New Pyrrole Inhibitors of Monoamine Oxidase: Synthesis, Biological Evaluation, and Structural Determinants of MAO-A and MAO-B Selectivity
La Regina, Giuseppe, Silvestri, Romano, Artico, Marino, Lavecchia, Antonio, Novellino, Ettore, Befani, Olivia, Turini, Paola, Agostinelli, Enzo
Published in Journal of medicinal chemistry (08.03.2007)
Published in Journal of medicinal chemistry (08.03.2007)
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Inhibition of monoamine oxidases by coumarin-3-acyl derivatives: biological activity and computational study
CHIMENTI, Franco, SECCI, Daniela, BOLASCO, Adriana, CHIMENTI, Paola, GRANESE, Arianna, BEFANI, Olivia, TURINI, Paola, ALCARO, Stefano, ORTUSO, Francesco
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
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Synthesis, Biological Evaluation and 3D-QSAR of 1,3,5-Trisubstituted-4,5- Dihydro-(1H)-Pyrazole Derivatives as Potent and Highly Selective Monoamine Oxidase A Inhibitors
CHIMENTI, Franco, BOLASCO, Adriana, ALCARO, Stefano, ORTUSO, Francesco, LANGER, Thierry, MANNA, Fedele, SECCI, Daniela, CHIMENTI, Paola, GRANESE, Arianna, BEFANI, Olivia, TURINI, Paola, CIRILLI, Roberto, LA TORRE, Francesco
Published in Current medicinal chemistry (01.01.2006)
Published in Current medicinal chemistry (01.01.2006)
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Design, Synthesis, and Biological Activities of Pyrrolylethanoneamine Derivatives, a Novel Class of Monoamine Oxidases Inhibitors
Di Santo, Roberto, Costi, Roberta, Roux, Alessandra, Artico, Marino, Befani, Olivia, Meninno, Tiziana, Agostinelli, Enzo, Palmegiani, Paola, Turini, Paola, Cirilli, Roberto, Ferretti, Rosella, Gallinella, Bruno, La Torre, Francesco
Published in Journal of medicinal chemistry (30.06.2005)
Published in Journal of medicinal chemistry (30.06.2005)
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Journal Article
Synthesis and biochemical evaluation of (R)-5-acyloxymethyl- and (S)-5-acylaminomethyl-3-(1H-pyrrol-1-yl)-2-oxazolidinones as new anti-monoamine oxidase (anti-MAO) agents
Mai, Antonello, Artico, Marino, Valente, Sergio, Cerbara, Ilaria, Befani, Olivia, Vedova, Paola Turini Laura Dalla, Agostinelli, Enzo
Published in ARKIVOC (09.01.2004)
Published in ARKIVOC (09.01.2004)
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Synthesis, structure–activity relationships and molecular modeling studies of new indole inhibitors of monoamine oxidases A and B
La Regina, Giuseppe, Silvestri, Romano, Gatti, Valerio, Lavecchia, Antonio, Novellino, Ettore, Befani, Olivia, Turini, Paola, Agostinelli, Enzo
Published in Bioorganic & medicinal chemistry (15.11.2008)
Published in Bioorganic & medicinal chemistry (15.11.2008)
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Journal Article
Quercetin as the Active Principle of Hypericum hircinum Exerts a Selective Inhibitory Activity against MAO-A: Extraction, Biological Analysis, and Computational Study
Chimenti, F, Cottiglia, F, Bonsignore, L, Casu, L, Casu, M, Floris, C, Secci, D, Bolasco, A, Chimenti, P, Granese, A
Published in Journal of natural products (Washington, D.C.) (01.06.2006)
Published in Journal of natural products (Washington, D.C.) (01.06.2006)
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Journal Article
Synthesis, Molecular Modeling Studies, and Selective Inhibitory Activity against Monoamine Oxidase of 1-Thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)- pyrazole Derivatives
Chimenti, Franco, Maccioni, Elias, Secci, Daniela, Bolasco, Adriana, Chimenti, Paola, Granese, Arianna, Befani, Olivia, Turini, Paola, Alcaro, Stefano, Ortuso, Francesco, Cirilli, Roberto, La Torre, Francesco, Cardia, Maria C, Distinto, Simona
Published in Journal of medicinal chemistry (17.11.2005)
Published in Journal of medicinal chemistry (17.11.2005)
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Journal Article
Synthesis and Selective Inhibitory Activity of 1-Acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole Derivatives against Monoamine Oxidase
Chimenti, Franco, Bolasco, Adriana, Manna, Fedele, Secci, Daniela, Chimenti, Paola, Befani, Olivia, Turini, Paola, Giovannini, Valentina, Mondovì, Bruno, Cirilli, Roberto, La Torre, Francesco
Published in Journal of medicinal chemistry (08.04.2004)
Published in Journal of medicinal chemistry (08.04.2004)
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Journal Article
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N, N′-bis[2-oxo-2 H-benzopyran]-3-carboxamides
Chimenti, Franco, Secci, Daniela, Bolasco, Adriana, Chimenti, Paola, Granese, Arianna, Carradori, Simone, Befani, Olivia, Turini, Paola, Alcaro, Stefano, Ortuso, Francesco
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
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Journal Article
