Binding Mode and Structure-Activity Relationships around Direct Inhibitors of the Nrf2-Keap1 Complex
Jnoff, Eric, Albrecht, Claudia, Barker, John J., Barker, Oliver, Beaumont, Edward, Bromidge, Steven, Brookfield, Frederick, Brooks, Mark, Bubert, Christian, Ceska, Tom, Corden, Vincent, Dawson, Graham, Duclos, Stephanie, Fryatt, Tara, Genicot, Christophe, Jigorel, Emilie, Kwong, Jason, Maghames, Rosemary, Mushi, Innocent, Pike, Richard, Sands, Zara A., Smith, Myron A., Stimson, Christopher C., Courade, Jean-Philippe
Published in ChemMedChem (01.04.2014)
Published in ChemMedChem (01.04.2014)
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Crystal structure of human peptidylarginine deiminase type VI (PAD6) provides insights into its inactivity
Ranaivoson, Fanomezana M, Bande, Rieke, Cardaun, Isabell, De Riso, Antonio, Gärtner, Annette, Loke, Pui, Reinisch, Christina, Vogirala, Prasuna, Beaumont, Edward
Published in IUCrJ (01.05.2024)
Published in IUCrJ (01.05.2024)
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Validation of a small molecule inhibitor of PDE6D-RAS interaction with favorable anti-leukemic effects
Canovas Nunes, Sara, De Vita, Serena, Anighoro, Andrew, Autelitano, François, Beaumont, Edward, Klingbeil, Pamela, McGuinness, Meaghan, Duvert, Beatrice, Harris, Chad, Yang, Lu, Pokharel, Sheela Pangeni, Chen, Chun-Wei, Ermann, Monika, Williams, David A, Xu, Haiming
Published in Blood cancer journal (New York) (14.04.2022)
Published in Blood cancer journal (New York) (14.04.2022)
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Structural insights into WcbI, a novel polysaccharide-biosynthesis enzyme
Vivoli, Mirella, Ayres, Emily, Beaumont, Edward, Isupov, Michail N, Harmer, Nicholas J
Published in IUCrJ (01.01.2014)
Published in IUCrJ (01.01.2014)
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Development of a Selective Inhibitor of Protein Arginine Deiminase 2
Muth, Aaron, Subramanian, Venkataraman, Beaumont, Edward, Nagar, Mitesh, Kerry, Philip, McEwan, Paul, Srinath, Hema, Clancy, Kathleen, Parelkar, Sangram, Thompson, Paul R
Published in Journal of medicinal chemistry (13.04.2017)
Published in Journal of medicinal chemistry (13.04.2017)
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Small Molecule Inhibition of PDE6D-RAS Interaction Suppresses the Growth of Acute Lymphoblastic Leukemia Cell Lines
Canovas Nunes, Sara, Xu, Haiming, De Vita, Serena, Anighoro, Andrew, Autelitano, Francois, Beaumont, Edward, Klingbeil, Pamela, McGuinness, Meaghan, Duvert, Beatrice, Harris, Chad E., Yang, Lu, Pokharel, Sheela Pangeni, Chen, Chun-Wei David, Ermann, Monika, Williams, David A.
