A potent and selective metabotropic glutamate receptor 4 positive allosteric modulator improves movement in rodent models of Parkinson's disease
Le Poul, Emmanuel, Boléa, Christelle, Girard, Francoise, Poli, Sonia, Charvin, Delphine, Campo, Brice, Bortoli, Julien, Bessif, Abdhelak, Luo, Bin, Koser, Amy Jo, Hodge, Lisa M, Smith, Karen M, DiLella, Anthony G, Liverton, Nigel, Hess, Fred, Browne, Susan E, Reynolds, Ian J
Published in The Journal of pharmacology and experimental therapeutics (01.10.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2012)
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Characterization of the novel positive allosteric modulator of the metabotropic glutamate receptor 4 ADX88178 in rodent models of neuropsychiatric disorders
Kalinichev, Mikhail, Le Poul, Emmanuel, Boléa, Christelle, Girard, Françoise, Campo, Brice, Fonsi, Massimiliano, Royer-Urios, Isabelle, Browne, Susan E, Uslaner, Jason M, Davis, Matthew J, Raber, Jacob, Duvoisin, Robert, Bate, Simon T, Reynolds, Ian J, Poli, Sonia, Celanire, Sylvain
Published in The Journal of pharmacology and experimental therapeutics (01.09.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2014)
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mGluR5 negative allosteric modulators overview: a medicinal chemistry approach towards a series of novel therapeutic agents
Rocher, Jean-Philippe, Bonnet, Béatrice, Boléa, Christelle, Lütjens, Robert, Le Poul, Emmanuel, Poli, Sonia, Epping-Jordan, Mark, Bessis, Anne-Sophie, Ludwig, Bernard, Mutel, Vincent
Published in Current topics in medicinal chemistry (01.03.2011)
Published in Current topics in medicinal chemistry (01.03.2011)
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Effect of the Metabotropic Glutamate Receptor Type 5 Negative Allosteric Modulator Dipraglurant on Motor and Non-Motor Symptoms of Parkinson's Disease
Epping-Jordan, Mark P, Girard, Françoise, Bessis, Anne-Sophie, Mutel, Vincent, Boléa, Christelle, Derouet, Francis, Bessif, Abdelhak, Mingard, Brice, Barbier, Stéphanie, Paradis, Justine S, Rocher, Jean-Philippe, Lütjens, Robert, Kalinichev, Mikhail, Poli, Sonia
Published in Cells (Basel, Switzerland) (24.03.2023)
Published in Cells (Basel, Switzerland) (24.03.2023)
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Discovery of 1,5-Disubstituted Pyridones: A New Class of Positive Allosteric Modulators of the Metabotropic Glutamate 2 Receptor
Cid, Jose María, Duvey, Guillaume, Cluzeau, Philippe, Nhem, Vanthea, Macary, Karim, Raux, Alexandre, Poirier, Nicolas, Muller, Jessica, Boléa, Christelle, Finn, Terry, Poli, Sonia, Epping-Jordan, Mark, Chamelot, Emilie, Derouet, Francis, Girard, Francoise, Macdonald, Gregor J, Vega, Juan Antonio, de Lucas, Ana Isabel, Matesanz, Encarnación, Lavreysen, Hilde, Linares, María Lourdes, Oehlrich, Daniel, Oyarzábal, Julen, Tresadern, Gary, Trabanco, Andrés A, Andrés, Jose Ignacio, Le Poul, Emmanuel, Imogai, Hassan, Lutjens, Robert, Rocher, Jean-Philippe
Published in ACS chemical neuroscience (15.12.2010)
Published in ACS chemical neuroscience (15.12.2010)
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Development of new camphor based N,S chiral ligands and their application in transfer hydrogenationElectronic supplementary information (ESI) available: 13C NMR spectra. See http://www.rsc.org/suppdata/ob/b4/b402805h
Gayet, Arnaud, Bolea, Christelle, Andersson, Pher G.
Published in Organic & biomolecular chemistry (28.06.2004)
Published in Organic & biomolecular chemistry (28.06.2004)
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