Search Results - "BERESIS, RICHARD" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Neuroactive Steroids. 2. 3α-Hydroxy-3β-methyl-21-(4-cyano‑1H‑pyrazol-1′-yl)-19-nor-5β-pregnan-20-one (SAGE-217): A Clinical Next Generation Neuroactive Steroid Positive Allosteric Modulator of the (γ-Aminobutyric Acid)A Receptor

Neuroactive Steroids. 2. 3α-Hydroxy-3β-methyl-21-(4-cyano‑1H‑pyrazol-1′-yl)-19-nor-5β-pregnan-20-one (SAGE-217): A Clinical Next Generation Neuroactive Steroid Positive Allosteric Modulator of the (γ-Aminobutyric Acid)A Receptor

by Martinez Botella, Gabriel, Salituro, Francesco G, Harrison, Boyd L, Beresis, Richard T, Bai, Zhu, Blanco, Maria-Jesus, Belfort, Gabriel M, Dai, Jing, Loya, Carlos M, Ackley, Michael A, Althaus, Alison L, Grossman, Scott J, Hoffmann, Ethan, Doherty, James J, Robichaud, Albert J
Published in Journal of medicinal chemistry (28.09.2017)

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Journal Article

Neuroactive Steroids. 1. Positive Allosteric Modulators of the (γ-Aminobutyric Acid)A Receptor: Structure–Activity Relationships of Heterocyclic Substitution at C‑21

Neuroactive Steroids. 1. Positive Allosteric Modulators of the (γ-Aminobutyric Acid)A Receptor: Structure–Activity Relationships of Heterocyclic Substitution at C‑21

by Martinez Botella, Gabriel, Salituro, Francesco G, Harrison, Boyd L, Beresis, Richard T, Bai, Zhu, Shen, Kaisheng, Belfort, Gabriel M, Loya, Carlos M, Ackley, Michael A, Grossman, Scott J, Hoffmann, Ethan, Jia, Shiling, Wang, Jiamiao, Doherty, James J, Robichaud, Albert J
Published in Journal of medicinal chemistry (23.04.2015)

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Journal Article

Methods to assess small molecule allosteric modulators of the STRAD pseudokinase

Methods to assess small molecule allosteric modulators of the STRAD pseudokinase

by Qing, Tingting, Liu, Jin, Liu, Fen, Mitchell, Dom C, Beresis, Richard T, Gordan, John D
Published in Methods in enzymology (2022)

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Molecular modeling aided design of nicotinic acid receptor GPR109A agonists

Molecular modeling aided design of nicotinic acid receptor GPR109A agonists

by Deng, Qiaolin, Frie, Jessica L., Marley, Daria M., Beresis, Richard T., Ren, Ning, Cai, Tian-Quan, Taggart, Andrew K.P., Cheng, Kang, Carballo-Jane, Ester, Wang, Junying, Tong, Xinchun, Waters, M. Gerard, Tata, James R., Colletti, Steven L.
Published in Bioorganic & medicinal chemistry (15.09.2008)

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Disubstituted pyrimidines as Lck inhibitors

Disubstituted pyrimidines as Lck inhibitors

by Hunt, Julianne A., Beresis, Richard T., Goulet, Joung L., Holmes, Mark A., Hong, Xinfang J., Kovacs, Ernest, Mills, Sander G., Ruzek, Rowena D., Wong, Frederick, Hermes, Jeffrey D., Park, Young-Whan, Salowe, Scott P., Sonatore, Lisa M., Wu, Lin, Woods, Andrea, Zaller, Dennis M., Sinclair, Peter J.
Published in Bioorganic & medicinal chemistry letters (15.09.2009)

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Journal Article

Synthesis of the Vancomycin CD and DE Ring Systems

Synthesis of the Vancomycin CD and DE Ring Systems

by Boger, Dale L, Borzilleri, Robert M, Nukui, Seiji, Beresis, Richard T
Published in Journal of organic chemistry (11.07.1997)

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Journal Article

Studies Directed toward the Synthesis of Ulapualide A. Asymmetric Synthesis of the C8−C25 Tris-Oxazole Fragment

Studies Directed toward the Synthesis of Ulapualide A. Asymmetric Synthesis of the C8−C25 Tris-Oxazole Fragment

by Panek, James S, Beresis, Richard T
Published in Journal of organic chemistry (20.09.1996)

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Journal Article

Mechanistic Evaluation and In Vivo Validation of a Novel HIPK2 Inhibitor as Anti-Fibrosis Therapy for Kidney Disease: FR-PO946

Mechanistic Evaluation and In Vivo Validation of a Novel HIPK2 Inhibitor as Anti-Fibrosis Therapy for Kidney Disease: FR-PO946

by Lee, Kyung, Feng, Ye, Chen, Yibang, Beresis, Richard T., Drakas, Robert, He, John C.
Published in Journal of the American Society of Nephrology (01.11.2022)

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A Novel Allosteric HIPK2 Inhibitor Attenuates Renal Fibrosis with Superior Pharmacokinetic, Selectivity, and Safety Profiles: PO2474

A Novel Allosteric HIPK2 Inhibitor Attenuates Renal Fibrosis with Superior Pharmacokinetic, Selectivity, and Safety Profiles: PO2474

by Lee, Kyung, Feng, Ye, Chen, Ya, Beresis, Richard T., Drakas, Robert, He, John C.
Published in Journal of the American Society of Nephrology (01.10.2021)

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Journal Article

Thermal Atropisomerism of Aglucovancomycin Derivatives: Preparation of (M,M,M)- and (P,M,M)-Aglucovancomycins

