Decarboxylative Peptide Macrocyclization through Photoredox Catalysis
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Published in Angewandte Chemie International Edition (16.01.2017)
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Published in Bioorganic & medicinal chemistry letters (15.04.2006)
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
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Decarboxylative Peptide Macrocyclization through Photoredox Catalysis
McCarver, Stefan J., Qiao, Jennifer X., Carpenter, Joseph, Borzilleri, Robert M., Poss, Michael A., Eastgate, Martin D., Miller, Michael M., MacMillan, David W. C.
Published in Angewandte Chemie (16.01.2017)
Published in Angewandte Chemie (16.01.2017)
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The Discovery of Macrocyclic XIAP Antagonists from a DNA-Programmed Chemistry Library, and Their Optimization To Give Lead Compounds with in Vivo Antitumor Activity
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Development of a Stereoselective and Scalable Synthesis for the Potent Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor, BMT-297376; N‑((R)‑1-((cis)‑4-(3-(Difluoromethyl)-2-methoxypyridin-4-yl)cyclohexyl)propyl)-6-methoxynicotinamide
Nimje, Roshan Y, Kuppusamy, Prakasam, Krishnamoorthy, Suresh, Shanmugam, Yoganand, Ramasamy, Duraisamy, Manoharan, Haridhas, Arunachalam, Pirama Nayagam, Balog, Aaron, Cherney, Emily C, Zhang, Liping, Borzilleri, Robert M, Hong, Zhenqiu, Kempson, James, Rampulla, Richard R, Mathur, Arvind, Gupta, Anuradha
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Donnell, Andrew F., Zhang, Yong, Stang, Erik M., Wei, Donna D., Tebben, Andrew J., Perez, Heidi L., Schroeder, Gretchen M., Pan, Chin, Rao, Chetana, Borzilleri, Robert M., Vite, Gregory D., Gangwar, Sanjeev
Published in Bioorganic & medicinal chemistry letters (01.12.2017)
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Published in ACS medicinal chemistry letters (08.11.2018)
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Published in ACS medicinal chemistry letters (13.02.2020)
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Discovery of tetrahydroisoquinoline-based bivalent heterodimeric IAP antagonists
Kim, Kyoung Soon, Zhang, Liping, Williams, David, Perez, Heidi L., Stang, Erik, Borzilleri, Robert M., Posy, Shana, Lei, Ming, Chaudhry, Charu, Emanuel, Stuart, Talbott, Randy
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Published in Bioorganic & medicinal chemistry letters (01.11.2014)
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