Synthesis and binding affinities of novel spirocyclic lactam peptidomimetics of somatostatin
Damour, D, Barreau, M, Blanchard, JC, Burgevin, MC, Doble, A, Pantel, G, Labaudiniere, R, Mignani, S
Published in Chemistry letters (01.09.1998)
Published in Chemistry letters (01.09.1998)
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Synthesis and pharmacological properties of 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, a new competitive AMPA/KA receptor antagonist
Mignani, Serge, Aloup, Jean-Claude, Barreau, Michel, Blanchard, Jean Charles, Böhme, Georg Andrees, Boireau, Alain, Damour, Dominique, Debono, Marc-Williams, Dubroeucq, Marie-Christine, Genevois-Borella, Arielle, Imperato, Assunta, Jimonet, Patrick, Pratt, Jeremy, Randle, John C.R., Reibaud, Michel, Ribeill, Yves, Stutzmann, Jean-Marie
Published in Drug development research (01.11.1999)
Published in Drug development research (01.11.1999)
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Riluzole Series. Synthesis and in Vivo “Antiglutamate” Activity of 6-Substituted-2-benzothiazolamines and 3-Substituted-2-imino-benzothiazolines
Jimonet, Patrick, Audiau, François, Barreau, Michel, Blanchard, Jean-Charles, Boireau, Alain, Bour, Yvette, Coléno, Marie-Annick, Doble, Adam, Doerflinger, Gilles, Do Huu, Claudine, Donat, Marie-Hélène, Duchesne, Jean Marie, Ganil, Pierre, Guérémy, Claude, Honoré, Eliane, Just, Bernard, Kerphirique, Roselyne, Gontier, Sylvie, Hubert, Philippe, Laduron, Pierre M, Le Blevec, Joseph, Meunier, Mireille, Miquet, Jean-Marie, Nemecek, Conception, Pasquet, Martine, Piot, Odile, Pratt, Jeremy, Rataud, Jean, Reibaud, Michel, Stutzmann, Jean-Marie, Mignani, Serge
Published in Journal of medicinal chemistry (29.07.1999)
Published in Journal of medicinal chemistry (29.07.1999)
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Stereoselective synthesis of racemic α-amino-acid derivatives with a β-lactam skeleton: Application of the Staudinger reaction to chiral imines of methyl glyoxylate
Barreau, Michel, Commerçon, Alain, Mignani, Serge, Mouysset, Dominique, Perfetti, Patricia, Stella, Lucien
Published in Tetrahedron (17.09.1998)
Published in Tetrahedron (17.09.1998)
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1,8-BENZONAPHTHYRIDINE DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM
GIRARD, PHILIPPE, PICAUT, GUY, BARREAU, MICHEL, ANTOINE, MICHEL, DESCONCLOIS, JEAN-FRANCOIS
Year of Publication 01.05.1999
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Year of Publication 01.05.1999
Patent
1,8-BENZONAPHTHYRIDINE DERIVATIVES THEIR PREPARATION
GIRARD, PHILIPPE, ANTOINE, MECHEL, PICAUT, GUY, BARREAU, MICHEL, DESCONCLOIS, JEAN-FRANCOIS
Year of Publication 15.07.1998
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Year of Publication 15.07.1998
Patent
Synthesis and biological evaluation of O-alkylated tropolones and related α-ketohydroxy derivatives as ribonucleotide reductase inhibitors
Tamburlin-Thumin, Isabelle, Crozet, Michel P., Barrière, Jean-Claude, Barreau, Michel, Riou, Jean-François, Lavelle, François
Published in European journal of medicinal chemistry (01.06.2001)
Published in European journal of medicinal chemistry (01.06.2001)
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Construction of 2,3- and 3,4-Functionalized Silacyclopentanes: Synthesis of 6-Aza-2,2-Diphenyl-2-Silabicyclo[3.1.0]Hexane and 6-Aza-3,3-Diphenyl-3-Silabicyclo[3.1.0]Hexane Derivatives
Mignani, Serge, Barreau, Michel, Damour, Dominique, Renaudon, Alain, Dejean, Valérie, Manuel, Georges
Published in Synthetic communications (01.04.1998)
Published in Synthetic communications (01.04.1998)
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Radical-induced cyclizations of 1-sila-cyclopent-2-ene derivatives: Synthesis of novel azasilabicyclic compounds
Damour, D, Barreau, M, Dhaleine, F, Doerflinger, G, Vuilhorgne, M, Mignani, S
Published in Synlett (01.09.1996)
Published in Synlett (01.09.1996)
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1,1-diphenyl-3-dialkylamino-1-silacyclopentane derivatives: A new class of potent and selective 5-HT 2A antagonists
Damour, Dominique, Barreau, Michel, Dutruc-Rosset, Gilles, Doble, Adam, Piot, Odile, Mignani, Serge
Published in Bioorganic & medicinal chemistry letters (1994)
Published in Bioorganic & medicinal chemistry letters (1994)
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Journal Article
1,1-diphenyl-3-dialkylamino-1-silacyclopentane derivatives: A new class of potent and selective 5-HT2A antagonists
Damour, Dominique, Barreau, Michel, Dutruc-Rosset, Gilles, Doble, Adam, Piot, Odile, Mignani, Serge
Published in Bioorganic & medicinal chemistry letters (10.02.1994)
Published in Bioorganic & medicinal chemistry letters (10.02.1994)
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Journal Article
An efficient preparative route to fused imidazo[1,2-a]pyrazin-4-one derivatives
Damour, D, Aloup, JC, Barreau, M, Genevois-Borella, A, Jimonet, P, Leconte, JP, Ribeill, Y, Vuilhorgne, M, Mignani, S
Published in Heterocycles (01.01.1999)
Published in Heterocycles (01.01.1999)
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