Published in Blood (23.11.2021)
Published in Blood (23.11.2021)
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PAD4의 공유결합성 억제제
BEAUMONT EDWARD JEAN, LOKE PUI LENG, KERRY PHILIP STEPHEN, KUMARAVEL GNANASAMBANDAM, LECCI CRISTINA, PALFREY JORDAN JOHN, DEVRAJ RAJESH, NORTH CARL, MENICONI MIRCO, TYE HEATHER
Year of Publication 03.04.2019
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Year of Publication 03.04.2019
Patent
Synchronous Photoinitiation of Endothelial NO Synthase Activity by a Nanotrigger Targeted at Its NADPH Site
Beaumont, Edward, Lambry, Jean-Christophe, Gautier, Clément, Robin, Anne-Claire, Gmouh, Said, Berka, Vladimir, Tsai, Ah-Lim, Blanchard-Desce, Mireille, Slama-Schwok, Anny
Published in Journal of the American Chemical Society (21.02.2007)
Published in Journal of the American Chemical Society (21.02.2007)
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Journal Article
PAD4의 헤테로아릴 억제제
KERRY PHILLIP STEPHEN, LECCI CRISTINA, DEVRAJ RAJESH, MENICONI MIRCO, PALFREY JORDAN, MONCK NAT, BEAUMONT EDWARD, GADOULEAU ELISE, GLEAVE LAURA, PAPADOPOULOS KOSTAS, ATTON HOLLY, KUMARAVEL GNANASAMBANDAM, WOODS PHILIP A, TYE HEATHER
Year of Publication 08.10.2018
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Year of Publication 08.10.2018
Patent
Inside Cover: Binding Mode and Structure-Activity Relationships around Direct Inhibitors of the Nrf2-Keap1 Complex (ChemMedChem 4/2014)
Jnoff, Eric, Albrecht, Claudia, Barker, John J., Barker, Oliver, Beaumont, Edward, Bromidge, Steven, Brookfield, Frederick, Brooks, Mark, Bubert, Christian, Ceska, Tom, Corden, Vincent, Dawson, Graham, Duclos, Stephanie, Fryatt, Tara, Genicot, Christophe, Jigorel, Emilie, Kwong, Jason, Maghames, Rosemary, Mushi, Innocent, Pike, Richard, Sands, Zara A., Smith, Myron A., Stimson, Christopher C., Courade, Jean-Philippe
Published in ChemMedChem (01.04.2014)
Published in ChemMedChem (01.04.2014)
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Journal Article
PAD4의 비시클릭 억제제
PARROTT SHELLEY, BROMBRIDGE STEVE, LECCI CRISTINA, LOKE PUI, COOPER SOPHIE, DEVRAJ RAJESH, BOWLES LEE, NORTH CARL, MENICONI MIRCO, PALFREY JORDAN, MONCK NAT, PARKER MICHAEL F, BEAUMONT EDWARD, GADOULEAU ELISE, KOTEY ADRIAN, GLEAVE LAURA, RIDGILL MARK, KUMARAVEL GNANASAMBANDAM, TYE HEATHER, KRULLE THOMAS, KERRY PHILIP
Year of Publication 04.09.2018
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Year of Publication 04.09.2018
Patent
NO Formation by Neuronal NO-Synthase can be Controlled by Ultrafast Electron Injection from a Nanotrigger
Beaumont, Edward, Lambry, Jean-Christophe, Blanchard-Desce, Mireille, Martasek, Pavel, Panda, Satya P, van Faassen, Ernst E.H, Brochon, Jean-Claude, Deprez, Eric, Slama-Schwok, Anny
Published in Chembiochem : a European journal of chemical biology (02.03.2009)
Published in Chembiochem : a European journal of chemical biology (02.03.2009)
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Journal Article
O46. Photoinduced electron transfer from a novel nanotrigger addressed to the NADPH site within the endothelial NO-synthase to the flavin moieties of the protein
Beaumont, Edward, Robin, Anne-Claire, Berka, Vladimir, Tsai, Ah-Lim, Blanchard-Desce, Mireille, Lambry, Jean-Christophe, Slama-Schwok, Anny
Published in Nitric oxide (01.06.2006)
Published in Nitric oxide (01.06.2006)
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Journal Article
Photoinduced electron transfer from a novel nanotrigger addressed to the NADPH site within the endothelial NO-synthase to the flavin moieties of the protein
Beaumont, Edward, Robin, Anne-Claire, Berka, Vladimir, Tsai, Ah-Lim, Blanchard-Desce, Mireille, Lambry, Jean-Christophe, Slama-Schwok, Anny
Published in Nitric oxide (2006)
Published in Nitric oxide (2006)
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Journal Article
Heteroaryl inhibitors of PAD4
Papadopoulos, Kostas, Gadouleau, Elise, Monck, Nat, Beaumont, Edward, Palfrey, Jordan, Tye, Heather, Meniconi, Mirco, Woods, Philip A, Gleave, Laura, Kerry, Philip Stephen, Atton, Holly, Devraj, Rajesh, Kumaravel, Gnanasambandam, Lecci, Cristina
Year of Publication 13.02.2024
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Year of Publication 13.02.2024
Patent