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Structure-Based Drug Design of Novel, Potent, and Selective Azabenzimidazoles (ABI) as ATR Inhibitors
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Published in ACS medicinal chemistry letters (08.01.2015)
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Total Synthesis of (+)-Zaragozic Acid C
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Published in Journal of organic chemistry (20.10.2000)
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Synthesis of the C1-side chain of zaragozic acid D and progress towards a total synthesis
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Published in Tetrahedron (13.01.2003)
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Preparation of Chlorosilyl Enolates
Denmark, Scott E, Stavenger, Robert A, Winter, Stephen B. D, Wong, Ken-Tsung, Barsanti, Paul A
Published in Journal of organic chemistry (11.12.1998)
Published in Journal of organic chemistry (11.12.1998)
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HU CHENG, BARSANTI PAUL A, SENDZIK MARTIN, PFISTER KEITH B, SUTTON JAMES
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DING YU, HU CHENG, BARSANTI PAUL A, HAN, WOO SEOK, ABRAMS TINYA, PAN YUE, DUHL DAVID
Year of Publication 09.09.2013
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Year of Publication 09.09.2013
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Year of Publication 23.10.2013
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BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS
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Year of Publication 27.11.2015
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Design and Discovery of N‑(2-Methyl-5′-morpholino-6′-((tetrahydro‑2H‑pyran-4-yl)oxy)-[3,3′-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide (RAF709): A Potent, Selective, and Efficacious RAF Inhibitor Targeting RAS Mutant Cancers
Nishiguchi, Gisele A, Rico, Alice, Tanner, Huw, Aversa, Robert J, Taft, Benjamin R, Subramanian, Sharadha, Setti, Lina, Burger, Matthew T, Wan, Lifeng, Tamez, Victoriano, Smith, Aaron, Lou, Yan, Barsanti, Paul A, Appleton, Brent A, Mamo, Mulugeta, Tandeske, Laura, Dix, Ina, Tellew, John E, Huang, Shenlin, Mathews Griner, Lesley A, Cooke, Vesselina G, Van Abbema, Anne, Merritt, Hanne, Ma, Sylvia, Gampa, Kalyani, Feng, Fei, Yuan, Jing, Wang, Yingyun, Haling, Jacob R, Vaziri, Sepideh, Hekmat-Nejad, Mohammad, Jansen, Johanna M, Polyakov, Valery, Zang, Richard, Sethuraman, Vijay, Amiri, Payman, Singh, Mallika, Lees, Emma, Shao, Wenlin, Stuart, Darrin D, Dillon, Michael P, Ramurthy, Savithri
Published in Journal of medicinal chemistry (22.06.2017)
Published in Journal of medicinal chemistry (22.06.2017)
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BIPYRIDINES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES
HU CHENG, BARSANTI PAUL A, SENDZIK MARTIN, NG SIMON C, JIN XIANMING, PFISTER KEITH B, SUTTON JAMES
Year of Publication 21.08.2012
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Year of Publication 21.08.2012
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HU CHENG, LIN XIAODONG, BARSANTI PAUL A, KEYES ROBERT, SENDZIK MARTIN, JIN JEFF, WAN LIFENG, PAN YUE, KUCEJKO ROBERT, PFISTER KEITH B, SUTTON JAMES
Year of Publication 20.04.2012
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Year of Publication 20.04.2012
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Abstract 2696: Genetic and pharmacologic evaluation of the ubiquitin ligase CBL-B as a small-molecule, tumor immunotherapy target
Gosling, Jennifa, Rountree, Ryan, Taherbhoy, Asad, Wang, Chenbo, Cummins, Thomas, Cohen, Frederick, Tanaka, Hiroko, Weiss, Dahlia, Cardozo, Mario, Karim, Christopher, Tan, May, Juan, Joseph, Tenn-McClellan, Austin, Soly, Szerenke Kiss von, Sheung, Julie, Boyle, Kathleen, Dhamnaskar, Ketki, Kurylo, Katherine, Bruffey, Jilliane, McKinnell, Jennifer, Karr, Dane, Christianson, Andria, Vries, Anne-Renee Van Der Vuurst de, Sivakumar, Pallavur, Gallop, Mark, Barsanti, Paul A., Saha, Anjanabha, Bence, Neil F., Zapf, Christoph W.
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS
XIA YI, BARSANTI PAUL A, WALTER ANNETTE O, MENDENHALL KRIS G, RENHOWE PAUL A, DUHL DAVID
Year of Publication 27.07.2009
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Year of Publication 27.07.2009
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