A Global Model for Forecasting Political Instability
Goldstone, Jack A., Bates, Robert H., Epstein, David L., Gurr, Ted Robert, Lustik, Michael B., Marshall, Monty G., Ulfelder, Jay, Woodward, Mark
Published in American journal of political science (01.01.2010)
Published in American journal of political science (01.01.2010)
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Journal Article
αβ,α′β′-Diepoxyketones are mechanism-based inhibitors of nucleophilic cysteine enzymes
de Munnik, Mariska, Lithgow, Jasper, Brewitz, Lennart, Christensen, Kirsten E, Bates, Robert H, Rodriguez-Miquel, Beatriz, Schofield, Christopher J
Published in Chemical communications (Cambridge, England) (26.10.2023)
Published in Chemical communications (Cambridge, England) (26.10.2023)
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Journal Article
Improved BM212 MmpL3 inhibitor analogue shows efficacy in acute murine model of tuberculosis infection
Poce, Giovanna, Bates, Robert H, Alfonso, Salvatore, Cocozza, Martina, Porretta, Giulio Cesare, Ballell, Lluís, Rullas, Joaquin, Ortega, Fátima, De Logu, Alessandro, Agus, Emanuela, La Rosa, Valentina, Pasca, Maria Rosalia, De Rossi, Edda, Wae, Baojie, Franzblau, Scott G, Manetti, Fabrizio, Botta, Maurizio, Biava, Mariangela
Published in PloS one (21.02.2013)
Published in PloS one (21.02.2013)
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Journal Article
Democratic Transitions
Epstein, David L., Bates, Robert, Goldstone, Jack, Kristensen, Ida, O'Halloran, Sharyn
Published in American journal of political science (01.07.2006)
Published in American journal of political science (01.07.2006)
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Journal Article
Identification of KasA as the cellular target of an anti-tubercular scaffold
Abrahams, Katherine A., Chung, Chun-wa, Ghidelli-Disse, Sonja, Rullas, Joaquín, Rebollo-López, María José, Gurcha, Sudagar S., Cox, Jonathan A. G., Mendoza, Alfonso, Jiménez-Navarro, Elena, Martínez-Martínez, María Santos, Neu, Margarete, Shillings, Anthony, Homes, Paul, Argyrou, Argyrides, Casanueva, Ruth, Loman, Nicholas J., Moynihan, Patrick J., Lelièvre, Joël, Selenski, Carolyn, Axtman, Matthew, Kremer, Laurent, Bantscheff, Marcus, Angulo-Barturen, Iñigo, Izquierdo, Mónica Cacho, Cammack, Nicholas C., Drewes, Gerard, Ballell, Lluis, Barros, David, Besra, Gurdyal S., Bates, Robert H.
Published in Nature communications (01.09.2016)
Published in Nature communications (01.09.2016)
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Journal Article
Release of 50 new, drug-like compounds and their computational target predictions for open source anti-tubercular drug discovery
Rebollo-Lopez, María Jose, Lelièvre, Joël, Alvarez-Gomez, Daniel, Castro-Pichel, Julia, Martínez-Jiménez, Francisco, Papadatos, George, Kumar, Vinod, Colmenarejo, Gonzalo, Mugumbate, Grace, Hurle, Mark, Barroso, Vanessa, Young, Rob J, Martinez-Hoyos, María, González del Río, Rubén, Bates, Robert H, Lopez-Roman, Eva Maria, Mendoza-Losana, Alfonso, Brown, James R, Alvarez-Ruiz, Emilio, Marti-Renom, Marc A, Overington, John P, Cammack, Nicholas, Ballell, Lluís, Barros-Aguire, David
