Search Results - "BOCK M G" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists

Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists

by Evans, B. E, Rittle, K. E, Bock, M. G, DiPardo, R. M, Freidinger, R. M, Whitter, W. L, Lundell, G. F, Veber, D. F, Anderson, P. S, Chang, R. S. L, Lotti, V. J, Cerino, D. J, Chen, T. B, Kling, P. J, Kunkel, K. A, Springer, J. P, Hirshfield, J
Published in Journal of medicinal chemistry (01.12.1988)

Get full text

Journal Article

Design of Potent, Orally Effective, Nonpeptidal Antagonists of the Peptide Hormone Cholecystokinin

Design of Potent, Orally Effective, Nonpeptidal Antagonists of the Peptide Hormone Cholecystokinin

by Evans, Ben E., Bock, Mark G., Rittle, Kenneth E., DiPardo, Robert M., Whitter, Willie L., Veber, Daniel F., Anderson, Paul S., Freidinger, Roger M.
Published in Proceedings of the National Academy of Sciences - PNAS (01.07.1986)

Get full text

Journal Article

Bradykinin antagonists: new opportunities

Bradykinin antagonists: new opportunities

by Bock, Mark G, Longmore, Jeanette
Published in Current Opinion in Chemical Biology (01.08.2000)

Get full text

Book Review Journal Article

Characterization of the binding of [3H]L-365,260: a new potent and selective brain cholecystokinin (CCK-B) and gastrin receptor antagonist radioligand

Characterization of the binding of [3H]L-365,260: a new potent and selective brain cholecystokinin (CCK-B) and gastrin receptor antagonist radioligand

by CHANG, R. S. L, CHEN, T. B, BOCK, M. G, FREIDINGER, R. M, CHEN, R, ROSEGAY, A, LOTTI, V. J
Published in Molecular pharmacology (01.06.1989)

Get full text

Journal Article

Benzodiazepine gastrin and brain cholecystokinin receptor ligands; L-365,260

Benzodiazepine gastrin and brain cholecystokinin receptor ligands; L-365,260

by Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Veber, Daniel F, Anderson, Paul S, Freidinger, Roger M
Published in Journal of medicinal chemistry (01.01.1989)

Get full text

Journal Article

Development of 1,4-benzodiazepine cholecystokinin type B antagonists

Development of 1,4-benzodiazepine cholecystokinin type B antagonists

by Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Garsky, Victor M, Gilbert, Kevin F, Leighton, James L, Carson, Kenneth L
Published in Journal of medicinal chemistry (24.12.1993)

Get full text

Journal Article

Design of nonpeptidal ligands for a peptide receptor: cholecystokinin antagonists

Design of nonpeptidal ligands for a peptide receptor: cholecystokinin antagonists

by Evans, B. E, Rittle, K. E, Bock, M. G, DiPardo, R. M, Freidinger, R. M, Whitter, W. L, Gould, N. P, Lundell, G. F, Homnick, C. F
Published in Journal of medicinal chemistry (01.07.1987)

Get full text

Journal Article

Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus

Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus

by Kuo, Michelle S., Bock, Mark G., Freidinger, Roger M., Guidotti, Maribeth T., Lis, Edward V., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Williams, Peter D., Woyden, Carla J.
Published in Bioorganic & medicinal chemistry letters (03.11.1998)

Get full text

Journal Article

In vitro pharmacological profile of a novel structural class of oxytocin antagonists

by PETTIBONE, D. J, CLINESCHMIDT, B. V, WILLIAMS, P. D, LOWENSOHN, R. I, LIS, E. V, REISS, D. R, TOTARO, J. A, WOYDEN, C. J, BOCK, M. G, FREIDINGER, R. M, TUNG, R. D, VEBER, D. F
Published in The Journal of pharmacology and experimental therapeutics (01.01.1991)

Get full text

Journal Article

Antagonism of oxytocin in rats and pregnant rhesus monkeys by the novel cyclic hexapeptides, L-366,682 and L-366,948

Antagonism of oxytocin in rats and pregnant rhesus monkeys by the novel cyclic hexapeptides, L-366,682 and L-366,948

by CLINESCHMIDT, B. V, PETTIBONE, D. J, FREIDINGER, R. M, VEBER, D. F, WILLIAMS, P. D, REISS, D. R, LIS, E. V, HALUSKA, G. J, NOVY, M. J, COOK, M. J, CUKIERSKI, M. A, KAUFMAN, M. J, BOCK, M. G
Published in The Journal of pharmacology and experimental therapeutics (01.03.1991)

Get full text

Journal Article

Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product

Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product

by Williams, Peter D, Bock, Mark G, Tung, Roger D, Garsky, Victor M, Perlow, Debra S, Erb, Jill M, Lundell, G. F, Gould, Norman P, Whitter, Willie L
Published in Journal of medicinal chemistry (01.10.1992)

