Search Results - "BERNHARDT,GUENTHER" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Structural basis of small-molecule inhibition of human multidrug transporter ABCG2

Structural basis of small-molecule inhibition of human multidrug transporter ABCG2

by Jackson, Scott M., Manolaridis, Ioannis, Kowal, Julia, Zechner, Melanie, Taylor, Nicholas M. I., Bause, Manuel, Bauer, Stefanie, Bartholomaeus, Ruben, Bernhardt, Guenther, Koenig, Burkhard, Buschauer, Armin, Stahlberg, Henning, Altmann, Karl-Heinz, Locher, Kaspar P.
Published in Nature structural & molecular biology (01.04.2018)

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Label-Free Investigations on the G Protein Dependent Signaling Pathways of Histamine Receptors

Label-Free Investigations on the G Protein Dependent Signaling Pathways of Histamine Receptors

by Seibel-Ehlert, Ulla, Plank, Nicole, Inoue, Asuka, Bernhardt, Guenther, Strasser, Andrea
Published in International journal of molecular sciences (09.09.2021)

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Structural basis of ligand binding modes at the neuropeptide Y Y1 receptor

Structural basis of ligand binding modes at the neuropeptide Y Y1 receptor

by Yang, Zhenlin, Han, Shuo, Keller, Max, Kaiser, Anette, Bender, Brian J., Bosse, Mathias, Burkert, Kerstin, Kögler, Lisa M., Wifling, David, Bernhardt, Guenther, Plank, Nicole, Littmann, Timo, Schmidt, Peter, Yi, Cuiying, Li, Beibei, Ye, Sheng, Zhang, Rongguang, Xu, Bo, Larhammar, Dan, Stevens, Raymond C., Huster, Daniel, Meiler, Jens, Zhao, Qiang, Beck-Sickinger, Annette G., Buschauer, Armin, Wu, Beili
Published in Nature (London) (01.04.2018)

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Distribution and subcellular localization of a water-soluble hematoporphyrin–platinum(II) complex in human bladder cancer cells

Distribution and subcellular localization of a water-soluble hematoporphyrin–platinum(II) complex in human bladder cancer cells

by Lottner, Christian, Knuechel, Ruth, Bernhardt, Guenther, Brunner, Henri
Published in Cancer letters (25.11.2004)

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Water-soluble inhibitors of ABCG2 (BCRP) – A fragment-based and computational approach

Water-soluble inhibitors of ABCG2 (BCRP) – A fragment-based and computational approach

by Antoni, Frauke, Wifling, David, Bernhardt, Günther
Published in European journal of medicinal chemistry (15.01.2021)

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Derivatives of nitrogen mustard anticancer agents with improved cytotoxicity

Derivatives of nitrogen mustard anticancer agents with improved cytotoxicity

by Antoni, Frauke, Bernhardt, Günther
Published in Archiv der Pharmazie (Weinheim) (01.04.2021)

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Oligopeptides as Neuropeptide Y Y-4 Receptor Ligands: Identification of a High-Affinity Tetrapeptide Agonist and a Hexapeptide Antagonist

Oligopeptides as Neuropeptide Y Y-4 Receptor Ligands: Identification of a High-Affinity Tetrapeptide Agonist and a Hexapeptide Antagonist

by Konieczny, Adam, Braun, Diana, Wifling, David, Bernhardt, Guenther, Keller, Max
Published in Journal of medicinal chemistry (13.08.2020)

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UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H-3 and H-4 Receptors

UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H-3 and H-4 Receptors

by Bartole, Edith, Graetz, Lukas, Littmann, Timo, Wifling, David, Seibel, Ulla, Buschauer, Armin, Bernhardt, Guenther
Published in Journal of medicinal chemistry (28.05.2020)

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Modifications at Arg and Ile Give Neurotensin(8–13) Derivatives with High Stability and Retained NTS1 Receptor Affinity

Modifications at Arg and Ile Give Neurotensin(8–13) Derivatives with High Stability and Retained NTS1 Receptor Affinity

by Schindler, Lisa, Bernhardt, Günther, Keller, Max
Published in ACS medicinal chemistry letters (13.06.2019)

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[H-3]UR-DEBa176: A 2,4-Diaminopyrimidine-Type Radioligand Enabling Binding Studies at the Human, Mouse, and Rat Histamine H-4 Receptors

[H-3]UR-DEBa176: A 2,4-Diaminopyrimidine-Type Radioligand Enabling Binding Studies at the Human, Mouse, and Rat Histamine H-4 Receptors

by Bartole, Edith, Littmann, Timo, Tanaka, Miho, Ozawa, Takeaki, Buschauer, Armin, Bernhardt, Guenther
Published in Journal of medicinal chemistry (12.09.2019)

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Histamine H1- and H4-receptor signaling cooperatively regulate MAPK activation

