5-Piperazinyl-3-sulfonylindazoles as Potent and Selective 5-Hydroxytryptamine-6 Antagonists
Liu, Kevin G, Robichaud, Albert J, Bernotas, Ronald C, Yan, Yinfa, Lo, Jennifer R, Zhang, Mei-Yi, Hughes, Zoe A, Huselton, Christine, Zhang, Guo Ming, Zhang, Jean Y, Kowal, Dianne M, Smith, Deborah L, Schechter, Lee E, Comery, Thomas A
Published in Journal of medicinal chemistry (11.11.2010)
Published in Journal of medicinal chemistry (11.11.2010)
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Journal Article
3-(3-Aryloxyaryl)imidazo[1,2- a]pyridine sulfones as liver X receptor agonists
Singhaus, Robert R., Bernotas, Ronald C., Steffan, Robert, Matelan, Edward, Quinet, Elaine, Nambi, Ponnal, Feingold, Irene, Huselton, Christine, Wilhelmsson, Anna, Goos-Nilsson, Annika, Wrobel, Jay
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Journal Article
Biarylether amide quinolines as liver X receptor agonists
Bernotas, Ronald C., Singhaus, Robert R., Kaufman, David H., Ullrich, John, Fletcher, Horace, Quinet, Elaine, Nambi, Ponnal, Unwalla, Rayomand, Wilhelmsson, Anna, Goos-Nilsson, Annika, Farnegardh, Mathias, Wrobel, Jay
Published in Bioorganic & medicinal chemistry (15.02.2009)
Published in Bioorganic & medicinal chemistry (15.02.2009)
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Journal Article
1-(3-Aryloxyaryl)benzimidazole sulfones are liver X receptor agonists
Travins, Jeremy M., Bernotas, Ronald C., Kaufman, David H., Quinet, Elaine, Nambi, Ponnal, Feingold, Irene, Huselton, Christine, Wilhelmsson, Anna, Goos-Nilsson, Annika, Wrobel, Jay
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Journal Article
4-(3-Aryloxyaryl)quinoline sulfones are potent liver X receptor agonists
Bernotas, Ronald C., Singhaus, Robert R., Kaufman, David H., Travins, Jeremy M., Ullrich, John W., Unwalla, Rayomand, Quinet, Elaine, Evans, Mark, Nambi, Ponnal, Olland, Andrea, Kauppi, Björn, Wilhelmsson, Anna, Goos-Nilsson, Annika, Wrobel, Jay
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
Discovery of 5-Arylsulfonamido-3- (pyrrolidin-2-ylmethyl)-1H-indole Derivatives as Potent, Selective 5-HT6 Receptor Agonists and Antagonists
Cole, Derek C, Lennox, William J, Lombardi, Sabrina, Ellingboe, John W, Bernotas, Ronald C, Tawa, Gregory J, Mazandarani, Hossein, Smith, Deborah L, Zhang, Guoming, Coupet, Joseph, Schechter, Lee E
Published in Journal of medicinal chemistry (27.01.2005)
Published in Journal of medicinal chemistry (27.01.2005)
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Journal Article
Discovery of N1-(6-Chloroimidazo[2,1-b][1,3]thiazole-5-sulfonyl)tryptamine as a Potent, Selective, and Orally Active 5-HT6 Receptor Agonist
Cole, Derek C, Stock, Joseph R, Lennox, William J, Bernotas, Ronald C, Ellingboe, John W, Boikess, Steve, Coupet, Joseph, Smith, Deborah L, Leung, Louis, Zhang, Guo-Ming, Feng, Xidong, Kelly, Michael F, Galante, Rocco, Huang, Pingzhong, Dawson, Lee A, Marquis, Karen, Rosenzweig-Lipson, Sharon, Beyer, Chad E, Schechter, Lee E
Published in Journal of medicinal chemistry (15.11.2007)
Published in Journal of medicinal chemistry (15.11.2007)
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Journal Article
Novel 1-aminoethyl-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines are potent 5-HT6 agonists
BERNOTAS, Ronald C, LENICEK, Steven, PING LI, COUPET, Joseph, ROSENZWEIG-LIPSON, Sharon, BEYER, Chad E, SCHECHTER, Lee E, ANTANE, Schuyler, COLE, Derek C, HARRISON, Boyd L, ROBICHAUD, Albert J, GUO MING ZHANG, SMITH, Deborah, PLATT, Brian, QIAN LIN
Published in Bioorganic & medicinal chemistry (01.07.2009)