Published in PloS one (07.12.2015)
Published in PloS one (07.12.2015)
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Journal Article
High-throughput screen with the l,d-transpeptidase LdtMt2 of Mycobacterium tuberculosis reveals novel classes of covalently reacting inhibitors
de Munnik, Mariska, Lang, Pauline A, De Dios Anton, Francisco, Cacho, Mónica, Bates, Robert H, Brem, Jürgen, Beatriz Rodríguez Miquel, Schofield, Christopher J
Published in Chemical science (Cambridge) (30.05.2023)
Published in Chemical science (Cambridge) (30.05.2023)
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Journal Article
Searching for New Leads for Tuberculosis: Design, Synthesis, and Biological Evaluation of Novel 2‑Quinolin-4-yloxyacetamides
Pitta, Eleni, Rogacki, Maciej K, Balabon, Olga, Huss, Sophie, Cunningham, Fraser, Lopez-Roman, Eva Maria, Joossens, Jurgen, Augustyns, Koen, Ballell, Lluis, Bates, Robert H, Van der Veken, Pieter
Published in Journal of medicinal chemistry (28.07.2016)
Published in Journal of medicinal chemistry (28.07.2016)
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Journal Article
High-throughput screen with the l,d-transpeptidase Ldt Mt2 of Mycobacterium tuberculosis reveals novel classes of covalently reacting inhibitors
de Munnik, Mariska, Lang, Pauline A, De Dios Anton, Francisco, Cacho, Mónica, Bates, Robert H, Brem, Jürgen, Rodríguez Miquel, Beatriz, Schofield, Christopher J
Published in Chemical science (Cambridge) (05.07.2023)
Published in Chemical science (Cambridge) (05.07.2023)
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Journal Article
Optimization of Hydantoins as Potent Antimycobacterial Decaprenylphosphoryl-β‑d‑Ribose Oxidase (DprE1) Inhibitors
Balabon, Olga, Pitta, Eleni, Rogacki, Maciej K, Meiler, Eugenia, Casanueva, Ruth, Guijarro, Laura, Huss, Sophie, Lopez-Roman, Eva Maria, Santos-Villarejo, Ángel, Augustyns, Koen, Ballell, Lluis, Aguirre, David Barros, Bates, Robert H, Cunningham, Fraser, Cacho, Monica, Van der Veken, Pieter
Published in Journal of medicinal chemistry (28.05.2020)
Published in Journal of medicinal chemistry (28.05.2020)
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Journal Article
A service evaluation of passive remote monitoring technology for patients in a high-secure forensic psychiatric hospital: a qualitative study
Dewa, Lindsay H, Broyd, Josephine, Hira, Rita, Dudley, Alison, Hafferty, Jonathan D, Bates, Robert, Aylin, Paul
Published in BMC psychiatry (14.12.2023)
Published in BMC psychiatry (14.12.2023)
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Journal Article
Identification and Profiling of HydantoinsA Novel Class of Potent Antimycobacterial DprE1 Inhibitors
Rogacki, Maciej K, Pitta, Eleni, Balabon, Olga, Huss, Sophie, Lopez-Roman, Eva Maria, Argyrou, Argyrides, Blanco-Ruano, Delia, Cacho, Monica, Vande Velde, Christophe M. L, Augustyns, Koen, Ballell, Lluis, Barros, David, Bates, Robert H, Cunningham, Fraser, Van der Veken, Pieter
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
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Journal Article
The Tuberculosis Drug Accelerator at year 10: what have we learned?
