Discovery of N-[4-(Quinolin-4-yloxy)phenyl]benzenesulfonamides as Novel AXL Kinase Inhibitors
Szabadkai, István, Torka, Robert, Garamvölgyi, Rita, Baska, Ferenc, Gyulavári, Pál, Boros, Sándor, Illyés, Eszter, Choidas, Axel, Ullrich, Axel, Őrfi, László
Published in Journal of medicinal chemistry (26.07.2018)
Published in Journal of medicinal chemistry (26.07.2018)
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The Novel Psychoactive Substance Cumyl-CH-MEGACLONE: Human Phase-I Metabolism, Basic Pharmacological Characterization and Comparison to Other Synthetic Cannabinoid Receptor Agonists with a γ-Carboline-1-One Core
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Published in Journal of analytical toxicology (12.03.2021)
Published in Journal of analytical toxicology (12.03.2021)
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Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH
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Published in European journal of medicinal chemistry (15.07.2019)
Published in European journal of medicinal chemistry (15.07.2019)
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Novel compounds with potent CDK9 inhibitory activity for the treatment of myeloma
Czudor, Zsófia, Balogh, Mária, Bánhegyi, Péter, Boros, Sándor, Breza, Nóra, Dobos, Judit, Fábián, Márk, Horváth, Zoltán, Illyés, Eszter, Markó, Péter, Sipos, Anna, Szántai-Kis, Csaba, Szokol, Bálint, Őrfi, László
Published in Bioorganic & medicinal chemistry letters (15.02.2018)
Published in Bioorganic & medicinal chemistry letters (15.02.2018)
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Design and synthesis of new imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrazine derivatives with antiproliferative activity against melanoma cells
Garamvölgyi, Rita, Dobos, Judit, Sipos, Anna, Boros, Sándor, Illyés, Eszter, Baska, Ferenc, Kékesi, László, Szabadkai, István, Szántai-Kis, Csaba, Kéri, György, Őrfi, László
Published in European journal of medicinal chemistry (27.01.2016)
Published in European journal of medicinal chemistry (27.01.2016)
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Active Ca2+ reabsorption in the connecting tubule
Boros, Sandor, Bindels, René J. M., Hoenderop, Joost G. J.
Published in Pflügers Archiv (01.05.2009)
Published in Pflügers Archiv (01.05.2009)
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Synthesis and characterization of amino acid substituted sunitinib analogues for the treatment of AML
Nemes, Zoltán, Takács-Novák, Krisztina, Völgyi, Gergely, Valko, Klara, Béni, Szabolcs, Horváth, Zoltán, Szokol, Bálint, Breza, Nóra, Dobos, Judit, Szántai-Kis, Csaba, Illyés, Eszter, Boros, Sándor, Kok, Robbert Jan, Őrfi, László
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
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Discovery and optimization of novel benzothiophene-3-carboxamides as highly potent inhibitors of Aurora kinases A and B
Gyulavári, Pál, Szokol, Bálint, Szabadkai, István, Brauswetter, Diána, Bánhegyi, Péter, Varga, Attila, Markó, Péter, Boros, Sándor, Illyés, Eszter, Szántai-Kis, Csaba, Krekó, Marcell, Czudor, Zsófia, Őrfi, László
Published in Bioorganic & medicinal chemistry letters (15.10.2018)
Published in Bioorganic & medicinal chemistry letters (15.10.2018)
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Novel compounds reducing IRS-1 serine phosphorylation for treatment of diabetes
Simon-Szabó, Laura, Kokas, Márton, Greff, Zoltán, Boros, Sándor, Bánhegyi, Péter, Zsákai, Lilián, Szántai-Kis, Csaba, Vantus, Tibor, Mandl, József, Bánhegyi, Gábor, Vályi-Nagy, István, Őrfi, László, Ullrich, Axel, Csala, Miklós, Kéri, György
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
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Suzuki-aza-Wittig, Suzuki-condensation and aza-Wittig-electrocyclic ring-closure tandem reactions for synthesis of fused nitrogen-containing ring systems
Krajsovszky, Gábor, Károlyházy, László, Dunkel, Petra, Boros, Sándor, Grillo, Antonino, Mátyus, Péter
Published in ARKIVOC (21.09.2011)
Published in ARKIVOC (21.09.2011)
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Unexpected transformations of an azoxyquinoxaline
Hermecz, István, Molnár, Annamária, Boros, Sándor, Simon, Kálmán, Gönczi, Csaba
Published in ARKIVOC (02.08.2010)
Published in ARKIVOC (02.08.2010)
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Site-specific transamidation and deamidation of the small heat-shock protein Hsp20 by tissue transglutaminase
Boros, Sandor, Åhrman, Emma, Wunderink, Lisa, Kamps, Bram, de Jong, Wilfried W., Boelens, Wilbert C., Emanuelsson, Cecilia Sundby
Published in Proteins, structure, function, and bioinformatics (01.03.2006)
Published in Proteins, structure, function, and bioinformatics (01.03.2006)
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A novel and convenient method for the preparation of 5-(diphenylmethylene)-1H-pyrrol-2(5H)-ones; synthesis and mechanistic study
Faigl, Ferenc, Deák, Szilvia, Mucsi, Zoltán, Hergert, Tamás, Balázs, László, Sándor, Boros, Balázs, Barbara, Holczbauer, Tamás, Nyerges, Miklós, Mátravölgyi, Béla
Published in Tetrahedron (01.09.2016)
Published in Tetrahedron (01.09.2016)
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A novel and convenient method for the preparation of 5-(diphenylmethylene)-1 H -pyrrol-2(5 H )-ones; synthesis and mechanistic study
Faigl, Ferenc, Deák, Szilvia, Mucsi, Zoltán, Hergert, Tamás, Balázs, László, Sándor, Boros, Balázs, Barbara, Holczbauer, Tamás, Nyerges, Miklós, Mátravölgyi, Béla
Published in Tetrahedron (01.09.2016)
Published in Tetrahedron (01.09.2016)
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Reductive transformations of unsaturated azabicyclic nitrolactams
Pilipecz, Mihály Viktor, Varga, Tamás Róbert, Scheiber, Pál, Mucsi, Zoltán, Fàvre-Mourgues, Amélie, Boros, Sándor, Balázs, László, Tóth, Gábor, Nemes, Péter
Published in Tetrahedron (08.07.2012)
Published in Tetrahedron (08.07.2012)
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Dioxirane Oxidation of 3-Arylideneflavanones: Diastereoselective Formation of trans,trans Spiroepoxides from the E Isomers
Nemes, Csaba, Levai, Albert, Patonay, Tamas, Toth, Gabor, Boros, Sandor, Halasz, Judit, Adam, Waldemar, Golsch, Dieter
Published in Journal of organic chemistry (01.02.1994)
Published in Journal of organic chemistry (01.02.1994)
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