Relaxin Reverses Cardiac and Renal Fibrosis in Spontaneously Hypertensive Rats
Lekgabe, Edna D, Kiriazis, Helen, Zhao, Chongxin, Xu, Qi, Moore, Xiao Lei, Su, Yidan, Bathgate, Ross A.D, Du, Xiao-Jun, Samuel, Chrishan S
Published in Hypertension (Dallas, Tex. 1979) (01.08.2005)
Published in Hypertension (Dallas, Tex. 1979) (01.08.2005)
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The A-chain of Human Relaxin Family Peptides Has Distinct Roles in the Binding and Activation of the Different Relaxin Family Peptide Receptors
Hossain, Mohammed Akhter, Rosengren, K. Johan, Haugaard-Jönsson, Linda M., Zhang, Soude, Layfield, Sharon, Ferraro, Tania, Daly, Norelle L., Tregear, Geoffrey W., Wade, John D., Bathgate, Ross A.D.
Published in The Journal of biological chemistry (20.06.2008)
Published in The Journal of biological chemistry (20.06.2008)
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Expression of the Insulin-Like Peptide 3 (INSL3) Hormone-Receptor (LGR8) System in the Testis
Anand-Ivell, Ravinder J.K, Relan, Vandana, Balvers, Marga, Coiffec-Dorval, Isabelle, Fritsch, Martin, Bathgate, Ross A.D, Ivell, Richard
Published in Biology of reproduction (01.05.2006)
Published in Biology of reproduction (01.05.2006)
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Solution Structure and Characterization of the LGR8 Receptor Binding Surface of Insulin-like Peptide 3
Rosengren, K. Johan, Zhang, Suode, Lin, Feng, Daly, Norelle L., Scott, Daniel J., Hughes, Richard A., Bathgate, Ross A.D., Craik, David J., Wade, John D.
Published in The Journal of biological chemistry (22.09.2006)
Published in The Journal of biological chemistry (22.09.2006)
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Journal Article
Structure of the R3/I5 Chimeric Relaxin Peptide, a Selective GPCR135 and GPCR142 Agonist
Haugaard-Jönsson, Linda M., Hossain, Mohammed Akhter, Daly, Norelle L., Bathgate, Ross A.D., Wade, John D., Craik, David J., Rosengren, K. Johan
Published in The Journal of biological chemistry (29.08.2008)
Published in The Journal of biological chemistry (29.08.2008)
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Journal Article
Splice variants of the relaxin and INSL3 receptors reveal unanticipated molecular complexity
Muda, Marco, He, Chaomei, Martini, Paolo G.V., Ferraro, Tania, Layfield, Sharon, Taylor, Deanne, Chevrier, Colette, Schweickhardt, Rene, Kelton, Christie, Ryan, Peter L., Bathgate, Ross A.D.
Published in Molecular human reproduction (01.08.2005)
Published in Molecular human reproduction (01.08.2005)
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Journal Article
The relaxin receptor as a therapeutic target – perspectives from evolution and drug targeting
Bathgate, Ross A.D., Kocan, Martina, Scott, Daniel J., Hossain, M. Akhter, Good, Sara V., Yegorov, Sergey, Bogerd, Jan, Gooley, Paul R.
Published in Pharmacology & therapeutics (Oxford) (01.07.2018)
Published in Pharmacology & therapeutics (Oxford) (01.07.2018)
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Relaxin requires the angiotensin II type 2 receptor to abrogate renal interstitial fibrosis
Chow, Bryna S. Man, Kocan, Martina, Bosnyak, Sanja, Sarwar, Mohsin, Wigg, Belinda, Jones, Emma S., Widdop, Robert E., Summers, Roger J., Bathgate, Ross A.D., Hewitson, Tim D., Samuel, Chrishan S.
Published in Kidney international (01.07.2014)
Published in Kidney international (01.07.2014)
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A Novel Ultra-Stable, Monomeric Green Fluorescent Protein For Direct Volumetric Imaging of Whole Organs Using CLARITY
Scott, Daniel J., Gunn, Natalie J., Yong, Kelvin J., Wimmer, Verena C., Veldhuis, Nicholas A., Challis, Leesa M., Haidar, Mouna, Petrou, Steven, Bathgate, Ross A. D., Griffin, Michael D. W.
