Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation
Gilan, Omer, Rioja, Inmaculada, Knezevic, Kathy, Bell, Matthew J, Yeung, Miriam M, Harker, Nicola R, Lam, Enid Y N, Chung, Chun-Wa, Bamborough, Paul, Petretich, Massimo, Urh, Marjeta, Atkinson, Stephen J, Bassil, Anna K, Roberts, Emma J, Vassiliadis, Dane, Burr, Marian L, Preston, Alex G S, Wellaway, Christopher, Werner, Thilo, Gray, James R, Michon, Anne-Marie, Gobbetti, Thomas, Kumar, Vinod, Soden, Peter E, Haynes, Andrea, Vappiani, Johanna, Tough, David F, Taylor, Simon, Dawson, Sarah-Jane, Bantscheff, Marcus, Lindon, Matthew, Drewes, Gerard, Demont, Emmanuel H, Daniels, Danette L, Grandi, Paola, Prinjha, Rab K, Dawson, Mark A
Published in Science (American Association for the Advancement of Science) (24.04.2020)
Published in Science (American Association for the Advancement of Science) (24.04.2020)
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Potent antimyeloma activity of the novel bromodomain inhibitors I-BET151 and I-BET762
Chaidos, Aristeidis, Caputo, Valentina, Gouvedenou, Katerina, Liu, Binbin, Marigo, Ilaria, Chaudhry, Mohammed Suhail, Rotolo, Antonia, Tough, David F., Smithers, Nicholas N., Bassil, Anna K., Chapman, Trevor D., Harker, Nicola R., Barbash, Olena, Tummino, Peter, Al-Mahdi, Niam, Haynes, Andrea C., Cutler, Leanne, Le, BaoChau, Rahemtulla, Amin, Roberts, Irene, Kleijnen, Maurits, Witherington, Jason J., Parr, Nigel J., Prinjha, Rab K., Karadimitris, Anastasios
Published in Blood (30.01.2014)
Published in Blood (30.01.2014)
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Signaling function of PRC2 is essential for TCR-driven T cell responses
Dobenecker, Marc-Werner, Park, Joon Seok, Marcello, Jonas, McCabe, Michael T, Gregory, Richard, Knight, Steven D, Rioja, Inmaculada, Bassil, Anna K, Prinjha, Rabinder K, Tarakhovsky, Alexander
Published in The Journal of experimental medicine (02.04.2018)
Published in The Journal of experimental medicine (02.04.2018)
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Phase 1 and preclinical profiling of ESM‐HDAC391, a myeloid‐targeted histone deacetylase inhibitor, shows enhanced pharmacology and monocytopaenia
Furze, Rebecca C., Molnar, Judit, Parr, Nigel J., Ahmad, Faiz, Henry, Yvette, Howe, David, Singh, Rajendra, Toal, Martin, Bassil, Anna K., Bernard, Sharon G., Davis, Robert P., Gibson, Adele, Maller, N. Claire, Sharp, Catriona, Tough, David F., Prinjha, Rab K., Lewis, Huw D.
Published in British journal of clinical pharmacology (01.12.2022)
Published in British journal of clinical pharmacology (01.12.2022)
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UDP-glucose modulates gastric function through P2Y14 receptor-dependent and -independent mechanisms
Bassil, Anna K, Bourdu, Sophie, Townson, Karen A, Wheeldon, Alan, Jarvie, Emma M, Zebda, Noureddine, Abuin, Alejandro, Grau, Evelyn, Livi, George P, Punter, Lorraine, Latcham, Judith, Grimes, Angela M, Hurp, David P, Downham, Kelly M, Sanger, Gareth J, Winchester, Wendy J, Morrison, Alastair D, Moore, Gary B T
Published in American journal of physiology: Gastrointestinal and liver physiology (01.04.2009)
Published in American journal of physiology: Gastrointestinal and liver physiology (01.04.2009)
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Journal Article
Selective targeting of BD1 and BD2 of the BET proteins in cancer and immuno-inflammation
Gilan, Omer, Rioja, Inmaculada, Knezevic, Kathy, Bell, Matthew J, Yeung, Miriam M., Harker, Nicola R, Lam, Enid Y.N., Chung, Chun-wa, Bamborough, Paul, Petretich, Massimo, Urh, Marjeta, Atkinson, Stephen J, Bassil, Anna K, Roberts, Emma J, Vassiliadis, Dane, Burr, Marian L., Preston, Alex G.S, Wellaway, Christopher, Werner, Thilo, Gray, James R, Michon, Anne-Marie, Gobbetti, Thomas, Kumar, Vinod, Soden, Peter E, Haynes, Andrea, Vappiani, Johanna, Tough, David F, Taylor, Simon, Dawson, Sarah-Jane, Bantscheff, Marcus, Lindon, Matthew, Drewes, Gerard, Demont, Emmanuel H, Daniels, Danette L., Grandi, Paola, Prinjha, Rab K, Dawson, Mark A.
