Design of Selective and Soluble Inhibitors of Tumor Necrosis Factor-α Converting Enzyme (TACE)
Rabinowitz, Michael H, Andrews, Robert C, Becherer, J. David, Bickett, D. Mark, Bubacz, Dulce G, Conway, James G, Cowan, David J, Gaul, Micheal, Glennon, Kimberly, Lambert, Millard H, Leesnitzer, M. Anthony, McDougald, Darryl L, Moss, Marcia L, Musso, David L, Rizzolio, Michele C
Published in Journal of medicinal chemistry (22.11.2001)
Published in Journal of medicinal chemistry (22.11.2001)
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A High Throughput Fluorogenic Substrate for Interstitial Collagenase (MMP-1) and Gelatinase (MMP-9)
Bickett, D.M., Green, M.D., Berman, J., Dezube, M., Howe, A.S., Brown, P.J., Roth, J.T., Mcgeehan, G.M.
Published in Analytical biochemistry (01.07.1993)
Published in Analytical biochemistry (01.07.1993)
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Structural features and biochemical properties of TNF- α converting enzyme (TACE)
Moss, M.L., Jin, S.-L.C., Becherer, J.D., Bickett, D.M., Burkhart, W., Chen, W.-J., Hassler, D., Leesnitzer, M.T., McGeehan, G., Milla, M., Moyer, M., Rocque, W., Seaton, T., Schoenen, F., Warner, J., Willard, D.
Published in Journal of neuroimmunology (01.02.1997)
Published in Journal of neuroimmunology (01.02.1997)
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Metalloproteinase inhibitors for the disintegrin-like metalloproteinases ADAM10 and ADAM17 that differentially block constitutive and phorbol ester-inducible shedding of cell surface molecules
Ludwig, Andreas, Hundhausen, Christian, Lambert, Millard H, Broadway, Neil, Andrews, Robert C, Bickett, D Mark, Leesnitzer, M Anthony, Becherer, J David
Published in Combinatorial chemistry & high throughput screening (01.03.2005)
Published in Combinatorial chemistry & high throughput screening (01.03.2005)
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Characterization of the peptide substrate specificities of interstitial collagenase and 92-kDa gelatinase. Implications for substrate optimization
McGeehan, G M, Bickett, D M, Green, M, Kassel, D, Wiseman, J S, Berman, J
Published in The Journal of biological chemistry (30.12.1994)
Published in The Journal of biological chemistry (30.12.1994)
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MATRIX METALLOPROTEINASE INHIBITORS CONTAINING A (CARBOXYALKYL)AMINO ZINC LIGAND - MODIFICATION OF THE P1 AND P2' RESIDUES
BROWN, FK, BROWN, PJ, BICKETT, DM, CHAMBERS, CL, DAVIES, HG, DEATON, DN, DREWRY, D, FOLEY, M, MCELROY, AB, GREGSON, M, MCGEEHAN, GM, MYERS, PL, NORTON, D, SALOVICH, JM, SCHOENEN, FJ, WARD, P
Published in Journal of medicinal chemistry (04.03.1994)
Published in Journal of medicinal chemistry (04.03.1994)
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Substrate Specificity of Human Collagenase 3 Assessed Using a Phage-displayed Peptide Library
Deng, Su-Jun, Bickett, D. Mark, Mitchell, Justin L., Lambert, Millard H., Blackburn, R. Kevin, Carter, H. Luke, Neugebauer, Jennifer, Pahel, Gregory, Weiner, Michael P., Moss, Marcia L.
