A novel GABA(A) alpha 5 receptor inhibitor with therapeutic potential
Ling, István, Mihalik, Balázs, Etherington, Lori-An, Kapus, Gábor, Pálvölgyi, Adrienn, Gigler, Gábor, Kertész, Szabolcs, Gaál, Attila, Pallagi, Katalin, Kiricsi, Péter, Szabó, Éva, Szénási, Gábor, Papp, Lilla, Hársing, László G, Lévay, György, Spedding, Michael, Lambert, Jeremy J, Belelli, Delia, Barkóczy, József, Volk, Balázs, Simig, Gyula, Gacsályi, István, Antoni, Ferenc A
Published in European journal of pharmacology (05.10.2015)
Published in European journal of pharmacology (05.10.2015)
Get full text
Journal Article
Egis-11150: A candidate antipsychotic compound with procognitive efficacy in rodents
Gacsályi, István, Nagy, Katalin, Pallagi, Katalin, Lévay, György, Hársing, László G., Móricz, Krisztina, Kertész, Szabolcs, Varga, Péter, Haller, József, Gigler, Gábor, Szénási, Gábor, Barkóczy, József, Bíró, Judit, Spedding, Michael, Antoni, Ferenc A.
Published in Neuropharmacology (01.01.2013)
Published in Neuropharmacology (01.01.2013)
Get full text
Journal Article
Reduction of cerebral infarct size by non-competitive AMPA antagonists in rats subjected to permanent and transient focal ischemia
Matucz, Éva, Móricz, Krisztina, Gigler, Gábor, Simó, Annamária, Barkóczy, József, Lévay, György, Hársing, László G, Szénási, Gábor
Published in Brain research (03.09.2004)
Published in Brain research (03.09.2004)
Get full text
Journal Article
Therapeutic time window of neuroprotection by non-competitive AMPA antagonists in transient and permanent focal cerebral ischemia in rats
Matucz, Éva, Móricz, Krisztina, Gigler, Gábor, Benedek, Angéla, Barkóczy, József, Lévay, György, Hársing, László G., Szénási, Gábor
Published in Brain research (06.12.2006)
Published in Brain research (06.12.2006)
Get full text
Journal Article
Phenotypical Screening on Neuronal Plasticity in Hippocampal-Prefrontal Cortex Connectivity Reveals an Antipsychotic with a Novel Profile
Spedding, Michael, Sebban, Claude, Jay, Thérèse M, Rocher, Cyril, Tesolin-Decros, Brigitte, Chazot, Paul, Schenker, Esther, Szénási, Gabor, Lévay, György I, Megyeri, Katalin, Barkóczy, Jozsef, Hársing, Jr, Laszlo G, Thomson, Ian, Cunningham, Mark O, Whittington, Miles A, Etherington, Lori-An, Lambert, Jeremy J, Antoni, Ferenc A, Gacsályi, Istvan
Published in Cells (Basel, Switzerland) (31.03.2022)
Published in Cells (Basel, Switzerland) (31.03.2022)
Get full text
Journal Article
The Dolastatins. 17. Synthesis of Dolaproine and Related Diastereoisomers
Pettit, George R, Singh, Sheo Bux, Herald, Delbert L, Lloyd-Williams, Paul, Kantoci, Darko, Burkett, Douglas D, Barkoczy, Jozsef, Hogan, Fiona, Wardlaw, Terah R
Published in Journal of organic chemistry (01.10.1994)
Published in Journal of organic chemistry (01.10.1994)
Get full text
Journal Article
Selective inhibition of extra-synaptic α5-GABAA receptors by S44819, a new therapeutic agent
Etherington, Lori-An, Mihalik, Balázs, Pálvölgyi, Adrienn, Ling, István, Pallagi, Katalin, Kertész, Szabolcs, Varga, Péter, Gunn, Ben G., Brown, Adam R., Livesey, Matthew R., Monteiro, Olivia, Belelli, Delia, Barkóczy, József, Spedding, Michael, Gacsályi, István, Antoni, Ferenc A., Lambert, Jeremy J.
Published in Neuropharmacology (01.10.2017)
Published in Neuropharmacology (01.10.2017)
Get full text
Journal Article
Behavioural pharmacology of the α5-GABAA receptor antagonist S44819: Enhancement and remediation of cognitive performance in preclinical models
Gacsályi, István, Móricz, Krisztina, Gigler, Gábor, Wellmann, János, Nagy, Katalin, Ling, István, Barkóczy, József, Haller, József, Lambert, Jeremy J., Szénási, Gábor, Spedding, Michael, Antoni, Ferenc A.
Published in Neuropharmacology (01.10.2017)
Published in Neuropharmacology (01.10.2017)
Get full text
Journal Article
Loop-F of the α-subunit determines the pharmacologic profile of novel competitive inhibitors of GABAA receptors
Mihalik, Balázs, Pálvölgyi, Adrienn, Bogár, Ferenc, Megyeri, Katalin, Ling, István, Barkóczy, József, Bartha, Ferenc, Martinek, Tamás A., Gacsályi, István, Antoni, Ferenc A.
