Changing for the Better: Discovery of the Highly Potent and Selective CDK9 Inhibitor VIP152 Suitable for Once Weekly Intravenous Dosing for the Treatment of Cancer
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Published in Journal of medicinal chemistry (12.08.2021)
Published in Journal of medicinal chemistry (12.08.2021)
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A Novel NAMPT Inhibitor-Based Antibody–Drug Conjugate Payload Class for Cancer Therapy
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Published in Bioconjugate chemistry (15.06.2022)
Published in Bioconjugate chemistry (15.06.2022)
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Radiofluorinated Derivatives of 2‑(Phosphonomethyl)pentanedioic Acid as Inhibitors of Prostate Specific Membrane Antigen (PSMA) for the Imaging of Prostate Cancer
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Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
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Preclinical evaluation of BAY 1075553, a novel super(18)F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer
Lesche, Ralf, Kettschau, Georg, Gromov, Alexey V, Bohnke, Niels, Borkowski, Sandra, Monning, Ursula, Hegele-Hartung, Christa, Dohr, Olaf, Dinkelborg, Ludger M, Graham, Keith
Published in European journal of nuclear medicine and molecular imaging (01.01.2014)
Published in European journal of nuclear medicine and molecular imaging (01.01.2014)
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Preparation of (2R)-2-acetoxy-D-forosamine for the total synthesis of spinosyns
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Discovery of potent SOS1 inhibitors that block RAS activation via disruption of the RAS–SOS1 interaction
Hillig, Roman C., Sautier, Brice, Schroeder, Jens, Moosmayer, Dieter, Hilpmann, André, Stegmanna, Christian M., Werbeck, Nicolas D., Briem, Hans, Boemer, Ulf, Weiske, Joerg, Badock, Volker, Mastouri, Julia, Petersen, Kirstin, Siemeister, Gerhard, Kahmann, Jan D., Wegener, Dennis, Böhnke, Niels, Eis, Knut, Graham, Keith, Wortmann, Lars, von Nussbaum, Franz, Bader, Benjamin
Published in Proceedings of the National Academy of Sciences - PNAS (12.02.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (12.02.2019)
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Mono- and multimeric PSMA-targeting small molecule-thorium-227 conjugates for optimized efficacy and biodistribution in preclinical models
Böhnke, Niels, Indrevoll, Bård, Hammer, Stefanie, Papple, Alex, Kristian, Alexander, Briem, Hans, Celik, Arif, Mumberg, Dominik, Cuthbertson, Alan, Zitzmann-Kolbe, Sabine
Published in European journal of nuclear medicine and molecular imaging (01.02.2024)
Published in European journal of nuclear medicine and molecular imaging (01.02.2024)
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Abstract 2907: Identification and optimization of a novel NAMPT inhibitor-based ADC payload class for cancer therapy
Böhnke, Niels, Berger, Markus, Griebenow, Nils, Giese, Anja, Günther, Judith, Sommer, Anette, Hammer, Stefanie, Berndt, Sandra, Wengner, Antje M., Beier, Rudolf, Stelte-Ludwig, Beatrix, Mahlert, Christoph, Greven, Simone, Dietz, Lisa, Joerissen, Hannah, Rottmann, Antje, Erkelenz, Michael, Barak, Naomi, Bömer, Ulf, Mumber, Dominik, Kreft, Bertolt, Linden, Lars, Nising, Carl Friedrich, Weinmann, Hilmar
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Preclinical evaluation of BAY 1075553, a novel (18)F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer
Lesche, Ralf, Kettschau, Georg, Gromov, Alexey V, Böhnke, Niels, Borkowski, Sandra, Mönning, Ursula, Hegele-Hartung, Christa, Döhr, Olaf, Dinkelborg, Ludger M, Graham, Keith
Published in European journal of nuclear medicine and molecular imaging (01.01.2014)
Published in European journal of nuclear medicine and molecular imaging (01.01.2014)
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Journal Article
Preclinical evaluation of BAY 1075553, a novel 18F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer
Lesche, Ralf, Kettschau, Georg, Gromov, Alexey V., Böhnke, Niels, Borkowski, Sandra, Mönning, Ursula, Hegele-Hartung, Christa, Döhr, Olaf, Dinkelborg, Ludger M., Graham, Keith
Published in European journal of nuclear medicine and molecular imaging (2014)
Published in European journal of nuclear medicine and molecular imaging (2014)
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Tietze, Lutz F., Dietz, Simone, Böhnke, Niels, Düfert, M. Alexander, Objartel, Ina, Stalke, Dietmar
Published in European Journal of Organic Chemistry (01.11.2011)
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Book Review
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2-((2-(PHENYLOXYMETHYL)PYRIDIN-5-YL)OXY)-ETHANAMIN-DERIVATIVES AND RELATED COMPOUNDS AS PESTICIDES E.G. FOR CROP PROTECTION
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Year of Publication 28.10.2022
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Year of Publication 28.10.2022
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Year of Publication 14.03.2024
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Year of Publication 07.03.2023
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Year of Publication 07.03.2023
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TURBERG, ANDREAS, HORSTMANN, SEBASTIAN, SCHWARZ, HANS-GEORG, HARSCHNECK, TOBIAS, GORGENS, ULRICH, BOHNKE, NIELS, MAUE, MICHAEL, VELTEN, ROBERT, HAHN, JULIA JOHANNA, HALLENBACH, WERNER, ILG, KERSTIN, KOBBERLING, JOHANNES
Year of Publication 28.02.2023
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Year of Publication 28.02.2023
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Year of Publication 20.07.2021
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Year of Publication 20.07.2021
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5-FLUORO-N-(PYRIDIN-2-YL)PYRIDIN-2-AMINE DERIVATIVES CONTAINING A SULFONE GROUP
LIENAU, PHILIP, SIEMEISTER, GERHARD, BOHLMANN, ROLF, SCHOLZ, ARNE, BOMER, ULF, BOHNKE, NIELS, KOSEMUND, DIRK, LUCKING, ULRICH, ZORN, LUDWIG
Year of Publication 08.06.2021
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