Aldridge, Bree B., Barros-Aguirre, David, Barry, Clifton E., Bates, Robert H., Berthel, Steven J., Boshoff, Helena I., Chibale, Kelly, Chu, Xin-Jie, Cooper, Christopher B., Dartois, Véronique, Duncan, Ken, Fotouhi, Nader, Gusovsky, Fabian, Hipskind, Philip A., Kempf, Dale J., Lelièvre, Joël, Lenaerts, Anne J., McNamara, Case W., Mizrahi, Valerie, Nathan, Carl, Olsen, David B., Parish, Tanya, Petrassi, H. Michael, Pym, Alexander, Rhee, Kyu Y., Robertson, Gregory T., Rock, Jeremy Michael, Rubin, Eric J., Russell, Betsy, Russell, David G., Sacchettini, James C., Schnappinger, Dirk, Schrimpf, Michael, Upton, Anna M., Warner, Peter, Wyatt, Paul Graham, Yuan, Ying
Published in Nature medicine (01.08.2021)
Published in Nature medicine (01.08.2021)
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Journal Article
GSK2556286 Is a Novel Antitubercular Drug Candidate Effective In Vivo with the Potential To Shorten Tuberculosis Treatment
Nuermberger, Eric L, Martínez-Martínez, Maria Santos, Sanz, Olalla, Urones, Beatriz, Esquivias, Jorge, Soni, Heena, Tasneen, Rokeya, Tyagi, Sandeep, Li, Si-Yang, Converse, Paul J, Boshoff, Helena I, Robertson, Gregory T, Besra, Gurdyal S, Abrahams, Katherine A, Upton, Anna M, Mdluli, Khisimuzi, Boyle, Gary W, Turner, Sam, Fotouhi, Nader, Cammack, Nicholas C, Siles, Juan Miguel, Alonso, Marta, Escribano, Jaime, Lelievre, Joel, Rullas-Trincado, Joaquin, Pérez-Herrán, Esther, Bates, Robert H, Maher-Edwards, Gareth, Barros, David, Ballell, Lluís, Jiménez, Elena
Published in Antimicrobial agents and chemotherapy (21.06.2022)
Published in Antimicrobial agents and chemotherapy (21.06.2022)
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Journal Article
Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target
Wilson, Caroline, Ray, Peter, Zuccotto, Fabio, Hernandez, Jorge, Aggarwal, Anup, Mackenzie, Claire, Caldwell, Nicola, Taylor, Malcolm, Huggett, Margaret, Mathieson, Michael, Murugesan, Dinakaran, Smith, Alasdair, Davis, Susan, Cocco, Mattia, Parai, Maloy K, Acharya, Arjun, Tamaki, Fabio, Scullion, Paul, Epemolu, Ola, Riley, Jennifer, Stojanovski, Laste, Lopez-Román, Eva Maria, Torres-Gómez, Pedro Alfonso, Toledo, Ana Maria, Guijarro-Lopez, Laura, Camino, Isabel, Engelhart, Curtis A, Schnappinger, Dirk, Massoudi, Lisa M, Lenaerts, Anne, Robertson, Gregory T, Walpole, Chris, Matthews, David, Floyd, David, Sacchettini, James C, Read, Kevin D, Encinas, Lourdes, Bates, Robert H, Green, Simon R, Wyatt, Paul G
Published in Journal of medicinal chemistry (13.01.2022)
Published in Journal of medicinal chemistry (13.01.2022)
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Journal Article
Testing tuberculosis drug efficacy in a zebrafish high-throughput translational medicine screen
Ordas, Anita, Raterink, Robert-Jan, Cunningham, Fraser, Jansen, Hans J, Wiweger, Malgorzata I, Jong-Raadsen, Susanne, Bos, Sabine, Bates, Robert H, Barros, David, Meijer, Annemarie H, Vreeken, Rob J, Ballell-Pages, Lluís, Dirks, Ron P, Hankemeier, Thomas, Spaink, Herman P
Published in Antimicrobial agents and chemotherapy (01.02.2015)
Published in Antimicrobial agents and chemotherapy (01.02.2015)
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Journal Article
Bosutinib prevents vascular leakage by reducing focal adhesion turnover and reinforcing junctional integrity
Botros, Liza, Pronk, Manon C A, Juschten, Jenny, Liddle, John, Morsing, Sofia K H, van Buul, Jaap D, Bates, Robert H, Tuinman, Pieter R, van Bezu, Jan S M, Huveneers, Stephan, Bogaard, Harm Jan, van Hinsbergh, Victor W M, Hordijk, Peter L, Aman, Jurjan
Published in Journal of cell science (01.05.2020)
Published in Journal of cell science (01.05.2020)
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Journal Article