROUX, Simon, GALE-DAY, Zachary, ALLEN, Emily Elizabeth, NUHANT, Philippe Marcel, LIAO, Yusheng, TANG, Qing
Year of Publication 08.02.2023
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Year of Publication 08.02.2023
Patent
PYRROLO[2,3-F]INDAZOLE AND 2,4,5,10-TETRAZATRICYCLO[7.3.0.03,7]DODECA-1,3(7),5,8,11-PENTAENE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD)
HALL, Amy B, COTTRELL, Kevin Michael, BRODNEY, Michael Aaron, BOYD, Michael John, ZAKY, Mariam, GARCIA BARRANTES, Pedro Manuel, HURLEY, Dennis James, BOUCHER, Diane Marie, MAXWELL, John Patrick, FIMOGNARI, JR., Robert Francis, XU, Jinwang, JOHNSON, JR., Mac Arthur, DAMAGNEZ, Veronique, KESAVAN, Sarathy, GREY, JR., Ronald Lee, JONES, Peter, TAPLEY, Timothy Lewis, THOMSON, Stephen A, FANNING, Lev T., D, SWETT, Rebecca Jane, GIROUX, Simon, NUHANT, Philippe Marcel
Year of Publication 08.02.2023
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Year of Publication 08.02.2023
Patent
INDOLE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD)
ZHANG, Hu, HALL, Amy B, COTTRELL, Kevin Michael, ZAKY, Mariam, BOYD, Michael John, FLEMING, Gabrielle Simone, FANNING, Lev T.D, DEININGER, David D, RONKIN, Steven M, WANG, Jian, JONES, Peter, SWETT, Rebecca Jane, ALLEN, Emily Elizabeth, NUHANT, Philippe Marcel, WAAL, Nathan D, COLLIER, Philip Noel, MAXWELL, Brad, BRODNEY, Michael Aaron, HURLEY, Dennis James, BOUCHER, Diane Marie, CLARK, Michael Philip, FIMOGNARI, Jr., Robert Francis, MAXWELL, John Patrick, DAMAGNEZ, Veronique, BANDARAGE, Upul Keerthi, JOHNSON, Jr., Mac Arthur, DENG, Hongbo, TAPLEY, Timothy Lewis, THOMSON, Stephen A, GIROUX, Simon, TANG, Qing
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
Patent
1 H-pyrazolo(4,3-g)isoquinoline and 1 H-pyrazolo(4,3-g)quinoline derivatives as alpha-1 -antitrypsin modulators for treating alpha-1 -antitrypsin deficiency (AATD)
ZHANG, Hu, HALL, Amy B, COTTRELL, Kevin Michael, GARCIA BARRANTES, Pedro Manuel, HURLEY, Dennis James, GU, Wenxin, BOUCHER, Diane Marie, FANNING, Lev T.D, MAXWELL, John Patrick, XU, Jinwang, DAMAGNEZ, Veronique, KARNS, Alexander S, BANDARAGE, Upul Keerthi, TAPLEY, Timothy Lewis, DENINNO, Michael Paul, THOMSON, Stephen A, JOHNSON Jr., Mac Arthur, SWETT, Rebecca Jane, GIROUX, Simon, GALE-DAY, Zachary, ALLEN, Emily Elizabeth, NUHANT, Philippe Marcel, LIAO, Yusheng, TANG, Qing
Year of Publication 27.10.2022
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Year of Publication 27.10.2022
Patent
INDOLE DERIVATIVES AS ALPHA-1 -ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1 -ANTITRYPSIN DEFICIENCY (AATD)
ZHANG, Hu, HALL, Amy B, COTTRELL, Kevin Michael, ZAKY, Mariam, BOYD, Michael John, FLEMING, Gabrielle Simone, FANNING, Lev T.D, DEININGER, David D, RONKIN, Steven M, JOHNSON, JR., Mac Arthur, WANG, Jian, JONES, Peter, SWETT, Rebecca Jane, ALLEN, Emily Elizabeth, NUHANT, Philippe Marcel, WAAL, Nathan D, COLLIER, Philip Noel, MAXWELL, Brad, BRODNEY, Michael Aaron, HURLEY, Dennis James, BOUCHER, Diane Marie, CLARK, Michael Philip, MAXWELL, John Patrick, FIMOGNARI, JR., Robert Francis, DAMAGNEZ, Veronique, BANDARAGE, Upul Keerthi, DENG, Hongbo, TAPLEY, Timothy Lewis, THOMSON, Stephen A, GIROUX, Simon, TANG, Qing
