Intracellular Released Payload Influences Potency and Bystander-Killing Effects of Antibody-Drug Conjugates in Preclinical Models
Li, Fu, Emmerton, Kim K, Jonas, Mechthild, Zhang, Xinqun, Miyamoto, Jamie B, Setter, Jocelyn R, Nicholas, Nicole D, Okeley, Nicole M, Lyon, Robert P, Benjamin, Dennis R, Law, Che-Leung
Published in Cancer research (Chicago, Ill.) (01.05.2016)
Published in Cancer research (Chicago, Ill.) (01.05.2016)
Get full text
Journal Article
Intracellular Activation of SGN-35, a Potent Anti-CD30 Antibody-Drug Conjugate
OKELEY, Nicole M, MIYAMOTO, Jamie B, XINQUN ZHANG, SANDERSON, Russell J, BENJAMIN, Dennis R, SIEVERS, Eric L, SENTER, Peter D, ALLEY, Stephen C
Published in Clinical cancer research (01.02.2010)
Published in Clinical cancer research (01.02.2010)
Get full text
Journal Article
SGN-LIV1A: a novel antibody-drug conjugate targeting LIV-1 for the treatment of metastatic breast cancer
Sussman, Django, Smith, Leia M, Anderson, Martha E, Duniho, Steve, Hunter, Joshua H, Kostner, Heather, Miyamoto, Jamie B, Nesterova, Albina, Westendorf, Lori, Van Epps, Heather A, Whiting, Nancy, Benjamin, Dennis R
Published in Molecular cancer therapeutics (01.12.2014)
Published in Molecular cancer therapeutics (01.12.2014)
Get full text
Journal Article
Development of orally active inhibitors of protein and cellular fucosylation
Okeley, Nicole M., Alley, Stephen C., Anderson, Martha E., Boursalian, Tamar E., Burke, Patrick J., Emmerton, Kim M., Jeffrey, Scott C., Klussman, Kerry, Law, Che-Leung, Sussman, Django, Toki, Brian E., Westendorf, Lori, Zeng, Weiping, Zhang, Xinqun, Benjamin, Dennis R., Senter, Peter D.
Published in Proceedings of the National Academy of Sciences - PNAS (02.04.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (02.04.2013)
Get full text
Journal Article
The Pharmacologic Basis for Antibody-Auristatin Conjugate Activity
Alley, Stephen C, Zhang, Xinqun, Okeley, Nicole M, Anderson, Martha, Law, Che-Leung, Senter, Peter D, Benjamin, Dennis R
Published in The Journal of pharmacology and experimental therapeutics (01.09.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2009)
Get full text
Journal Article
The fucosylation inhibitor, 2-fluorofucose, inhibits vaso-occlusion, leukocyte-endothelium interactions and NF-ĸB activation in transgenic sickle mice
Belcher, John D, Chen, Chunsheng, Nguyen, Julia, Abdulla, Fuad, Nguyen, Phong, Nguyen, Minh, Okeley, Nicole M, Benjamin, Dennis R, Senter, Peter D, Vercellotti, Gregory M
Published in PloS one (23.02.2015)
Published in PloS one (23.02.2015)
Get full text
Journal Article
Detection and Selective Dissociation of Intact Ribosomes in a Mass Spectrometer
Rostom, Adam A., Fucini, Paola, Benjamin, Dennis R., Juenemann, Ralf, Nierhaus, Knud H., Hartl, F. Ulrich, Dobson, Christopher M., Robinson, Carol V.
Published in Proceedings of the National Academy of Sciences - PNAS (09.05.2000)
Published in Proceedings of the National Academy of Sciences - PNAS (09.05.2000)
Get full text
Journal Article
SGN-CD33A: a novel CD33-targeting antibody–drug conjugate using a pyrrolobenzodiazepine dimer is active in models of drug-resistant AML
Kung Sutherland, May S., Walter, Roland B., Jeffrey, Scott C., Burke, Patrick J., Yu, Changpu, Kostner, Heather, Stone, Ivan, Ryan, Maureen C., Sussman, Django, Lyon, Robert P., Zeng, Weiping, Harrington, Kimberly H., Klussman, Kerry, Westendorf, Lori, Meyer, David, Bernstein, Irwin D., Senter, Peter D., Benjamin, Dennis R., Drachman, Jonathan G., McEarchern, Julie A.