Published in The Journal of biological chemistry (06.10.2000)
Published in The Journal of biological chemistry (06.10.2000)
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Inhibition of tumor necrosis factor-alpha (TNF-alpha) production and arthritis in the rat by GW3333, a dual inhibitor of TNF-alpha-converting enzyme and matrix metalloproteinases
Conway, J G, Andrews, R C, Beaudet, B, Bickett, D M, Boncek, V, Brodie, T A, Clark, R L, Crumrine, R C, Leenitzer, M A, McDougald, D L, Han, B, Hedeen, K, Lin, P, Milla, M, Moss, M, Pink, H, Rabinowitz, M H, Tippin, T, Scates, P W, Selph, J, Stimpson, S A, Warner, J, Becherer, J D
Published in The Journal of pharmacology and experimental therapeutics (01.09.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.09.2001)
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6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE
FRYE, SV, HAFFNER, CD, MALONEY, PR, MOOK, RA, HINER, RN, BATCHELOR, KW, BRAMSON, HN, STUART, JD, SCHWEIKER, SL, VANARNOLD, J, BICKETT, DM, MOSS, ML, TIAN, GC, UNWALLA, RJ, LEE, FW, TIPPIN, TK, JAMES, MK, GRIZZLE, MK, LONG, JE, SCHUSTER, SV, DORSEY, GF
Published in Journal of medicinal chemistry (24.12.1993)
Published in Journal of medicinal chemistry (24.12.1993)
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Cloning of a disintegrin metalloproteinase that processes precursor tumour-necrosis factor-α
Moss, Marcia L, Jin, S.-L. Catherine, Milla, Marcos E, Burkhart, William, Carter, H. Luke, Chen, Wen-Ji, Clay, William C, Didsbury, John R, Hassler, Daniel, Hoffman, Christine R, Kost, Thomas A, Lambert, Millard H, Leesnitzer, M. Anthony, McCauley, Philip, McGeehan, Gerard, Mitchell, Justin, Moyer, Mary, Pahel, Gregory, Rocque, Warren, Overton, Laurie K, Schoenen, Frank, Seaton, Theresa, Su, Jui-Lan, Warner, Janet, Willard, Derril, Becherer, J. David
Published in Nature (London) (20.02.1997)
Published in Nature (London) (20.02.1997)
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Effect of matrix metalloproteinase inhibitors on tumor growth and spontaneous metastasis
Conway, J G, Trexler, S J, Wakefield, J A, Marron, B E, Emerson, D L, Bickett, D M, Deaton, D N, Garrison, D, Elder, M, McElroy, A, Willmott, N, Dockerty, A J, McGeehan, G M
Published in Clinical & experimental metastasis (01.03.1996)
Published in Clinical & experimental metastasis (01.03.1996)
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A high throughput fluorogenic substrate for stromelysin (MMP-3)
Bickett, D M, Green, M D, Wagner, C, Roth, J T, Berman, J, McGeehan, G M
Published in Annals of the New York Academy of Sciences (01.09.1994)
Published in Annals of the New York Academy of Sciences (01.09.1994)
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Defined substrate mixtures for mapping of proteinase specificities
McGeehan, G M, Bickett, D M, Wiseman, J S, Green, M, Berman, J
Published in Methods in enzymology (1995)
Published in Methods in enzymology (1995)
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Substrate specificity and novel selective inhibitors of TNF-alpha converting enzyme (TACE) from two-dimensional substrate mapping
Lambert, Millard H, Blackburn, R Kevin, Seaton, Theresa D, Kassel, Daniel B, Kinder, Daniel S, Leesnitzer, M Anthony, Bickett, D Mark, Warner, Janet R, Andersen, Marc W, Badiang, Jennifer G, Cowan, David J, Gaul, Michael D, Petrov, Kimberly G, Rabinowitz, Michael H, Wiethe, Robert W, Becherer, J David, McDougald, Darryl L, Musso, David L, Andrews, Robert C, Moss, Marcia L
Published in Combinatorial chemistry & high throughput screening (01.06.2005)
Published in Combinatorial chemistry & high throughput screening (01.06.2005)
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N-Hydroxyformamide peptidomimetics as TACE/Matrix metalloprotease inhibitors: oral activity via P1′ isobutyl substitution
Musso, David L., Andersen, Marc W., Andrews, Robert C., Austin, Richard, Beaudet, Elizabeth J., Becherer, J.David, Bubacz, Dulce G., Bickett, D.Mark, Chan, Joseph H., Conway, James G., Cowan, David J., Gaul, Michael D., Glennon, Kimberly C., Hedeen, Kevin M., Lambert, Millard H., Leesnitzer, M.Anthony, McDougald, Darryl L., Mitchell, Justin L., Moss, Marcia L., Rabinowitz, Michael H., Rizzolio, Michele C., Schaller, Lee T., Stanford, Jennifer B., Tippin, Timothy K., Warner, Janet R., Whitesell, L.Graham, Wiethe, Robert W.
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Structure-activity relationships for inhibition of type 1 and 2 human 5α-reductase and human adrenal 3β-hydroxy-Δ5-steroid dehydrogenase/3-keto-Δ5-steroid isomerase by 6-azaandrost-4-en-3-ones : optimization of the C17 substituent
FRYE, S. V, HAFFNER, C. D, SCHWEIKER, S. L, VAN ARNOLD, J, BICKETT, D. M, MOSS, M. L, GAOCHOA TIAN, LEE, F. W, TIPPIN, T. K, JAMES, M. K, GRIZZLE, M. K, LONG, J. E, MALONEY, P. R, CROOM, D. K, HINER, R. N, DORSEY, G. F, NOE, R. A, UNWALLA, R. J, BATCHELOR, K. W, BRAMSON, H. N, STUART, J. D
Published in Journal of medicinal chemistry (1995)
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Published in Journal of medicinal chemistry (1995)
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