Get full text

Journal Article

Cyclic hexapeptide oxytocin antagonists. Potency-, selectivity-, and solubility-enhancing modifications

Cyclic hexapeptide oxytocin antagonists. Potency-, selectivity-, and solubility-enhancing modifications

by Freidinger, Roger M, Williams, P. D, Tung, R. D, Bock, M. G, Pettibone, D. J, Clineschmidt, B. V, DiPardo, R. M, Erb, J. M, Garsky, V. M
Published in Journal of medicinal chemistry (01.07.1990)

Get full text

Journal Article

Receptor ligands which bind the oxytocin receptor with selectivity and high affinity. Chemical modification of a Streptomyces silvensis derived cyclic hexapeptide

Receptor ligands which bind the oxytocin receptor with selectivity and high affinity. Chemical modification of a Streptomyces silvensis derived cyclic hexapeptide

by Bock, Mark G, DiPardo, R. M, Williams, P. D, Pettibone, D. J, Clineschmidt, B. V, Ball, R. G, Veber, D. F, Freidinger, R. M
Published in Journal of medicinal chemistry (01.09.1990)

Get full text

Journal Article

Renin inhibitors containing hydrophilic groups. Tetrapeptides with enhanced aqueous solubility and nanomolar potency

Renin inhibitors containing hydrophilic groups. Tetrapeptides with enhanced aqueous solubility and nanomolar potency

by Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Freidinger, Roger M, Rittle, Kenneth E, Payne, Linda S, Boger, Joshua, Whitter, Willie L, LaMont, Bruce I
Published in Journal of medicinal chemistry (01.10.1988)

Get full text

Journal Article

Cholecystokinin-A receptor ligands based on the .kappa.-opioid agonist tifluadom

Cholecystokinin-A receptor ligands based on the .kappa.-opioid agonist tifluadom

by Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Veber, Daniel F, Freidinger, Roger M, Chang, Raymond S. L, Chen, T. B, Lotti, Victor J
Published in Journal of medicinal chemistry (01.01.1990)

Get full text

Journal Article

Development and pharmacological assessment of novel peptide and nonpeptide oxytocin antagonists

Development and pharmacological assessment of novel peptide and nonpeptide oxytocin antagonists

by Pettibone, Douglas J., Clineschmidt, Bradley V., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Veber, Daniel F., Williams, Peter D.
Published in Regulatory peptides (29.04.1993)

Get full text

Journal Article Conference Proceeding

Cholecystokinin antagonists. Synthesis and biological evaluation of 3-substituted 1,4-benzodiazepin-2-amines

Cholecystokinin antagonists. Synthesis and biological evaluation of 3-substituted 1,4-benzodiazepin-2-amines

by Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Freidinger, Roger M, Chang, Raymond S. L, Lotti, Victor J
Published in Journal of medicinal chemistry (01.01.1988)

Get full text

Journal Article

Discovery of a Novel, Selective, and Orally Bioavailable Class of Thrombin Inhibitors Incorporating Aminopyridyl Moieties at the P1 Position

Discovery of a Novel, Selective, and Orally Bioavailable Class of Thrombin Inhibitors Incorporating Aminopyridyl Moieties at the P1 Position

by Feng, Dong-Mei, Gardell, Stephen J, Lewis, S. Dale, Bock, Mark G, Chen, Zhongguo, Freidinger, Roger M, Naylor-Olsen, Adel M, Ramjit, Harri G, Woltmann, Richard, Baskin, Elizabeth P, Lynch, Joseph J, Lucas, Robert, Shafer, Jules A, Dancheck, Kimberley B, Chen, I-Wu, Mao, Shi-Shan, Krueger, Julie A, Hare, Timothy R, Mulichak, Anne M, Vacca, Joseph P
Published in Journal of medicinal chemistry (07.11.1997)

Get full text

Journal Article

Cholecystokinin antagonists. Synthesis and biological evaluation of 4-substituted 4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepines

Cholecystokinin antagonists. Synthesis and biological evaluation of 4-substituted 4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepines

by Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Veber, Daniel F, Freidinger, Roger M, Chang, Raymond S. L, Lotti, Victor J
Published in Journal of medicinal chemistry (01.01.1988)

Get full text

Journal Article

Cholecystokinin antagonists. Synthesis of asperlicin analogs with improved potency and water solubility

Cholecystokinin antagonists. Synthesis of asperlicin analogs with improved potency and water solubility

by Bock, Mark G, DiPardo, Robert M, Rittle, Kenneth E, Evans, Ben E, Freidinger, Roger M, Veber, Daniel F, Chang, Raymond S. L, Chen, Tsing Bau, Keegan, Maureen E, Lotti, Victor J
Published in Journal of medicinal chemistry (01.10.1986)

Get full text

Journal Article

1
2
3
4
5
6
Next
[6]