Published in European journal of pharmacology (05.03.2017)
Published in European journal of pharmacology (05.03.2017)
Get full text
Journal Article
A novel GABAA alpha 5 receptor inhibitor with therapeutic potential
Ling, István, Mihalik, Balázs, Etherington, Lori-An, Kapus, Gábor, Pálvölgyi, Adrienn, Gigler, Gábor, Kertész, Szabolcs, Gaál, Attila, Pallagi, Katalin, Kiricsi, Péter, Szabó, Éva, Szénási, Gábor, Papp, Lilla, Hársing, László G., Lévay, György, Spedding, Michael, Lambert, Jeremy J., Belelli, Delia, Barkóczy, József, Volk, Balázs, Simig, Gyula, Gacsályi, István, Antoni, Ferenc A.
Published in European journal of pharmacology (05.10.2015)
Published in European journal of pharmacology (05.10.2015)
Get full text
Journal Article
Behavioural pharmacology of the α5-GABA A receptor antagonist S44819: Enhancement and remediation of cognitive performance in preclinical models
Gacsályi, István, Móricz, Krisztina, Gigler, Gábor, Wellmann, János, Nagy, Katalin, Ling, István, Barkóczy, József, Haller, József, Lambert, Jeremy J, Szénási, Gábor, Spedding, Michael, Antoni, Ferenc A
Published in Neuropharmacology (01.10.2017)
Published in Neuropharmacology (01.10.2017)
Get full text
Journal Article
Selective inhibition of extra-synaptic α5-GABA A receptors by S44819, a new therapeutic agent
Etherington, Lori-An, Mihalik, Balázs, Pálvölgyi, Adrienn, Ling, István, Pallagi, Katalin, Kertész, Szabolcs, Varga, Péter, Gunn, Ben G, Brown, Adam R, Livesey, Matthew R, Monteiro, Olivia, Belelli, Delia, Barkóczy, József, Spedding, Michael, Gacsályi, István, Antoni, Ferenc A, Lambert, Jeremy J
Published in Neuropharmacology (01.10.2017)
Published in Neuropharmacology (01.10.2017)
Get full text
Journal Article
Loop-F of the α-subunit determines the pharmacologic profile of novel competitive inhibitors of GABA A receptors
Mihalik, Balázs, Pálvölgyi, Adrienn, Bogár, Ferenc, Megyeri, Katalin, Ling, István, Barkóczy, József, Bartha, Ferenc, Martinek, Tamás A, Gacsályi, István, Antoni, Ferenc A
Published in European journal of pharmacology (05.03.2017)
Published in European journal of pharmacology (05.03.2017)
Get full text
Journal Article
(Phenylpiperazinyl-butyl)oxindoles as Selective 5-HT7 Receptor Antagonists
Volk, Balázs, Barkóczy, József, Hegedus, Endre, Udvari, Szabolcs, Gacsályi, István, Mezei, Tibor, Pallagi, Katalin, Kompagne, Hajnalka, Lévay, György, Egyed, András, Hársing, Jr, László G, Spedding, Michael, Simig, Gyula
Published in Journal of medicinal chemistry (24.04.2008)
Published in Journal of medicinal chemistry (24.04.2008)
Get full text
Journal Article
(Phenylpiperazinyl-butyl)oxindoles as Selective 5-HT 7 Receptor Antagonists
Volk, Balázs, Barkóczy, József, Hegedus, Endre, Udvari, Szabolcs, Gacsályi, István, Mezei, Tibor, Pallagi, Katalin, Kompagne, Hajnalka, Lévay, György, Egyed, András, Hársing, Jr, László G., Spedding, Michael, Simig, Gyula
Published in Journal of medicinal chemistry (01.04.2008)
Published in Journal of medicinal chemistry (01.04.2008)
Get full text
Journal Article
Antagonism of AMPA receptors produces anxiolytic-like behavior in rodents: Effects of GYKI 52466 and its novel analogues
Kapus, Gábor L., Gacsályi, István, Vegh, Miklos, Kompagne, Hajnalka, Hegedűs, Endre, Leveleki, Csilla, Hársing, László G., Barkóczy, József, Bilkei-Gorzó, András, Lévay, György
Published in Psychopharmacologia (01.06.2008)
Published in Psychopharmacologia (01.06.2008)
Get full text
Journal Article
Comparison of the AMPA antagonist action of new 2,3-benzodiazepines in vitro and their neuroprotective effects in vivo
Kapus, Gábor, Kertész, Szabolcs, Gigler, Gábor, Simó, Annamária, Vegh, Miklos, Barkóczy, József, Hársing, László G, Szabó, Géza, Lévay, György
Published in Pharmaceutical research (01.02.2004)
Published in Pharmaceutical research (01.02.2004)
Get full text
Journal Article
The effects of AMPA receptor antagonists in models of stroke and neurodegeneration
Gressens, Pierre, Spedding, Michael, Gigler, Gabor, Kertesz, Szabolcs, Villa, Pascal, Medja, Fadia, Williamson, Toni, Kapus, Gabor, Levay, Gyorgy, Szenasi, Gabor, Barkoczy, Jozsef, Harsing, Laszlo G.
Published in European journal of pharmacology (05.09.2005)
Published in European journal of pharmacology (05.09.2005)
Get full text
Journal Article
On triazoles XLI. Synthesis of meso-ionic [1,2,4]triazolo[5,1-c]thiadiazoles
Reiter, J, Barkoczy, J, Argay, G, Kalman, A
Published in Journal of heterocyclic chemistry (01.03.2000)
Published in Journal of heterocyclic chemistry (01.03.2000)
Get more information
Journal Article