Rational design, synthesis, and structure–activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors
Basu, Sujay, Prathipati, Philip, Thorat, Sachin, Ansari, Shariq, Patel, Meena, Jain, Vaibhav, Jinugu, Ramana R., Niranjan, Sanjay, De, Siddhartha, Reddy, Satyanarayana
Published in Bioorganic & medicinal chemistry (01.01.2017)
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A(2B) adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B. Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R., Palle, Venkata P., Chugh, Anita, Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B. Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R., Palle, Venkata P., Chugh, Anita, Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A(2A) Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A., Thorat, Sachin, Shejul, Yogesh D., Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S., Meru, Ashwinkumar V., De, Siddhartha, Bhamidipati, Ravi K., Rouduri, Sreekanth R., Palle, Venkata P., Chug, Anita, Mookhtiar, Kasim A.
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia
Deshpande, Anil M., Bhuniya, Debnath, De, Siddhartha, Dave, Bhavesh, Vyavahare, Vinod P., Kurhade, Santosh H., Kandalkar, Sachin R., Naik, Keshav P., Kobal, Balasaheb S., Kaduskar, Rahul D., Basu, Sujay, Jain, Vaibhav, Patil, Pratima, Chaturvedi Joshi, Sandhya, Bhat, Ganesh, Raje, Amol A., Reddy, Satyanarayana, Gundu, Jayasagar, Madgula, Vamsi, Tambe, Suhas, Shitole, Prasad, Umrani, Dhananjay, Chugh, Anita, Palle, Venkata P., Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (16.06.2017)
Published in European journal of medicinal chemistry (16.06.2017)
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Journal Article
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A(1) receptor antagonists and their biological evaluation
Koul, Summon, Ramdas, Vidya, Barawkar, Dinesh A., Waman, Yogesh B., Prasad, Neela, Madadi, Santosh Kumar, Shejul, Yogesh D., Bonagiri, Rajesh, Basu, Sujay, Menon, Suraj, Reddy, Srinivasa B., Chaturvedi, Sandhya, Chennamaneni, Srinivas Rao, Bedse, Gaurav, Thakare, Rhishikesh, Gundu, Jayasagar, Chaudhary, Sumit, De, Siddhartha, Meru, Ashwinkumar V., Palle, Venkata, Chugh, Anita, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
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Journal Article
삼환식 화합물, 삼환식 화합물을 포함하는 조성물 및 이의 의약적 용도
PATEL MEENA, BONAGIRI RAJESH, MOOKHTIAR KASIM, KULKARNI BHEEMASHANKAR, BASU SUJAY, KHOSE GORAKSHA, BARAWKAR DINESH, SHEJUL YOGESH, THORAT SACHIN, PANMAND ANIL
Year of Publication 11.09.2020
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Year of Publication 11.09.2020
Patent
Revisiting glitazars: Thiophene substituted oxazole containing α-ethoxy phenylpropanoic acid derivatives as highly potent PPARα/γ dual agonists devoid of adverse effects in rodents
Raval, Preeti, Jain, Mukul, Goswami, Amitgiri, Basu, Sujay, Gite, Archana, Godha, Atul, Pingali, Harikishore, Raval, Saurin, Giri, Suresh, Suthar, Dinesh, Shah, Maanan, Patel, Pankaj
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A 2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
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Journal Article
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A 1 receptor antagonists and their biological evaluation
Koul, Summon, Ramdas, Vidya, Barawkar, Dinesh A, Waman, Yogesh B, Prasad, Neela, Madadi, Santosh Kumar, Shejul, Yogesh D, Bonagiri, Rajesh, Basu, Sujay, Menon, Suraj, Reddy, Srinivasa B, Chaturvedi, Sandhya, Chennamaneni, Srinivas Rao, Bedse, Gaurav, Thakare, Rhishikesh, Gundu, Jayasagar, Chaudhary, Sumit, De, Siddhartha, Meru, Ashwinkumar V, Palle, Venkata, Chugh, Anita, Mookhtiar, Kasim A
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
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Journal Article
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation
Koul, Summon, Ramdas, Vidya, Barawkar, Dinesh A., Waman, Yogesh B., Prasad, Neela, Madadi, Santosh Kumar, Shejul, Yogesh D., Bonagiri, Rajesh, Basu, Sujay, Menon, Suraj, Reddy, Srinivasa B., Chaturvedi, Sandhya, Chennamaneni, Srinivas Rao, Bedse, Gaurav, Thakare, Rhishikesh, Gundu, Jayasagar, Chaudhary, Sumit, De, Siddhartha, Meru, Ashwinkumar V., Palle, Venkata, Chugh, Anita, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
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Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A 2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors
Basu, Sujay, Prasad, Uppuleti Viplava, Barawkar, Dinesh A., De, Siddhartha, Palle, Venkata P., Menon, Suraj, Patel, Meena, Thorat, Sachin, Singh, Umesh P., Sarma, Koushik Das, Waman, Yogesh, Niranjan, Sanjay, Pathade, Vishal, Gaur, Ashwani, Reddy, Satyanarayana, Ansari, Shariq
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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Journal Article
Discovery of Potent and Selective A(2A) Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Naykodi, Minakshi, Shejul, Yogesh D., Patel, Meena, Thorat, Sachin, Panmand, Anil, Kashinath, K., Bonagiri, Rajesh, Prasad, Vandna, Bhat, Ganesh, Quraishi, Azfar, Chaudhary, Sumit, Magdum, Amol, Meru, Ashwinkumar V., Ghosh, Indraneel, Bhamidipati, Ravi K., Raje, Amol A., Madgula, Vamsi L. M., De, Siddhartha, Rouduri, Sreekanth R., Palle, Venkata P., Chugh, Anita, Hariharan, Narayanan, Mookhtiar, Kasim A.
Published in ACS medicinal chemistry letters (01.08.2017)
Published in ACS medicinal chemistry letters (01.08.2017)
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Journal Article
A 2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Waman, Yogesh, Patel, Meena, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Bonagiri, Rajesh, Jadhav, Dilip, Mukhopadhyay, Partha, Prasad, Vandna, Reddy, B Srinivasa, Goswami, Arnab, Chaturvedi, Sandhya, Menon, Suraj, Quraishi, Azfar, Ghosh, Indraneel, Dusange, Sushant, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Thakre, Rhishikesh, Bedse, Gaurav, Rouduri, Sreekanth, Gundu, Jayasagar, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
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Journal Article
A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Waman, Yogesh, Patel, Meena, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Bonagiri, Rajesh, Jadhav, Dilip, Mukhopadhyay, Partha, Prasad, Vandna, Reddy, B. Srinivasa, Goswami, Arnab, Chaturvedi, Sandhya, Menon, Suraj, Quraishi, Azfar, Ghosh, Indraneel, Dusange, Sushant, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Thakre, Rhishikesh, Bedse, Gaurav, Rouduri, Sreekanth, Gundu, Jayasagar, Palle, Venkata P., Chugh, Anita, Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
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Journal Article