Year of Publication 15.02.2023
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Year of Publication 15.02.2023
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SUBSTITUTED 5-HYDROXYINDOLE COMPOUNDS AS MODULATORS OF ALPHA-1 ANTITRYPSIN
MESSERSMITH, David, HALL, Amy B, COTTRELL, Kevin Michael, BOYD, Michael John, FLEMING, Gabrielle Simone, FANNING, Lev T.D, RONKIN, Steven M, JOHNSON, JR., Mac Arthur, WANG, Jian, MORRIS, Mark A, KESAVAN, Sarathy, JONES, Peter, SWETT, Rebecca Jane, NUHANT, Philippe Marcel, WAAL, Nathan D, COLLIER, Philip Noel, BRODNEY, Michael Aaron, HURLEY, Dennis James, BOUCHER, Diane Marie, CLARK, Michael Philip, MAXWELL, John Patrick, XU, Jinwang, DAMAGNEZ, Veronique, BANDARAGE, Upul Keerthi, DENG, Hongbo, TAPLEY, Timothy Lewis, THOMSON, Stephen A, GIROUX, Simon, TANG, Qing, DANIEL, Kevin Brett
Year of Publication 08.02.2023
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Year of Publication 08.02.2023
Patent
Indole derivatives as alpha-1 -antitrypsin modulators for treating alpha-1 -antitrypsin deficiency (AATD)
ZHANG, Hu, HALL, Amy B, COTTRELL, Kevin Michael, ZAKY, Mariam, BOYD, Michael John, FLEMING, Gabrielle Simone, JOHNSON, JR, FANNING, Lev T.D, DEININGER, David D, RONKIN, Steven M, WANG, Jian, JONES, Peter, FIMOGNARI, JR, SWETT, Rebecca Jane, ALLEN, Emily Elizabeth, NUHANT, Philippe Marcel, WAAL, Nathan D, COLLIER, Philip Noel, MAXWELL, Brad, BRODNEY, Michael Aaron, HURLEY, Dennis James, BOUCHER, Diane Marie, CLARK, Michael Philip, MAXWELL, John Patrick, DAMAGNEZ, Veronique, BANDARAGE, Upul Keerthi, DENG, Hongbo, TAPLEY, Timothy Lewis, THOMSON, Stephen A, GIROUX, Simon, TANG, Qing
Year of Publication 03.11.2022
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Year of Publication 03.11.2022
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Substituted 5-hydroxyindole compounds as modulators of alpha-1 antitrypsin
MESSERSMITH, David, HALL, Amy B, COTTRELL, Kevin Michael, BOYD, Michael John, FLEMING, Gabrielle Simone, RONKIN, Steven M, WANG, Jian, MORRIS, Mark A, KESAVAN, Sarathy, JONES, Peter, SWETT, Rebecca Jane, NUHANT, Philippe Marcel, WAAL, Nathan D, COLLIER, Philip Noel, BRODNEY, Michael Aaron, HURLEY, Dennis James, BOUCHER, Diane Marie, CLARK, Michael Philip, MAXWELL, John Patrick, XU, Jinwang, DAMAGNEZ, Veronique, BANDARAGE, Upul Keerthi, DENG, Hongbo, TAPLEY, Timothy Lewis, JOHNSON JR., Mac Arthur, THOMSON, Stephen A, GIROUX, Simon, FANNING, Lev T. D, TANG, Qing, DANIEL, Kevin Brett
Year of Publication 20.10.2022
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Year of Publication 20.10.2022
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