Homocamptothecins: Synthesis and Antitumor Activity of Novel E-Ring-Modified Camptothecin Analogues
Lavergne, Olivier, Lesueur-Ginot, Laurence, Pla Rodas, Francesc, Kasprzyk, Philip G, Pommier, Jacques, Demarquay, Danièle, Prévost, Grégoire, Ulibarri, Gérard, Rolland, Alain, Schiano-Liberatore, Anne-Marie, Harnett, Jeremiah, Pons, Dominique, Camara, José, Bigg, Dennis C. H
Published in Journal of medicinal chemistry (31.12.1998)
Published in Journal of medicinal chemistry (31.12.1998)
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Homocamptothecin, an E-ring modified camptothecin with enhanced lactone stability, retains topoisomerase I-targeted activity and antitumor properties
LESUEUR-GINOT, L, DEMARQUAY, D, KISS, R, KASPRZYK, P. G, DASSONNEVILLE, L, BAILLY, C, CAMARA, J, LAVERGNE, O, BIGG, D. C. H
Published in Cancer research (Chicago, Ill.) (15.06.1999)
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Published in Cancer research (Chicago, Ill.) (15.06.1999)
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Topoisomerase I-Mediated Antiproliferative Activity of Enantiomerically Pure Fluorinated Homocamptothecins
Lavergne, Olivier, Demarquay, Danièle, Bailly, Christian, Lanco, Christophe, Rolland, Alain, Huchet, Marion, Coulomb, Helène, Muller, Nicole, Baroggi, Nicole, Camara, José, Le Breton, Christine, Manginot, Eric, Cazaux, Jean-Bernard, Bigg, Dennis C. H
Published in Journal of medicinal chemistry (01.06.2000)
Published in Journal of medicinal chemistry (01.06.2000)
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BN 80927: A novel homocamptothecin with inhibitory activities on both topoisomerase I and topoisomerase II
Lavergne, Olivier, Harnett, Jeremiah, Rolland, Alain, Lanco, Christophe, Lesueur-Ginot, Laurence, Demarquay, Danièle, Huchet, Marion, Coulomb, Hélène, Bigg, Dennis C.H.
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
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Homocamptothecin, an E-Ring-modified Camptothecin, Exerts More Potent Antiproliferative Activity than Other Topoisomerase I Inhibitors in Human Colon Cancers Obtained from Surgery and Maintained in Vitro under Histotypical Culture Conditions
PHILIPPART, P, HARPER, L, MENDES DA COSTA, P, KISS, R, CHABOTEAUX, C, DECAESTECKER, C, BRONCKART, Y, GORDOVER, L, LESUEUR-GINOT, L, MALONNE, H, LAVERGNE, O, BIGG, D. C. H
Published in Clinical cancer research (01.04.2000)
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Published in Clinical cancer research (01.04.2000)
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Chiral resolution of enantiomers of homocamptothecin derivatives, antitumor topoisomerase I inhibitors, using high performance liquid chromatography on polysaccharide-based chiral stationary phases
GOOSSENS, J. F, FOULON, C, BAILLY, C, BIGG, D. C. H, BONTE, J. P, VACCHER, C
Published in Chromatographia (01.03.2004)
Published in Chromatographia (01.03.2004)
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Aluminum Chloride-Promoted Aminolysis of N-Tosyl Lactams
Bon, Eric, Biggs, Dennis C. H, Bertrand, Guy, Bigg, Dennis C. H
Published in Journal of organic chemistry (01.04.1994)
Published in Journal of organic chemistry (01.04.1994)
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Flexible 1-[(2-Aminoethoxy)alkyl]-3-ar(o)yl(thio)ureas as Novel Acetylcholinesterase Inhibitors. Synthesis and Biochemical Evaluation
Vidaluc, Jean-Louis, Calmel, Francis, Bigg, Dennis C. H, Carilla, Elisabeth, Briley, Mike
Published in Journal of medicinal chemistry (21.07.1995)
Published in Journal of medicinal chemistry (21.07.1995)
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