Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B. Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R., Palle, Venkata P., Chugh, Anita, Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
Get full text
Journal Article
Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2′s-hydroxy-3′s-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors
Kandalkar, Sachin R., Ramaiah, Parimi Atchuta, Joshi, Manoj, Wavhal, Atul, Waman, Yogesh, Raje, Amol A., Tambe, Ashwini, Ansari, Shariq, De, Siddhartha, Palle, Venkata P., Mookhtiar, Kasim A., Deshpande, Anil M., Barawkar, Dinesh A.
Published in Bioorganic & medicinal chemistry (15.10.2017)
Published in Bioorganic & medicinal chemistry (15.10.2017)
Get full text
Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
Get full text
Journal Article
Design and synthesis of novel xanthine derivatives as potent and selective A 2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Patel, Meena, Waman, Yogesh, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Naykodi, Minakshi, Goswami, Arnab, Reddy, B Srinivasa, Prasad, Vandna, Chaturvedi, Sandhya, Quraishi, Azfar, Menon, Suraj, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Ghosh, Indraneel, Mustafa, Syed, De, Siddhartha, Jain, Vaibhav, Banerjee, Ena Ray, Rouduri, Sreekanth R, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (07.07.2017)
Published in European journal of medicinal chemistry (07.07.2017)
Get full text
Journal Article
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A 1 receptor antagonists and their biological evaluation
Koul, Summon, Ramdas, Vidya, Barawkar, Dinesh A, Waman, Yogesh B, Prasad, Neela, Madadi, Santosh Kumar, Shejul, Yogesh D, Bonagiri, Rajesh, Basu, Sujay, Menon, Suraj, Reddy, Srinivasa B, Chaturvedi, Sandhya, Chennamaneni, Srinivas Rao, Bedse, Gaurav, Thakare, Rhishikesh, Gundu, Jayasagar, Chaudhary, Sumit, De, Siddhartha, Meru, Ashwinkumar V, Palle, Venkata, Chugh, Anita, Mookhtiar, Kasim A
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
Get full text
Journal Article
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation
Koul, Summon, Ramdas, Vidya, Barawkar, Dinesh A., Waman, Yogesh B., Prasad, Neela, Madadi, Santosh Kumar, Shejul, Yogesh D., Bonagiri, Rajesh, Basu, Sujay, Menon, Suraj, Reddy, Srinivasa B., Chaturvedi, Sandhya, Chennamaneni, Srinivas Rao, Bedse, Gaurav, Thakare, Rhishikesh, Gundu, Jayasagar, Chaudhary, Sumit, De, Siddhartha, Meru, Ashwinkumar V., Palle, Venkata, Chugh, Anita, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry (15.03.2017)
Published in Bioorganic & medicinal chemistry (15.03.2017)
Get full text
Journal Article
Highly efficient one-pot amination of carboxylate-substituted nitrogen-containing heteroaryl chlorides via Staudinger reaction
Kandalkar, Sachin R., Kaduskar, Rahul D., Ramaiah, Parimi Atchuta, Barawkar, Dinesh A., Bhuniya, Debnath, Deshpande, Anil M.
Published in Tetrahedron letters (30.01.2013)
Published in Tetrahedron letters (30.01.2013)
Get full text
Journal Article
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A 2A Receptor Antagonists and Their Biological Evaluation
Basu, Sujay, Barawkar, Dinesh A, Thorat, Sachin, Shejul, Yogesh D, Patel, Meena, Naykodi, Minakshi, Jain, Vaibhav, Salve, Yogesh, Prasad, Vandna, Chaudhary, Sumit, Ghosh, Indraneel, Bhat, Ganesh, Quraishi, Azfar, Patil, Harish, Ansari, Shariq, Menon, Suraj, Unadkat, Vishal, Thakare, Rhishikesh, Seervi, Madhav S, Meru, Ashwinkumar V, De, Siddhartha, Bhamidipati, Ravi K, Rouduri, Sreekanth R, Palle, Venkata P, Chug, Anita, Mookhtiar, Kasim A
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
Get full text
Journal Article
Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors
Basu, Sujay, Prasad, Uppuleti Viplava, Barawkar, Dinesh A., De, Siddhartha, Palle, Venkata P., Menon, Suraj, Patel, Meena, Thorat, Sachin, Singh, Umesh P., Sarma, Koushik Das, Waman, Yogesh, Niranjan, Sanjay, Pathade, Vishal, Gaur, Ashwani, Reddy, Satyanarayana, Ansari, Shariq
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Get full text
Journal Article
A 2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Waman, Yogesh, Patel, Meena, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Bonagiri, Rajesh, Jadhav, Dilip, Mukhopadhyay, Partha, Prasad, Vandna, Reddy, B Srinivasa, Goswami, Arnab, Chaturvedi, Sandhya, Menon, Suraj, Quraishi, Azfar, Ghosh, Indraneel, Dusange, Sushant, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Thakre, Rhishikesh, Bedse, Gaurav, Rouduri, Sreekanth, Gundu, Jayasagar, Palle, Venkata P, Chugh, Anita, Mookhtiar, Kasim A
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
Get full text
Journal Article
A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives
Basu, Sujay, Barawkar, Dinesh A., Ramdas, Vidya, Waman, Yogesh, Patel, Meena, Panmand, Anil, Kumar, Santosh, Thorat, Sachin, Bonagiri, Rajesh, Jadhav, Dilip, Mukhopadhyay, Partha, Prasad, Vandna, Reddy, B. Srinivasa, Goswami, Arnab, Chaturvedi, Sandhya, Menon, Suraj, Quraishi, Azfar, Ghosh, Indraneel, Dusange, Sushant, Paliwal, Shalini, Kulkarni, Abhay, Karande, Vikas, Thakre, Rhishikesh, Bedse, Gaurav, Rouduri, Sreekanth, Gundu, Jayasagar, Palle, Venkata P., Chugh, Anita, Mookhtiar, Kasim A.
