Species comparison and pharmacological characterization of human, monkey, rat, and mouse TRPA1 channels
Bianchi, Bruce R, Zhang, Xu-Feng, Reilly, Regina M, Kym, Philip R, Yao, Betty B, Chen, Jun
Published in The Journal of pharmacology and experimental therapeutics (01.05.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2012)
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Journal Article
A-995662 [(R)-8-(4-methyl-5-(4-(trifluoromethyl)phenyl)oxazol-2-ylamino)-1,2,3,4-tetrahydronaphthalen-2-ol], a novel, selective TRPV1 receptor antagonist, reduces spinal release of glutamate and CGRP in a rat knee joint pain model
Puttfarcken, Pamela S., Han, Ping, Joshi, Shailen K., Neelands, Torben R., Gauvin, Donna M., Baker, Scott J., Lewis, La Geisha R., Bianchi, Bruce R., Mikusa, Joseph P., Koenig, John R., Perner, Richard J., Kort, Michael E., Honore, Prisca, Faltynek, Connie R., Kym, Philip R., Reilly, Regina M.
Published in Pain (Amsterdam) (01.08.2010)
Published in Pain (Amsterdam) (01.08.2010)
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Journal Article
NOR-Batzelladine L from the sponge Monanchora sp. displays antiviral acyivity against Herpes Simplex virus type 1
Kohn, LK, Porto, PSS, Bianchi, BR, Santos, MFC, Berlinck, RGS, Arns, CW
Published in Planta Medica (19.07.2012)
Published in Planta Medica (19.07.2012)
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Conference Proceeding
A-425619 [1-Isoquinolin-5-yl-3-(4-trifluoromethyl-benzyl)-urea], a Novel and Selective Transient Receptor Potential Type V1 Receptor Antagonist, Blocks Channel Activation by Vanilloids, Heat, and Acid
El Kouhen, Rachid, Surowy, Carol S, Bianchi, Bruce R, Neelands, Torben R, McDonald, Heath A, Niforatos, Wende, Gomtsyan, Arthur, Lee, Chih-Hung, Honore, Prisca, Sullivan, James P, Jarvis, Michael F, Faltynek, Connie R
Published in The Journal of pharmacology and experimental therapeutics (01.07.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2005)
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Journal Article
(R)-(5-tert-Butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)-urea (ABT-102) Blocks Polymodal Activation of Transient Receptor Potential Vanilloid 1 Receptors in Vitro and Heat-Evoked Firing of Spinal Dorsal Horn Neurons in Vivo
Surowy, Carol S, Neelands, Torben R, Bianchi, Bruce R, McGaraughty, Steve, El Kouhen, Rachid, Han, Ping, Chu, Katharine L, McDonald, Heath A, Vos, Melissa, Niforatos, Wende, Bayburt, Erol K, Gomtsyan, Arthur, Lee, Chih-Hung, Honore, Prisca, Sullivan, James P, Jarvis, Michael F, Faltynek, Connie R
Published in The Journal of pharmacology and experimental therapeutics (01.09.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2008)
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Journal Article
Pharmacological characterization of recombinant human and rat P2X receptor subtypes
Bianchi, Bruce R, Lynch, Kevin J, Touma, Edward, Niforatos, Wende, Burgard, Edward C, Alexander, Karen M, Park, Helen S, Yu, Haixia, Metzger, Randy, Kowaluk, Elizabeth, Jarvis, Michael F, van Biesen, Tim
Published in European journal of pharmacology (02.07.1999)
Published in European journal of pharmacology (02.07.1999)
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Journal Article
[3H]A-778317 [1-((R)-5-tert-Butyl-indan-1-yl)-3-isoquinolin-5-yl-urea]: a Novel, Stereoselective, High-Affinity Antagonist Is a Useful Radioligand for the Human Transient Receptor Potential Vanilloid-1 (TRPV1) Receptor
Bianchi, Bruce R, El Kouhen, Rachid, Neelands, Torben R, Lee, Chih-Hung, Gomtsyan, Arthur, Raja, Shirish N, Vaidyanathan, Sriajan N, Surber, Bruce, McDonald, Heath A, Surowy, Carol S, Faltynek, Connie R, Moreland, Robert B, Jarvis, Michael F, Puttfarcken, Pamela S
Published in The Journal of pharmacology and experimental therapeutics (01.10.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2007)
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Journal Article
Characterization of cloned human dopamine D1 receptor-mediated calcium release in 293 cells
Lin, C W, Miller, T R, Witte, D G, Bianchi, B R, Stashko, M, Manelli, A M, Frail, D E
Published in Molecular pharmacology (01.01.1995)