Thermal Atropisomerism of Aglucovancomycin Derivatives: Preparation of (M,M,M)- and (P,M,M)-Aglucovancomycins

by Boger, Dale L, Miyazaki, Susumu, Loiseleur, Olivier, Beresis, Richard T, Castle, Steven L, Wu, Jason H, Jin, Qing
Published in Journal of the American Chemical Society (09.09.1998)

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Journal Article

Neuroactive Steroids. 2.3 alpha-Hydroxy-3 beta-methyl-21-(4-cyano-1H-pyrazol-1 '-yl)-19-nor-5 beta-pregnan-20-one (SAGE-217): A Clinical Next Generation Neuroactive Steroid Positive Allosteric Modulator of the (gamma-Aminobutyric Acid)(A) Receptor

Neuroactive Steroids. 2.3 alpha-Hydroxy-3 beta-methyl-21-(4-cyano-1H-pyrazol-1 '-yl)-19-nor-5 beta-pregnan-20-one (SAGE-217): A Clinical Next Generation Neuroactive Steroid Positive Allosteric Modulator of the (gamma-Aminobutyric Acid)(A) Receptor

by Botella, Gabriel Martinez, Salituro, Francesco G., Harrison, Boyd L., Beresis, Richard T., Bai, Zhu, Blanco, Maria-Jesus, Belfort, Gabriel M., Dai, Jing, Loya, Carlos M., Ackley, Michael A., Althaus, Alison L., Grossman, Scott J., Hoffmann, Ethan, Doherty, James J., Robichaud, Albert J.
Published in Journal of medicinal chemistry (28.09.2017)

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Journal Article

Oligomeric State and Drug Binding of the SARS-CoV‑2 Envelope Protein Are Sensitive to the Ectodomain

Oligomeric State and Drug Binding of the SARS-CoV‑2 Envelope Protein Are Sensitive to the Ectodomain

by Somberg, Noah H., Sučec, Iva, Medeiros-Silva, João, Jo, Hyunil, Beresis, Richard, Syed, Abdullah M., Doudna, Jennifer A., Hong, Mei
Published in Journal of the American Chemical Society (04.09.2024)

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Journal Article

신장 섬유증의 치료를 위한 HIPK2의 옥사디아졸릴 디하이드로피라노[2,3-b]피리딘 억제제

신장 섬유증의 치료를 위한 HIPK2의 옥사디아졸릴 디하이드로피라노[2,3-b]피리딘 억제제

by BERESIS RICHARD T, LEE KYUNG, HE JOHN CIJIANG
Year of Publication 07.11.2023

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Patent

Vancomycin CD and DE Macrocyclization and Atropisomerism Studies

Vancomycin CD and DE Macrocyclization and Atropisomerism Studies

by Boger, Dale L, Castle, Steven L, Miyazaki, Susumu, Wu, Jason H, Beresis, Richard T, Loiseleur, Olivier
Published in Journal of organic chemistry (08.01.1999)

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Journal Article

STRAD-결합제 및 이의 용도

STRAD-결합제 및 이의 용도

by GORDAN JOHN, MITCHELL DOMINIQUE, BERESIS RICHARD, ADLER MARC
Year of Publication 10.11.2022

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Patent

NEUROACTIVE STEROIDS COMPOSITIONS AND USES THEREOF

NEUROACTIVE STEROIDS COMPOSITIONS AND USES THEREOF

by BOTELLA GABRIEL MARTINEZ, BERESIS RICHARD THOMAS, SALITURO FRANCESCO G, ROBICHAUD ALBERT JEAN, HARRISON BOYD L
Year of Publication 14.05.2024

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Patent

Studies Directed toward the Synthesis of Ulapualide A. Asymmetric Synthesis of the C26−C42 Fragment

Studies Directed toward the Synthesis of Ulapualide A. Asymmetric Synthesis of the C26−C42 Fragment

by Panek, James S, Beresis, Richard T, Celatka, Cassandra A
Published in Journal of organic chemistry (20.09.1996)

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Journal Article

19- C33- C21-N- 19-NOR C33-DISUBSTITUTED C21-N-PYRAZOLYL STEROIDS AND METHODS OF USE THEREOF

19- C33- C21-N- 19-NOR C33-DISUBSTITUTED C21-N-PYRAZOLYL STEROIDS AND METHODS OF USE THEREOF

by BOTELLA GABRIEL MARTINEZ, BERESIS RICHARD THOMAS, SALITURO FRANCESCO G, ROBICHAUD ALBERT JEAN, HARRISON BOYD L
Year of Publication 22.12.2023

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Patent

Dual antagonists of alpha 5 beta 1/alpha v beta 1 integrin for airway hyperresponsiveness

Dual antagonists of alpha 5 beta 1/alpha v beta 1 integrin for airway hyperresponsiveness

by Sundaram, Aparna, Chen, Chun, Reed, Nilgun Isik, Liu, Sean, Yeon, Seul Ki, McIntosh, Joel, Tang, You-Zhi, Yang, Hyunjun, Adler, Marc, Beresis, Richard, Seiple, Ian B., Sheppard, Dean, DeGrado, William F., Jo, Hyunil
Published in Bioorganic & medicinal chemistry letters (15.11.2020)

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Journal Article

19-NOR C3,3-DISUBSTITUTED C21-N-PYRAZOLYL STEROIDS AND METHODS OF USE THEREOF

19-NOR C3,3-DISUBSTITUTED C21-N-PYRAZOLYL STEROIDS AND METHODS OF USE THEREOF

by GABRIEL MARTINEZ BOTELLA, SALITURO FRANCESCO G, BOYD L HARRISON, ALBERT JEAN ROBICHAUD, THOMAS BERESIS RICHARD
Year of Publication 18.10.2023

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Patent

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