Histamine H1- and H4-receptor signaling cooperatively regulate MAPK activation

by Beermann, Silke, Bernhardt, Guenther, Seifert, Roland, Buschauer, Armin, Neumann, Detlef
Published in Biochemical pharmacology (01.12.2015)

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Structural basis of ligand binding modes at the neuropeptide Y Y 1 receptor

Structural basis of ligand binding modes at the neuropeptide Y Y 1 receptor

by Yang, Zhenlin, Han, Shuo, Keller, Max, Kaiser, Anette, Bender, Brian J, Bosse, Mathias, Burkert, Kerstin, Kögler, Lisa M, Wifling, David, Bernhardt, Guenther, Plank, Nicole, Littmann, Timo, Schmidt, Peter, Yi, Cuiying, Li, Beibei, Ye, Sheng, Zhang, Rongguang, Xu, Bo, Larhammar, Dan, Stevens, Raymond C, Huster, Daniel, Meiler, Jens, Zhao, Qiang, Beck-Sickinger, Annette G, Buschauer, Armin, Wu, Beili
Published in Nature (London) (26.04.2018)

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A split luciferase-based probe for quantitative proximal determination of Gαq signalling in live cells

A split luciferase-based probe for quantitative proximal determination of Gαq signalling in live cells

by Littmann, Timo, Ozawa, Takeaki, Hoffmann, Carsten, Buschauer, Armin, Bernhardt, Günther
Published in Scientific reports (21.11.2018)

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Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M-2 Muscarinic Acetylcholine Receptor

Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M-2 Muscarinic Acetylcholine Receptor

by Pegoli, Andrea, She, Xueke, Wifling, David, Huebner, Harald, Bernhardt, Guenther, Gmeiner, Peter, Keller, Max
Published in Journal of medicinal chemistry (27.04.2017)

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High Affinity Agonists of the Neuropeptide Y (NPY) Y-4 Receptor Derived from the C-Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling

High Affinity Agonists of the Neuropeptide Y (NPY) Y-4 Receptor Derived from the C-Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling

by Kuhn, Kilian K., Ertl, Thomas, Dukorn, Stefanie, Keller, Max, Bernhardt, Guenther, Reiser, Oliver, Buschauer, Armin
Published in Journal of medicinal chemistry (14.07.2016)

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Tariquidar-related triazoles as potent, selective and stable inhibitors of ABCG2 (BCRP)

Tariquidar-related triazoles as potent, selective and stable inhibitors of ABCG2 (BCRP)

by Antoni, Frauke, Bause, Manuel, Scholler, Matthias, Bauer, Stefanie, Stark, Simone A., Jackson, Scott M., Manolaridis, Ioannis, Locher, Kaspar P., König, Burkhard, Buschauer, Armin, Bernhardt, Günther
Published in European journal of medicinal chemistry (01.04.2020)

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Flavonoid derivatives as selective ABCC1 modulators: Synthesis and functional characterization

Flavonoid derivatives as selective ABCC1 modulators: Synthesis and functional characterization

by Obreque-Balboa, José Esteban, Sun, Qiu, Bernhardt, Günther, König, Burkhard, Buschauer, Armin
Published in European journal of medicinal chemistry (15.02.2016)

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Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity

Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity

by Pegoli, Andrea, Wifling, David, Gruber, Corinna G, She, Xueke, Hübner, Harald, Bernhardt, Günther, Gmeiner, Peter, Keller, Max
Published in Journal of medicinal chemistry (13.06.2019)

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Replacement of Thr(32) and GIn(34) in the C-Terminal Neuropeptide Y Fragment 25-36 by cis-Cyclobutane and cis-Cyclopentane beta-Amino Acids Shifts Selectivity toward the Y-4 Receptor

Replacement of Thr(32) and GIn(34) in the C-Terminal Neuropeptide Y Fragment 25-36 by cis-Cyclobutane and cis-Cyclopentane beta-Amino Acids Shifts Selectivity toward the Y-4 Receptor

by Berlicki, Lukasz, Kaske, Melanie, Gutierrez-Abad, Raquel, Bernhardt, Guenther, Illa, Ona, Ortuno, Rosa M., Cabrele, Chiara, Buschauer, Armin, Reiser, Oliver
Published in Journal of medicinal chemistry (14.11.2013)

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Dimeric carbamoylguanidine-type histamine H-2 receptor ligands: A new class of potent and selective agonists

Dimeric carbamoylguanidine-type histamine H-2 receptor ligands: A new class of potent and selective agonists

by Kagermeier, Nicole, Werner, Kristin, Keller, Max, Baumeister, Paul, Bernhardt, Guenther, Seifert, Roland, Buschauer, Armin
Published in Bioorganic & medicinal chemistry (15.07.2015)

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