Identification of the Clinical Candidate (R)‑(1-(4-Fluorophenyl)-6-((1-methyl‑1H‑pyrazol-4-yl)sulfonyl)-4,4a,5,6,7,8-hexahydro‑1H‑pyrazolo[3,4‑g]isoquinolin-4a-yl)(4-(trifluoromethyl)pyridin-2-yl)methanone (CORT125134): A Selective Glucocorticoid Receptor (GR) Antagonist
Hunt, Hazel J, Belanoff, Joseph K, Walters, Iain, Gourdet, Benoit, Thomas, Jennifer, Barton, Naomi, Unitt, John, Phillips, Timothy, Swift, Denise, Eaton, Emily
Published in Journal of medicinal chemistry (27.04.2017)
Published in Journal of medicinal chemistry (27.04.2017)
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Journal Article
To homeostasis and beyond! Recent advances in the medicinal chemistry of heterobifunctional derivatives
Castagna, Diana, Gourdet, Benoit, Hjerpe, Roland, MacFaul, Philip, Novak, Andrew, Revol, Guillaume, Rochette, Etienne, Jordan, Allan
Published in Progress in medicinal chemistry (2024)
Published in Progress in medicinal chemistry (2024)
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Journal Article
1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as potent GR antagonists with reduced hERG inhibition and an improved pharmacokinetic profile
Hunt, Hazel J., Belanoff, Joseph K., Golding, Emily, Gourdet, Benoit, Phillips, Timothy, Swift, Denise, Thomas, Jennifer, Unitt, John F., Walters, Iain
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
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Journal Article
Identification of the Clinical Candidate ( R )-(1-(4-Fluorophenyl)-6-((1-methyl-1 H -pyrazol-4-yl)sulfonyl)-4,4a,5,6,7,8-hexahydro-1 H -pyrazolo[3,4- g ]isoquinolin-4a-yl)(4-(trifluoromethyl)pyridin-2-yl)methanone (CORT125134): A Selective Glucocorticoid Receptor (GR) Antagonist
Hunt, Hazel J., Belanoff, Joseph K., Walters, Iain, Gourdet, Benoit, Thomas, Jennifer, Barton, Naomi, Unitt, John, Phillips, Timothy, Swift, Denise, Eaton, Emily
Published in Journal of medicinal chemistry (27.04.2017)
Published in Journal of medicinal chemistry (27.04.2017)
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Journal Article
ADO-RESISTANT CYSTEAMINE ANALOGS AND USES THEREOF
LORNA DUFFY, ZANKEL TODD C, BENOIT GOURDET, TIMOTHY PHILLIPS, JOHN UNITT
Year of Publication 30.09.2021
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Year of Publication 30.09.2021
Patent
Abstract 3111: The Sygnature CHARMD platform - combinatorial high-throughput assembly and review of molecular degraders
Hjerpe, Roland, Birch, Louise, Brien, Alex, Cusin, Lola, Duffy, Lorna, Gourdet, Benoit, Lawrence, Rachel, MacFaul, Philip, Mortlock, Hannah, Neal, Hannah, Pearce, Christopher, Pitti, Erica, Robles, Gonzalo, Rodrigues, Edith, Scott, Catriona, Singh, Rajesh, Thomson, Stuart, Zhang, Yujia, Jordan, Allan
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Journal Article
Abstract LB030: Building a platform of validated high throughput screening approaches for molecular glue degrader identification
Jordan, Allan, Addis, Philip, Allen, Toby, Ayra, Tarun, Beck, Sarah, Brant, Roslyn, Hjerpe, Roland, Gourdet, Benoit, Jennings, Martin, Lawrence, Rachel, Campbell-Maurer, Sigrun, Ng, Pei Cing, Parkinson, Lyn, Rejnowicz, Eva, Robles, Gonzalo, Rosethorne, Elizabeth, Shaw, Joshua, Smith, Duncan, Swift, Denise, Tait, Daniel, Thomson, Stuart, Tomlinson, Chris, Townley, Ailsa, Ward, Stephanie, Wilson, Clare
Published in Cancer research (Chicago, Ill.) (05.04.2024)
Published in Cancer research (Chicago, Ill.) (05.04.2024)
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Journal Article
Extremely regio-regular poly (3-alkylthiophene)s from simplified chain-growth Grignard metathesis polymerisations and the modification of their chain-ends
Hiorns, Roger C, Khoukh, Abdel, Gourdet, Benoit, Dagron-Lartigau, Christine
Published in Polymer international (01.06.2006)
Published in Polymer international (01.06.2006)
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Journal Article
Conference Proceeding