Preparation of Unsymmetrical Sulfonylureas from N,N‘-Sulfuryldiimidazoles
Beaudoin, Serge, Kinsey, Kenneth E, Burns, James F
Published in Journal of organic chemistry (10.01.2003)
Published in Journal of organic chemistry (10.01.2003)
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Journal Article
Asymmetric conjugate additions of chiral allyl- and crotylphosphonamide anions to .alpha.,.beta.-unsaturated carbonyl compounds: highly stereocontrolled access to vicinally substituted carbon centers and chemically asymmetrized chirons
Hanessian, Stephen, Gomtsyan, Arthur, Payne, Andrew, Herve, Yolande, Beaudoin, Serge
Published in Journal of organic chemistry (01.09.1993)
Published in Journal of organic chemistry (01.09.1993)
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Journal Article
Discovery of Clinical Candidate 4-[2-(5-Amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-1,3-thiazol-4-ylbenzenesulfonamide (PF-05089771): Design and Optimization of Diaryl Ether Aryl Sulfonamides as Selective Inhibitors of Na(V)1.7
Swain, Nigel. A., Batchelor, Dave, Beaudoin, Serge, Bechle, Bruce M., Bradley, Paul A., Brown, Alan D., Brown, Bruce, Butcher, Kent J., Butt, Richard P., Chapman, Mark L., Denton, Stephen, Ellis, David, Galan, Sebastien R. G., Gaulier, Steven M., Greener, Ben S., de Groot, Marcel J., Glossop, Mel S., Gurrell, Ian K., Hannan, Jo, Johnson, Matthew S., Lin, Zhixin, Markworth, Christopher J., Marron, Brian E., Milan, David S., Nakaawa, Shoko, Pike, Andy, Printzephoff, David, Rawson, David J., Ransley, Sarah J., Reister, Steven M., Sasaki, Kosuke, Storer, R. Ian, Stupple, Paul A., West, Christopher W.
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Discovery of Clinical Candidate 4‑[2-(5-Amino‑1H‑pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro‑N‑1,3-thiazol-4-ylbenzenesulfonamide (PF-05089771): Design and Optimization of Diaryl Ether Aryl Sulfonamides as Selective Inhibitors of NaV1.7
Swain, Nigel. A, Batchelor, Dave, Beaudoin, Serge, Bechle, Bruce M, Bradley, Paul A, Brown, Alan D, Brown, Bruce, Butcher, Ken J, Butt, Richard P, Chapman, Mark L, Denton, Stephen, Ellis, David, Galan, Sebastien R. G, Gaulier, Steven M, Greener, Ben S, de Groot, Marcel J, Glossop, Mel S, Gurrell, Ian K, Hannam, Jo, Johnson, Matthew S, Lin, Zhixin, Markworth, Christopher J, Marron, Brian E, Millan, David S, Nakagawa, Shoko, Pike, Andy, Printzenhoff, David, Rawson, David J, Ransley, Sarah J, Reister, Steven M, Sasaki, Kosuke, Storer, R. Ian, Stupple, Paul A, West, Christopher W
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Discovery of Clinical Candidate 4-[2-(5-Amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-1,3-thiazol-4-ylbenzenesulfonamide (PF-05089771): Design and Optimization of Diaryl Ether Aryl Sulfonamides as Selective Inhibitors of Na V 1.7
Swain, Nigel A, Batchelor, Dave, Beaudoin, Serge, Bechle, Bruce M, Bradley, Paul A, Brown, Alan D, Brown, Bruce, Butcher, Ken J, Butt, Richard P, Chapman, Mark L, Denton, Stephen, Ellis, David, Galan, Sebastien R G, Gaulier, Steven M, Greener, Ben S, de Groot, Marcel J, Glossop, Mel S, Gurrell, Ian K, Hannam, Jo, Johnson, Matthew S, Lin, Zhixin, Markworth, Christopher J, Marron, Brian E, Millan, David S, Nakagawa, Shoko, Pike, Andy, Printzenhoff, David, Rawson, David J, Ransley, Sarah J, Reister, Steven M, Sasaki, Kosuke, Storer, R Ian, Stupple, Paul A, West, Christopher W
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Aryl sulfonamido indane inhibitors of the Kv1.5 ion channel
Gross, Michael F., Beaudoin, Serge, McNaughton-Smith, Grant, Amato, George S., Castle, Neil A., Huang, Christine, Zou, Anruo, Yu, Weifeng
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
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Journal Article
SULFONAMIDE DERIVATIVES
MILLAN DAVID SIMON, BEAUDOIN SERGE, MARRON BRIAN EDWARD, REISTER STEVEN MICHAEL, ZHOU SHULAN, SASAKI KOSUKE, LAUFER SWEILER MICHAEL CHRISTOPHER, RAWSON DAVID JAMES, MARKWORTH CHRISTOPHER JOHN, WEST CHRISTOPHER WILLIAM, SWAIN NIGEL ALAN, STUPPLE PAUL ANTHONY, STORER ROBERT IAN
Year of Publication 22.09.2011
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Year of Publication 22.09.2011
Patent
Asymmetric dihydroxylation of olefins with a simple chiral ligand
Hanessian, Stephen, Meffre, Patrick, Girard, Mario, Beaudoin, Serge, Sanceau, Jean Yves, Bennani, Youssef
Published in Journal of organic chemistry (01.04.1993)
Published in Journal of organic chemistry (01.04.1993)
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Journal Article
Stereoselective synthesis of long-chain polyols by sequential homologation of enals with nonracemic .gamma.-silyloxy allylic stannanes and directed hydroxylation
Marshall, James A, Beaudoin, Serge, Lewinski, Krzysztof
Published in Journal of organic chemistry (01.10.1993)
Published in Journal of organic chemistry (01.10.1993)
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Journal Article
Sulfonamide derivatives
BEAUDOIN SERGE, MARKWORTH CHRISTOPHER JOHN, LAUFERSWEILER MICHAEL CHRISTOPHER
Year of Publication 31.12.2013
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Year of Publication 31.12.2013
Patent
Sodium Channel Inhibitors
BEAUDOIN SERGE, JOHNSON MATTHEW SCOTT, MARRON BRIAN EDWARD, SUTO MARK J
Year of Publication 04.12.2014
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Year of Publication 04.12.2014
Patent
Sodium channel inhibitors
BEAUDOIN SERGE, JOHNSON MATTHEW SCOTT, SUTO MARK J, MARRON BRAIN EDWARD
Year of Publication 07.10.2014
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Year of Publication 07.10.2014
Patent
SODIUM CHANNEL INHIBITORS
JOHNSON, MATTHEW SCOTT, MARRON, BRIAN EDWARD, SUTO, MARK J, BEAUDOIN, SERGE
Year of Publication 10.09.2014
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Year of Publication 10.09.2014
Patent
derivados de sulfonamida
DAVID JAMES RAWSON, PAUL ANTHONY STUPPLE, DAVID SIMON MILLAN, ROBERT IAN STORER, SERGE BEAUDOIN, MICHAEL CHRISTOPHER LAUFERSWEILER, CRHISTOPHER JOHN MARKWORTH, BRIAN EDWARD MARRON, CHRISTOPHER WILLIAM WEST, SHULAN ZHOU, STEVEN MICHAEL REISTER, NIGEL ALAN SWAIN, KOSUKE SASAKI
Year of Publication 01.11.2016
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Year of Publication 01.11.2016
Patent