A second generation of non-peptide cholecystokinin receptor antagonists and their possible therapeutic potential
Freedman, S B, Patel, S, Smith, A J, Chapman, K, Fletcher, A, Kemp, J A, Marshall, G R, Hargreaves, R J, Scholey, K, Mellin, E C
Published in Annals of the New York Academy of Sciences (01.03.1994)
Published in Annals of the New York Academy of Sciences (01.03.1994)
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1-((7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo [2.2.1]-heptan-1(S)-yl)methyl)sulfonyl)-4-(2-methylphenyl)piperaz ine (L-368,899): an orally bioavailable, non-peptide oxytocin antagonist with potential utility for managing preterm labor
Williams, P D, Anderson, P S, Ball, R G, Bock, M G, Carroll, L, Chiu, S H, Clineschmidt, B V, Culberson, J C, Erb, J M, Evans, B E
Published in Journal of medicinal chemistry (04.03.1994)
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Published in Journal of medicinal chemistry (04.03.1994)
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Second-generation benzodiazepine CCK-B antagonists. Development of subnanomolecular analogs with selectivity and water solubility
BOCK, M. G, DIPARDO, R. M, FLETCHER, A. E, CHAPMAN, K. L, ANDERSON, P. S, FREIDINGER, R. M, MELLIN, E. C, NEWTON, R. C, VEBER, D. F, FREEDMAN, S. B, SMITH, A. J, SMITA PATEL, KEMP, J. A, MARSHALL, G. R
Published in Journal of medicinal chemistry (1994)
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Published in Journal of medicinal chemistry (1994)
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Progress in the development of oxytocin antagonists for use in preterm labor
Pettibone, D J, Guidotti, M, Harrell, C M, Jasper, J R, Lis, E V, O'Brien, J A, Reiss, D R, Woyden, C J, Bock, M G, Evans, B E
Published in Advances in experimental medicine and biology (1995)
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Published in Advances in experimental medicine and biology (1995)
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1-7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo[2.2.1]-heptan-1(S)-ylmethylsulfonyl-4-(2-methylphenyl)piperazine (L-368,899) : an orally bioavailable, non-peptide oxytocin antagonist with potential utility for managing preterm labor
WILLIAMS, P. D, ANDERSON, P. S, FITZPATRICK, S. L, FREIDINGER, R. M, KAUFMAN, M. J, LUNDELL, G. F, MURPHY, J. S, PAWLUCZYK, J. M, PERLOW, D. S, PETTIBONE, D. J, PITZENBERGER, S. M, THOMPSON, K. L, BALL, R. G, VEBER, D. F, BOCK, M. G, CARROLL, L.-A, SHUET-HING LEE CHIU, CLINESCHMIDT, B. V, CULBERSON, J. C, ERB, J. M, EVANS, B. E
Published in Journal of medicinal chemistry (1994)
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Published in Journal of medicinal chemistry (1994)
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Characterization of the binding of ( super(3)H)L-365,260: A new potent and selective brain cholecystokinin (CCK-B) and gastrin receptor antagonist radioligand
Chang, RSL, Chen, T B, Bock, M G, Freidinger, R M, Chen, R, Rosegay, A, Lotti, V J
Published in Molecular pharmacology (01.01.1989)
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Published in Molecular pharmacology (01.01.1989)
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NANOMOLAR-AFFINITY, NONPEPTIDE OXYTOCIN RECEPTOR ANTAGONISTS
EVANS, BE, LUNDELL, GF, GILBERT, KF, BOCK, MG, RITTLE, KE, CARROLL, LA, WILLIAMS, PD, PAWLUCZYK, JM, LEIGHTON, JL, YOUNG, MB, ERB, JM, HOBBS, DW, GOULD, NP, DIPARDO, RM, HOFFMAN, JB, PERLOW, DS, WHITTER, WL, VEBER, DF, PETTIBONE, DJ, CLINESCHMIDT, BV, ANDERSON, PS, FREIDINGER, RM
Published in Journal of medicinal chemistry (10.12.1993)
Published in Journal of medicinal chemistry (10.12.1993)
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Dipetide analogues. Synthesis of a potent renin inhibitor
Bock, M G, DiPardo, R M, Evans, B E, Rittle, KE, Boger, J S, Freidinger, R M, Veber, D F
Published in Journal of the Chemical Society. Chemical communications (01.01.1985)
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Published in Journal of the Chemical Society. Chemical communications (01.01.1985)
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Total synthesis of (.+-.)-N-methylmaysenine
Corey, E. J, Weigel, Leland O, Floyd, David, Bock, Mark G
Published in Journal of the American Chemical Society (01.04.1978)
Published in Journal of the American Chemical Society (01.04.1978)
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Theoretical estimation of pKa values of pyrazinylguanidine derivatives
Bock, Mark G, Schlegel, H. Bernard, Smith, Graham M
Published in Journal of organic chemistry (01.04.1981)
Published in Journal of organic chemistry (01.04.1981)
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