Published in Scientific reports (12.01.2018)
Published in Scientific reports (12.01.2018)
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Spawning induction of the high-value white teatfish sea cucumber, Holothuria fuscogilva, using recombinant relaxin-like gonad stimulating peptide (RGP)
Nocillado, Josephine, Duy, Nguyen Dinh Quang, Chieu, Hoang Dinh, Turner, Luke, Bathgate, Ross A.D., Wang, Tianfang, Hossain, Mohammed Akhter, Hung, Nguyen Van, Ninh, Nguyen Huu, Cummins, Scott F., Elizur, Abigail
Published in Aquaculture (30.01.2022)
Published in Aquaculture (30.01.2022)
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Journal Article
Ligands selectively tune the local and global motions of neurotensin receptor 1 (NTS1)
Bumbak, Fabian, Pons, Miquel, Inoue, Asuka, Paniagua, Juan Carlos, Yan, Fei, Wu, Hongwei, Robson, Scott A., Bathgate, Ross A.D., Scott, Daniel J., Gooley, Paul R., Ziarek, Joshua J.
Published in Cell reports (Cambridge) (31.01.2023)
Published in Cell reports (Cambridge) (31.01.2023)
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Probing the correlation between ligand efficacy and conformational diversity at the α1A-adrenoreceptor reveals allosteric coupling of its microswitches
Wu, Feng-Jie, Williams, Lisa M., Abdul-Ridha, Alaa, Gunatilaka, Avanka, Vaid, Tasneem M., Kocan, Martina, Whitehead, Alice R., Griffin, Michael D.W., Bathgate, Ross A.D., Scott, Daniel J., Gooley, Paul R.
Published in The Journal of biological chemistry (22.05.2020)
Published in The Journal of biological chemistry (22.05.2020)
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Optimization and 13CH3 methionine labeling of a signaling competent neurotensin receptor 1 variant for NMR studies
Bumbak, Fabian, Keen, Alastair C., Gunn, Natalie J., Gooley, Paul R., Bathgate, Ross A.D., Scott, Daniel J.
Published in Biochimica et biophysica acta. Biomembranes (01.06.2018)
Published in Biochimica et biophysica acta. Biomembranes (01.06.2018)
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The single-chain relaxin mimetic, B7-33, maintains the cardioprotective effects of relaxin and more rapidly reduces left ventricular fibrosis compared to perindopril in an experimental model of cardiomyopathy
Alam, Fariha, Gaspari, Tracey A., Kemp-Harper, Barbara K., Low, Edward, Aw, Aaron, Ferens, Dorota, Spizzo, Iresha, Jefferis, Ann-Maree, Praveen, Praveen, Widdop, Robert E., Bathgate, Ross A.D., Hossain, Mohammed Akhter, Samuel, Chrishan S.
Published in Biomedicine & pharmacotherapy (01.04.2023)
Published in Biomedicine & pharmacotherapy (01.04.2023)
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Journal Article
Minimization of Human Relaxin-3 Leading to High-Affinity Analogues with Increased Selectivity for Relaxin-Family Peptide 3 Receptor (RXFP3) over RXFP1
Shabanpoor, Fazel, Akhter Hossain, Mohammad, Ryan, Philip J, Belgi, Alessia, Layfield, Sharon, Kocan, Martina, Zhang, Suode, Samuel, Chrishan S, Gundlach, Andrew L, Bathgate, Ross A.D, Separovic, Frances, Wade, John D
Published in Journal of medicinal chemistry (23.02.2012)
Published in Journal of medicinal chemistry (23.02.2012)
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Distribution of relaxin-3 and RXFP3 within arousal, stress, affective, and cognitive circuits of mouse brain
Smith, Craig M., Shen, Pei-Juan, Banerjee, Avantika, Bonaventure, Pascal, Ma, Sherie, Bathgate, Ross A.D., Sutton, Steven W., Gundlach, Andrew L.
Published in Journal of comparative neurology (1911) (01.10.2010)
Published in Journal of comparative neurology (1911) (01.10.2010)
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High-Throughput Screening Campaign Identified a Potential Small Molecule RXFP3/4 Agonist
Lin, Guangyao, Feng, Yang, Cai, Xiaoqing, Zhou, Caihong, Shao, Lijun, Chen, Yan, Chen, Linhai, Liu, Qing, Zhou, Qingtong, Bathgate, Ross A D, Yang, Dehua, Wang, Ming-Wei
Published in Molecules (Basel, Switzerland) (11.12.2021)
Published in Molecules (Basel, Switzerland) (11.12.2021)
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