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Published in Molecular pharmacology (01.01.1995)
Journal Article
Human astrocytoma U138MG cells express predominantly type-A endothelin receptor
Wu-Wong, Jinshyun R, Chiou, William, Magnuson, Scott R, Bianchi, Bruce R, Lin, Chun Wel
Published in Biochimica et biophysica acta (28.05.1996)
Published in Biochimica et biophysica acta (28.05.1996)
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Journal Article
Boc-CCK-4 derivatives containing side-chain ureas as potent and selective CCK-A receptor agonists
Shiosaki, Kazumi, Lin, Chun Wel, Kopecka, Hana, Tufano, Michael D, Bianchi, Bruce R, Miller, Thomas R, Witte, David G, Nadzan, Alex M
Published in Journal of medicinal chemistry (01.09.1991)
Published in Journal of medicinal chemistry (01.09.1991)
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Journal Article
A71378: a CCK agonist with high potency and selectivity for CCK-A receptors
Lin, C W, Holladay, M W, Witte, D G, Miller, T R, Wolfram, C A, Bianchi, B R, Bennett, M J, Nadzan, A M
Published in The American journal of physiology (01.04.1990)
Published in The American journal of physiology (01.04.1990)
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Journal Article
Tetrapeptide CCK-A Agonists: Effect of Backbone N-Methylations on in vitro and in vivo CCK Activity
Holladay, Mark W, Kopecka, Hana, Miller, Thomas R, Bednarz, Lisa, Nikkel, A. L, Bianchi, Bruce R, Witte, David G, Shiosaki, Kazumi, Lin, Chun Wel
Published in Journal of medicinal chemistry (01.03.1994)
Published in Journal of medicinal chemistry (01.03.1994)
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Journal Article
Evidence that type A CCK receptors facilitate dopamine efflux in rat brain
Vickroy, T W, Bianchi, B R, Kerwin, Jr, J F, Kopecka, H, Nadzan, A M
Published in European journal of pharmacology (02.08.1988)
Published in European journal of pharmacology (02.08.1988)
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Journal Article
Tetrapeptide CCK agonists: structure-activity studies on modifications at the N-terminus
Elliott, Richard L, Kopecka, Hana, Bennett, Michael J, Shue, Youe Kong, Craig, Richard, Lin, Chun Wel, Bianchi, Bruce R, Miller, Thomas R, Witte, David G
Published in Journal of medicinal chemistry (01.01.1994)
Published in Journal of medicinal chemistry (01.01.1994)
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Journal Article
NOVEL ASP(32)-REPLACEMENT TETRAPEPTIDE ANALOGS AS POTENT AND SELECTIVE CCK-A AGONISTS
ELLIOTT, RL, KOPECKA, H, TUFANO, MD, SHUE, YK, GAURI, AJ, LIN, CW, BIANCHI, BR, MILLER, TR, WITTE, DG, STASHKO, MA, ASIN, KE, NIKKEL, AL, BEDNARZ, L, NADZAN, AM
Published in Journal of medicinal chemistry (27.05.1994)
Published in Journal of medicinal chemistry (27.05.1994)
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Journal Article
Development of potent and selective CCK-A receptor agonists from Boc-CCK-4: tetrapeptides containing Lys(N.epsilon.)-amide residues
Shiosaki, Kazumi, Lin, Chun Wel, Kopecka, Hana, Craig, Richard A, Bianchi, Bruce R, Miller, Thomas R, Witte, David G, Stashko, Michael, Nadzan, Alex M
Published in Journal of medicinal chemistry (01.05.1992)
Published in Journal of medicinal chemistry (01.05.1992)
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Journal Article
CCK-A-Selective Tetrapeptides Containing Lys(N.epsilon.)-Amide Residues: Favorable in vivo and in vitro Effects of N-Methylation at the Aspartyl Residue
Bennett, Michael J, Nikkel, A. L, Bianchi, Bruce R, Miller, Thomas R, Bednarz, Lisa, Witte, David G, Stashko, Michael, Wang, Song Shung, Gore, Paul A
Published in Journal of medicinal chemistry (01.05.1994)
Published in Journal of medicinal chemistry (01.05.1994)
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Journal Article
Cholecystokinin receptors: relationships among phosphoinositide breakdown, amylase release and receptor affinity in pancreas
Lin, C W, Bianchi, B R, Grant, D, Miller, T, Danaher, E A, Tufano, M D, Kopecka, H, Nadzan, A M
Published in The Journal of pharmacology and experimental therapeutics (01.03.1986)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1986)
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