Published in Blood (22.08.2013)
Published in Blood (22.08.2013)
Get full text
Journal Article
Mouse Strains Influence Clearance and Efficacy of Antibody and Antibody-Drug Conjugate Via Fc-FcγR Interaction
Li, Fu, Ulrich, Michelle L, Shih, Vincent Feng-Sheng, Cochran, Julia H, Hunter, Joshua H, Westendorf, Lori, Neale, Jason, Benjamin, Dennis R
Published in Molecular cancer therapeutics (01.04.2019)
Published in Molecular cancer therapeutics (01.04.2019)
Get full text
Journal Article
Tumor-Associated Macrophages Can Contribute to Antitumor Activity through FcγR-Mediated Processing of Antibody-Drug Conjugates
Li, Fu, Ulrich, Michelle, Jonas, Mechthild, Stone, Ivan J, Linares, Germein, Zhang, Xinqun, Westendorf, Lori, Benjamin, Dennis R, Law, Che-Leung
Published in Molecular cancer therapeutics (01.07.2017)
Published in Molecular cancer therapeutics (01.07.2017)
Get full text
Journal Article
Design, synthesis and selection of DNA-encoded small-molecule libraries
Morgan, Barry A, Clark, Matthew A, Acharya, Raksha A, Arico-Muendel, Christopher C, Belyanskaya, Svetlana L, Benjamin, Dennis R, Carlson, Neil R, Centrella, Paolo A, Chiu, Cynthia H, Creaser, Steffen P, Cuozzo, John W, Davie, Christopher P, Ding, Yun, Franklin, G Joseph, Franzen, Kurt D, Gefter, Malcolm L, Hale, Steven P, Hansen, Nils J V, Israel, David I, Jiang, Jinwei, Kavarana, Malcolm J, Kelley, Michael S, Kollmann, Christopher S, Li, Fan, Lind, Kenneth, Mataruse, Sibongile, Medeiros, Patricia F, Messer, Jeffrey A, Myers, Paul, O'Keefe, Heather, Oliff, Matthew C, Rise, Cecil E, Satz, Alexander L, Skinner, Steven R, Svendsen, Jennifer L, Tang, Lujia, van Vloten, Kurt, Wagner, Richard W, Yao, Gang, Zhao, Baoguang
Published in Nature Chemical Biology (01.09.2009)
Published in Nature Chemical Biology (01.09.2009)
Get full text
Journal Article
Characterization of SGN-CD123A, A Potent CD123-Directed Antibody-Drug Conjugate for Acute Myeloid Leukemia
Li, Fu, Sutherland, May Kung, Yu, Changpu, Walter, Roland B, Westendorf, Lori, Valliere-Douglass, John, Pan, Lucy, Cronkite, Ashley, Sussman, Django, Klussman, Kerry, Ulrich, Michelle, Anderson, Martha E, Stone, Ivan J, Zeng, Weiping, Jonas, Mechthild, Lewis, Timothy S, Goswami, Maitrayee, Wang, Sa A, Senter, Peter D, Law, Che-Leung, Feldman, Eric J, Benjamin, Dennis R
Published in Molecular cancer therapeutics (01.02.2018)
Published in Molecular cancer therapeutics (01.02.2018)
Get full text
Journal Article
Carbamate Analogues of Fumagillin as Potent, Targeted Inhibitors of Methionine Aminopeptidase-2
Arico-Muendel, Christopher C, Benjamin, Dennis R, Caiazzo, Teresa M, Centrella, Paolo A, Contonio, Brooke D, Cook, Charles M, Doyle, Elisabeth G, Hannig, Gerhard, Labenski, Matthew T, Searle, Lily L, Lind, Kenneth, Morgan, Barry A, Olson, Gary, Paradise, Christopher L, Self, Christopher, Skinner, Steven R, Sluboski, Barbara, Svendsen, Jennifer L, Thompson, Charles D, Westlin, William, White, Kerry F
Published in Journal of medicinal chemistry (24.12.2009)
Published in Journal of medicinal chemistry (24.12.2009)
Get full text
Journal Article
Orally Active Fumagillin Analogues: Transformations of a Reactive Warhead in the Gastric Environment
Arico-Muendel, Christopher C, Blanchette, Heather, Benjamin, Dennis R, Caiazzo, Teresa M, Centrella, Paolo A, DeLorey, Jennifer, Doyle, Elisabeth G, Johnson, Steven R, Labenski, Matthew T, Morgan, Barry A, O’Donovan, Gary, Sarjeant, Amy A, Skinner, Steven, Thompson, Charles D, Griffin, Sarah T, Westlin, William, White, Kerry F
Published in ACS medicinal chemistry letters (11.04.2013)
Published in ACS medicinal chemistry letters (11.04.2013)
Get full text
Journal Article
Solvent Effects on the Conformation of the Transmembrane Peptide Gramicidin A: Insights from Electrospray Ionization Mass Spectrometry
Bouchard, Mario, Benjamin, Dennis R., Tito, Paula, Robinson, Carol V., Dobson, Christopher M.
Published in Biophysical journal (01.02.2000)
Published in Biophysical journal (01.02.2000)
Get full text
Journal Article
SGN-CD33A in Combination with Cytarabine or Hypomethylating Agents Demonstrates Enhanced Anti-Leukemic Activity in Preclinical Models of AML
Sutherland, May S.K., Yu, Changpu, Anderson, Martha, Emmerton, Kim, Zeng, Weiping, O’Meara, Megan M., Kennedy, Dana A., Ryan, Maureen C., Benjamin, Dennis R.
Published in Blood (06.12.2014)
Published in Blood (06.12.2014)
Get full text
Journal Article
Fucosylation Inhibitor, 2-Fluorofucose, Inhibits NF-κB Activation and Vaso-Occlusion In Transgenic Sickle Mice
Belcher, John D, Chen, Chunsheng, Nguyen, Julia, Okeley, Nicole M., Senter, Peter D., Benjamin, Dennis R., Vercellotti, Gregory M
Published in Blood (15.11.2013)
Published in Blood (15.11.2013)
Get full text
Journal Article