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Wéber, Csaba, Bielik, Attila, Szendrei, Györgyi I, Greiner, István
Published in Tetrahedron letters (15.04.2002)
Published in Tetrahedron letters (15.04.2002)
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Identification of nitric oxide donors by biomimetic HTS application
Balogh, György T, Dalmadi, Balázs, Bielik, Attila, Keserü, György M
Published in Combinatorial chemistry & high throughput screening (01.06.2005)
Published in Combinatorial chemistry & high throughput screening (01.06.2005)
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Discovery and Preclinical Characterization of 3‑((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications
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Published in Journal of medicinal chemistry (23.03.2017)
Published in Journal of medicinal chemistry (23.03.2017)
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Journal Article
Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators
Galambos, János, Bielik, Attila, Wágner, Gábor, Domány, György, Kóti, János, Béni, Zoltán, Szigetvári, Áron, Sánta, Zsuzsanna, Orgován, Zoltán, Bobok, Amrita, Kiss, Béla, Mikó-Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Krasavin, Mikhail, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M.
Published in European journal of medicinal chemistry (16.06.2017)
Published in European journal of medicinal chemistry (16.06.2017)
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Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs
Wágner, Gábor, Wéber, Csaba, Nyéki, Olga, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
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Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists
Galambos, János, Wágner, Gábor, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Gyertyán, István, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Corrigendum to “Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs” [Bioorg. Med. Chem. Lett. 20 (2010) 3737–3741]
Wágner, Gábor, Wéber, Csaba, Nyéki, Olga, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
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Journal Article
Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluRS NAMs
WAGNER, Gábor, WEBER, Csaba, NAGY, József, KURKO, Dalma, GAL, Krisztina, GREINER, István, SZOMBATHELYI, Zsolt, KESERU, György M, DOMANY, György, NYEKI, Olga, NOGRADI, Katalin, BIELIK, Attila, MOLNAR, László, BOBOK, Amrita, HORVATH, Attila, KISS, Béla, KOLOK, Sándor
Published in Bioorganic & medicinal chemistry letters (2010)
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Published in Bioorganic & medicinal chemistry letters (2010)
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Novel sulfonamides having dual dopamine D2 and D3 receptor affinity show in vivo antipsychotic efficacy with beneficial cognitive and EPS profile
Ágai-Csongor, Éva, Nógrádi, Katalin, Galambos, János, Vágó, István, Bielik, Attila, Magdó, Ildikó, Ignácz-Szendrei, Györgyi, Keserű, György Miklós, Greiner, István, Laszlovszky, István, Béla Kiss, Éva Schmidt, Judit Laszy, Katalin Sághy, Gyertyán, István, Zájer-Balázs, Mária, Gémesi, Larisza, Domány, György
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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Solid-phase synthesis of 6-hydroxy-2,4-diaminoquinazolines
Wéber, Csaba, Bielik, Attila, Demeter, Ádám, Borza, István, Szendrei, Györgyi I., Keserű, György M., Greiner, István
Published in Tetrahedron (26.09.2005)
Published in Tetrahedron (26.09.2005)
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Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists
BORZA, Istvan, KOLOK, Sandor, BIELIK, Attila, NAGY, Jozsef, FARKAS, Sandor, DOMANY, György, GERE, Aniko, AGAI-CSONGOR, Eva, AGAI, Béla, TARKANYI, Gabor, HORVATH, Csilla, BARTA-SZALAI, Gizella, BOZO, Eva, KISS, Csilla
Published in Bioorganic & medicinal chemistry letters (03.11.2003)
Published in Bioorganic & medicinal chemistry letters (03.11.2003)
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Scheduling a Flexible, Open-Architecture Robotic Workstation under LabWindows
Bánki, Zsolt, Báthor, Miklós, Molnár, László, Bielik, Attila, Keserű, György M.
Published in Journal of Laboratory Automation (01.06.2005)
Published in Journal of Laboratory Automation (01.06.2005)
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Year of Publication 30.04.2014
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Year of Publication 28.07.2011
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Year of Publication 28.07.2011
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Year of Publication 15.09.2010
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DOMANY GYORGY, BARTANE SZALAI GIZELLA, BIELIK ATTILA, KOVACSNE BOZO EVA, FARKAS SANDOR, BORZA ISTVAN, IGNACZNE SZENDREI GYORGYI, KOLOK SANDOR, NAGY JOZSEF, VAGO ISTVAN, HORVATH CSILLA, KESERU GYORGYI
Year of Publication 06.07.2011
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Year of Publication 06.07.2011
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Year of Publication 03.09.2008
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Year of Publication 03.09.2008
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