Targeted Protein Degradation by Electrophilic PROTACs that Stereoselectively and Site-Specifically Engage DCAF1
Tao, Yongfeng, Remillard, David, Vinogradova, Ekaterina V., Yokoyama, Minoru, Banchenko, Sofia, Schwefel, David, Melillo, Bruno, Schreiber, Stuart L., Zhang, Xiaoyu, Cravatt, Benjamin F.
Published in Journal of the American Chemical Society (12.10.2022)
Published in Journal of the American Chemical Society (12.10.2022)
Get full text
Journal Article
Mapping Enzyme Active Sites in Complex Proteomes
Adam, Gregory C, Burbaum, Jonathan, Kozarich, John W, Patricelli, Matthew P, Cravatt, Benjamin F
Published in Journal of the American Chemical Society (11.02.2004)
Published in Journal of the American Chemical Society (11.02.2004)
Get full text
Journal Article
Monoacylglycerol Lipase Regulates a Fatty Acid Network that Promotes Cancer Pathogenesis
Nomura, Daniel K., Long, Jonathan Z., Niessen, Sherry, Hoover, Heather S., Ng, Shu-Wing, Cravatt, Benjamin F.
Published in Cell (08.01.2010)
Published in Cell (08.01.2010)
Get full text
Journal Article
Formation of prostamides from anandamide in FAAH knockout mice analyzed by HPLC with tandem mass spectrometry
Weber, Allan, Ni, Jinsong, Ling, Kah-Hiing John, Acheampong, Andrew, Tang-Liu, Diane D-S., Burk, Robert, Cravatt, Benjamin F., Woodward, David
Published in Journal of lipid research (01.04.2004)
Published in Journal of lipid research (01.04.2004)
Get full text
Journal Article
Synthesis and Sulfur Electrophilicity of the Nuphar Thiaspirane Pharmacophore
Tada, Norihiro, Jansen, Daniel J, Mower, Matthew P, Blewett, Megan M, Umotoy, Jeffrey C, Cravatt, Benjamin F, Wolan, Dennis W, Shenvi, Ryan A
Published in ACS central science (22.06.2016)
Published in ACS central science (22.06.2016)
Get full text
Journal Article
The enzymatic inactivation of the fatty acid amide class of signaling lipids
Get full text
Book Review
Journal Article
Expedited mapping of the ligandable proteome using fully functionalized enantiomeric probe pairs
Wang, Yujia, Dix, Melissa M., Bianco, Giulia, Remsberg, Jarrett R., Lee, Hsin-Yu, Kalocsay, Marian, Gygi, Steven P., Forli, Stefano, Vite, Gregory, Lawrence, R. Michael, Parker, Christopher G., Cravatt, Benjamin F.
Published in Nature chemistry (01.12.2019)
Published in Nature chemistry (01.12.2019)
Get full text
Journal Article
SPIN4 Is a Principal Endogenous Substrate of the E3 Ubiquitin Ligase DCAF16
Zhang, Xiaoyu, Thielert, Marvin, Li, Haoxin, Cravatt, Benjamin F
Published in Biochemistry (Easton) (09.03.2021)
Published in Biochemistry (Easton) (09.03.2021)
Get full text
Journal Article
Excessive alcohol intake produces persistent mechanical allodynia and dysregulates the endocannabinoid system in the lumbar dorsal root ganglia of genetically-selected Marchigian Sardinian alcohol-preferring rats
Borgonetti, Vittoria, Vozella, Valentina, Ware, Tim, Cruz, Bryan, Bullard, Ryan, Cravatt, Benjamin F., Galeotti, Nicoletta, Roberto, Marisa
Published in Pharmacological research (01.11.2024)
Published in Pharmacological research (01.11.2024)
Get full text
Journal Article
An Activity-Guided Map of Electrophile-Cysteine Interactions in Primary Human T Cells
Vinogradova, Ekaterina V., Zhang, Xiaoyu, Remillard, David, Lazar, Daniel C., Suciu, Radu M., Wang, Yujia, Bianco, Giulia, Yamashita, Yu, Crowley, Vincent M., Schafroth, Michael A., Yokoyama, Minoru, Konrad, David B., Lum, Kenneth M., Simon, Gabriel M., Kemper, Esther K., Lazear, Michael R., Yin, Sifei, Blewett, Megan M., Dix, Melissa M., Nguyen, Nhan, Shokhirev, Maxim N., Chin, Emily N., Lairson, Luke L., Melillo, Bruno, Schreiber, Stuart L., Forli, Stefano, Teijaro, John R., Cravatt, Benjamin F.
Published in Cell (20.08.2020)
Published in Cell (20.08.2020)
Get full text
Journal Article
Activity-based Protein Profiling Implicates Urokinase Activation as a Key Step in Human Fibrosarcoma Intravasation
Madsen, Mark A., Deryugina, Elena I., Niessen, Sherry, Cravatt, Benjamin F., Quigley, James P.
Published in The Journal of biological chemistry (09.06.2006)
Published in The Journal of biological chemistry (09.06.2006)
Get full text
Journal Article
Rapid Development of a Potent Photo-triggered Inhibitor of the Serine Hydrolase RBBP9
Liu, Xiaodan, Dix, Melissa, Speers, Anna E., Bachovchin, Daniel A., Zuhl, Andrea M., Cravatt, Benjamin F., Kodadek, Thomas J.
Published in Chembiochem : a European journal of chemical biology (24.09.2012)
Published in Chembiochem : a European journal of chemical biology (24.09.2012)
Get full text
Journal Article
Prolonged Monoacylglycerol Lipase Blockade Causes Equivalent Cannabinoid Receptor Type 1 Receptor–Mediated Adaptations in Fatty Acid Amide Hydrolase Wild-Type and Knockout Mice
Schlosburg, Joel E., Kinsey, Steven G., Ignatowska-Jankowska, Bogna, Ramesh, Divya, Abdullah, Rehab A., Tao, Qing, Booker, Lamont, Long, Jonathan Z., Selley, Dana E., Cravatt, Benjamin F., Lichtman, Aron H.
Published in The Journal of pharmacology and experimental therapeutics (01.08.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2014)
Get full text
Journal Article
Endocannabinoid Hydrolysis Generates Brain Prostaglandins That Promote Neuroinflammation
Nomura, Daniel K., Morrison, Bradley E., Blankman, Jacqueline L., Long, Jonathan Z., Kinsey, Steven G., Marcondes, Maria Cecilia G., Ward, Anna M., Hahn, Yun Kyung, Lichtman, Aron H., Conti, Bruno, Cravatt, Benjamin F.
Published in Science (American Association for the Advancement of Science) (11.11.2011)
Published in Science (American Association for the Advancement of Science) (11.11.2011)
Get full text
Journal Article