Published in Bioorganic & medicinal chemistry (01.07.2009)
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Journal Article
3-(Arylsulfonyl)-1-(azacyclyl)-1H-indoles are 5-HT6 receptor modulators
BERNOTAS, Ronald C, ANTANE, Schuyler, SHENOY, Rajesh, LE, Van-Duc, PING CHEN, HARRISON, Boyd L, ROBICHAUD, Albert J, GUO MING ZHANG, SMITH, Deborah, SCHECHTER, Lee E
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Journal Article
Synthesis of 4-(3-biaryl)quinoline sulfones as potent liver X receptor agonists
Ullrich, John W., Morris, Robert, Bernotas, Ronald C., Travins, Jeremy M., Jetter, James, Unwalla, Rayomand, Quinet, Elaine, Nambi, Ponnal, Feingold, Irene, Huselton, Christine, Enroth, Christofer, Wilhelmsson, Anna, Goos-Nilsson, Annika, Wrobel, Jay
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Journal Article
4-(3-Aryloxyaryl)quinoline alcohols are liver X receptor agonists
Bernotas, Ronald C., Kaufman, David H., Singhaus, Robert R., Ullrich, John, Unwalla, Rayomand, Quinet, Elaine, Nambi, Ponnal, Wilhelmsson, Anna, Goos-Nilsson, Annika, Wrobel, Jay
Published in Bioorganic & medicinal chemistry (01.12.2009)
Published in Bioorganic & medicinal chemistry (01.12.2009)
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Journal Article
1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-pyrrolopyridines are 5-HT6 receptor ligands
Bernotas, Ronald C., Antane, Schuyler A., Lenicek, Steven E., Haydar, Simon N., Robichaud, Albert J., Harrison, Boyd L., Zhang, Guo Ming, Smith, Deborah, Coupet, Joseph, Schechter, Lee E.
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Journal Article
Novel 1 -(azacyclyl ) -3 -arylsulfonyl -1H -pyrrolo[2,3 -b]pyridines as 5-HT6 agonists and antagonists
ELOKDAH, Hassan, LI, David, MCFARLANE, Geraldine, BERNOTAS, Ronald C, ROBICHAUD, Albert J, MAGOLDA, Ronald L, GUO MING ZHANG, SMITH, Deborah, SCHECHTER, Lee E
Published in Bioorganic & medicinal chemistry (15.09.2007)
Published in Bioorganic & medicinal chemistry (15.09.2007)
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Journal Article
Characterization of the Radical Trapping Activity of a Novel Series of Cyclic Nitrone Spin Traps (∗)
Thomas, Craig E., Ohlweiler, David F., Carr, Albert A., Nieduzak, Thaddeus R., Hay, David A., Adams, Ginette, Vaz, Roy, Bernotas, Ronald C.
Published in The Journal of biological chemistry (09.02.1996)
Published in The Journal of biological chemistry (09.02.1996)
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Journal Article
Evidence for a Novel Pentyl Radical Adduct of the Cyclic Nitrone Spin Trap MDL 101,002
Dage, Jeffrey L, Ackermann, Bradley L, Barbuch, Robert J, Bernotas, Ronald C, Ohlweiler, David F, Haegele, Klaus D, Thomas, Craig E
Published in Free radical biology & medicine (1997)
Published in Free radical biology & medicine (1997)
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Journal Article
Discovery of N-1-(6-chloroimidazo[2,1-b][1,3]-thiazole-5-sulfonyl)tryptamine as a potent, selective, and orally active 5-HT6 receptor agonist
Cole, Derek C., Stock, Joseph R., Lennox, William J., Bernotas, Ronald C., Ellingboe, John W., Boikess, Steve, Coupet, Joseph, Smith, Deborah L., Leung, Louis, Zhang, Guo-Ming, Feng, Xidong, Kelly, Michael F., Galante, Rocco, Huang, Pingzhong, Dawson, Lee A., Marquis, Karen, Rosenzweig-Lipson, Sharon, Beyer, Chad E., Schechter, Lee E.
Published in Journal of medicinal chemistry (15.11.2007)
Published in Journal of medicinal chemistry (15.11.2007)
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Journal Article