Monoamine Oxidase Isoform-Dependent Tautomeric Influence in the Recognition of 3,5-Diaryl Pyrazole Inhibitors
Chimenti, Franco, Fioravanti, Rossella, Bolasco, Adriana, Manna, Fedele, Chimenti, Paola, Secci, Daniela, Befani, Olivia, Turini, Paola, Ortuso, Francesco, Alcaro, Stefano
Published in Journal of medicinal chemistry (08.02.2007)
Published in Journal of medicinal chemistry (08.02.2007)
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Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives
Manna, Fedele, Chimenti, Franco, Bolasco, Adriana, Secci, Daniela, Bizzarri, Bruna, Befani, Olivia, Turini, Paola, Mondovı̀, Bruno, Alcaro, Stefano, Tafi, Andrea
Published in Bioorganic & medicinal chemistry letters (16.12.2002)
Published in Bioorganic & medicinal chemistry letters (16.12.2002)
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Enzymatic oxidation products of spermine induce greater cytotoxic effects on human multidrug‐resistant colon carcinoma cells (LoVo) than on their wild‐type counterparts
Calcabrini, Annarica, Arancia, Giuseppe, Marra, Manuela, Crateri, Pasqualina, Befani, Olivia, Martone, Alessandro, Agostinelli, Enzo
Published in International journal of cancer (01.05.2002)
Published in International journal of cancer (01.05.2002)
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Journal Article
Simple, Potent, and Selective Pyrrole Inhibitors of Monoamine Oxidase Types A and B
Silvestri, Romano, La Regina, Giuseppe, De Martino, Gabriella, Artico, Marino, Befani, Olivia, Palumbo, Marianna, Agostinelli, Enzo, Turini, Paola
Published in Journal of medicinal chemistry (13.03.2003)
Published in Journal of medicinal chemistry (13.03.2003)
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Journal Article
3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A
Mai, Antonello, Artico, Marino, Esposito, Monica, Sbardella, Gianluca, Massa, Silvio, Befani, Olivia, Turini, Paola, Giovannini, Valentina, Mondovì, Bruno
Published in Journal of medicinal chemistry (14.03.2002)
Published in Journal of medicinal chemistry (14.03.2002)
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Journal Article
Synthesis and Molecular Modelling of Novel Substituted-4,5-dihydro-(1H)-pyrazole Derivatives as Potent and Highly Selective Monoamine Oxidase-A Inhibitors
Chimenti, Franco, Bolasco, Adriana, Manna, Fedele, Secci, Daniela, Chimenti, Paola, Granese, Arianna, Befani, Olivia, Turini, Paola, Alcaro, Stefano, Ortuso, Francesco
Published in Chemical biology & drug design (01.03.2006)
Published in Chemical biology & drug design (01.03.2006)
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Journal Article
Enantiomers of C5-chiral 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives: Analytical and semipreparative HPLC separation, chiroptical properties, absolute configuration, and inhibitory activity against monoamine oxidase
Cirilli, Roberto, Ferretti, Rosella, Gallinella, Bruno, Turchetto, Luciana, Bolasco, Adriana, Secci, Daniela, Chimenti, Paola, Pierini, Marco, Fares, Vincenzo, Befani, Olivia, La Torre, Francesco
Published in Chirality (New York, N.Y.) (2004)
Published in Chirality (New York, N.Y.) (2004)
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Enantiomers of C 5 ‐chiral 1‐acetyl‐3,5‐diphenyl‐4,5‐dihydro‐(1 H )‐pyrazole derivatives: Analytical and semipreparative HPLC separation, chiroptical properties, absolute configuration, and inhibitory activity against monoamine oxidase
Cirilli, Roberto, Ferretti, Rosella, Gallinella, Bruno, Turchetto, Luciana, Bolasco, Adriana, Secci, Daniela, Chimenti, Paola, Pierini, Marco, Fares, Vincenzo, Befani, Olivia, La Torre, Francesco
Published in Chirality (New York, N.Y.) (01.11.2004)
Published in Chirality (New York, N.Y.) (01.11.2004)
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Effect of a plant histaminase on asthmalike reaction induced by inhaled antigen in sensitized guinea pig
Masini, Emanuela, Vannacci, Alfredo, Giannini, Lucia, Befani, Olivia, Nistri, Silvia, Alexandru Mateescu, Mircea, Mannaioni, Pier Francesco, Mondovì, Bruno, Federico, Rodolfo
Published in European journal of pharmacology (19.10.2004)
Published in European journal of pharmacology (19.10.2004)
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Research Article: Synthesis and Molecular Modelling of Novel Substituted-4,5-dihydro-(1H)-pyrazole Derivatives as Potent and Highly Selective Monoamine Oxidase-A Inhibitors
Chimenti, Franco, Bolasco, Adriana, Manna, Fedele, Secci, Daniela, Chimenti, Paola, Granese, Arianna, Befani, Olivia, Turini, Paola, Alcaro, Stefano, Ortuso, Francesco
Published in Chemical biology & drug design (01.03.2006)
Published in Chemical biology & drug design (01.03.2006)
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