Published in Science (American Association for the Advancement of Science) (19.03.2020)
Published in Science (American Association for the Advancement of Science) (19.03.2020)
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Journal Article
Potent Anti-Myeloma Activity Of The Novel Bromodomain Inhibitors I-BET151 and I-BET762
Chaidos, Aristeidis, Caputo, Valentina, Marigo, Ilaria, Liu, Binbin, Chaudhry, Suhail, Goudevenou, Katerina, Rotolo, Antonia, Tough, David F, Smithers, Nicholas N, Bassil, Anna K, Chapman, Trevor D, Harker, Nicola R, Barbash, Olena, Tummino, Peter, Al-Mahdi, Niam, Haynes, Andrea C, Cutler, Leanne, Le, BaoChau, Rahemtulla, Amin, Roberts, Irene, Kleijnen, Maurits, Witherington, Jason, Parr, Nigel J, Prinjha, Rab K, Karadimitris, Anastasios
Published in Blood (15.11.2013)
Published in Blood (15.11.2013)
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UDP-glucose modulates gastric function through P2Y 14 receptor-dependent and -independent mechanisms
Bassil, Anna K., Bourdu, Sophie, Townson, Karen A., Wheeldon, Alan, Jarvie, Emma M., Zebda, Noureddine, Abuin, Alejandro, Grau, Evelyn, Livi, George P., Punter, Lorraine, Latcham, Judith, Grimes, Angela M., Hurp, David P., Downham, Kelly M., Sanger, Gareth J., Winchester, Wendy J., Morrison, Alastair D., Moore, Gary B. T.
Published in American journal of physiology: Gastrointestinal and liver physiology (01.04.2009)
Published in American journal of physiology: Gastrointestinal and liver physiology (01.04.2009)
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Journal Article
UDP-glucose modulates gastric function through P2Y^sub 14^ receptor-dependent and -independent mechanisms
Bassil, Anna K, Bourdu, Sophie, Townson, Karen A, Wheeldon, Alan, Jarvie, Emma M, Zebda, Noureddine, Abuin, Alejandro, Grau, Evelyn, Livi, George P, Punter, Lorraine, Latcham, Judith, Grimes, Angela M, Hurp, David P, Downham, Kelly M, Sanger, Gareth J, Winchester, Wendy J, Morrison, Alastair D, Moore, Gary B T
Published in American journal of physiology: Gastrointestinal and liver physiology (01.04.2009)
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Published in American journal of physiology: Gastrointestinal and liver physiology (01.04.2009)
Journal Article
UDP-glucose modulates gastric function through P2Y14 receptor-dependent and -independent mechanisms
BASSIL, Anna K, BOURDU, Sophie, LATCHAM, Judith, GRIMES, Angela M, HURP, David P, DOWNHAM, Kelly M, SANGER, Gareth J, WINCHESTER, Wendy J, MORRISON, Alastair D, MOORE, Gary B. T, TOWNSON, Karen A, WHEELDON, Alan, JARVIE, Emma M, ZEBDA, Noureddine, ABUIN, Alejandro, GRAU, Evelyn, LIVI, George P, PUNTER, Lorraine
Published in American journal of physiology: Gastrointestinal and liver physiology (2009)
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Published in American journal of physiology: Gastrointestinal and liver physiology (2009)
Journal Article
Demonstration of functional neuronal beta3-adrenoceptors within the enteric nervous system
Cellek, Selim, Thangiah, Ramkumar, Bassil, Anna K, Campbell, Colin A, Gray, Karen M, Stretton, Jennifer L, Lalude, Olutunde, Vivekanandan, Shanmugam, Wheeldon, Alan, Winchester, Wendy J, Sanger, Gareth J, Schemann, Michael, Lee, Kevin
Published in Gastroenterology (New York, N.Y. 1943) (01.07.2007)
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Published in Gastroenterology (New York, N.Y. 1943) (01.07.2007)
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