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
Get full text
Journal Article
Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson’s Disease and Depression
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Naykodi, Minakshi, Shejul, Yogesh D, Patel, Meena, Thorat, Sachin, Panmand, Anil, Kashinath, K, Bonagiri, Rajesh, Prasad, Vandna, Bhat, Ganesh, Quraishi, Azfar, Chaudhary, Sumit, Magdum, Amol, Meru, Ashwinkumar V, Ghosh, Indraneel, Bhamidipati, Ravi K, Raje, Amol A, Madgula, Vamsi L. M, De, Siddhartha, Rouduri, Sreekanth R, Palle, Venkata P, Chugh, Anita, Hariharan, Narayanan, Mookhtiar, Kasim A
Published in ACS medicinal chemistry letters (10.08.2017)
Published in ACS medicinal chemistry letters (10.08.2017)
Get full text
Journal Article
Discovery of Potent and Selective A 2A Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression
Basu, Sujay, Barawkar, Dinesh A, Ramdas, Vidya, Naykodi, Minakshi, Shejul, Yogesh D, Patel, Meena, Thorat, Sachin, Panmand, Anil, Kashinath, K, Bonagiri, Rajesh, Prasad, Vandna, Bhat, Ganesh, Quraishi, Azfar, Chaudhary, Sumit, Magdum, Amol, Meru, Ashwinkumar V, Ghosh, Indraneel, Bhamidipati, Ravi K, Raje, Amol A, Madgula, Vamsi L M, De, Siddhartha, Rouduri, Sreekanth R, Palle, Venkata P, Chugh, Anita, Hariharan, Narayanan, Mookhtiar, Kasim A
Published in ACS medicinal chemistry letters (10.08.2017)
Published in ACS medicinal chemistry letters (10.08.2017)
Get full text
Journal Article
Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain l-2-hydroxy acid oxidase
Barawkar, Dinesh A., Bandyopadhyay, Anish, Deshpande, Anil, Koul, Summon, Kandalkar, Sachin, Patil, Pradeep, Khose, Goraksha, Vyas, Samir, Mone, Mahesh, Bhosale, Shubhangi, Singh, Umesh, De, Siddhartha, Meru, Ashwin, Gundu, Jayasagar, Chugh, Anita, Palle, Venkata P., Mookhtiar, Kasim A., Vacca, Joseph P., Chakravarty, Prasun K., Nargund, Ravi P., Wright, Samuel D., Roy, Sophie, Graziano, Michael P., Cully, Doris, Cai, Tian-Quan, Singh, Sheo B.
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
Get full text
Journal Article
Potent and Selective Inhibitors of Long Chain l-2-Hydroxy Acid Oxidase Reduced Blood Pressure in DOCA Salt-Treated Rats
Barawkar, Dinesh A, Meru, Ashwin, Bandyopadhyay, Anish, Banerjee, Abir, Deshpande, Anil M, Athare, Chandrashekhar, Koduru, Chandrasekhar, Khose, Goraksha, Gundu, Jayasagar, Mahajan, Koshu, Patil, Pradeep, Kandalkar, Sachin R, Niranjan, Sanjay, Bhosale, Shubhangi, De, Siddhartha, Mukhopadhyay, Sudit, Chaudhary, Sumit, Koul, Summon, Singh, Umesh, Chugh, Anita, Palle, Venkata P, Mookhtiar, Kasim A, Vacca, Joseph, Chakravarty, Prasun K, Nargund, Ravi P, Wright, Samuel D, Roy, Sophie, Graziano, Michael P, Singh, Sheo B, Cully, Doris, Cai, Tian-Quan
Published in ACS medicinal chemistry letters (08.12.2011)
Published in ACS medicinal chemistry letters (08.12.2011)
Get full text
Journal Article
Synthesis, Biophysical Properties, and Nuclease Resistance Properties of Mixed Backbone Oligodeoxynucleotides Containing Cationic Internucleoside Guanidinium Linkages: Deoxynucleic Guanidine/DNA Chimeras
Barawkar, Dinesh A., Bruice, Thomas C.
Published in Proceedings of the National Academy of Sciences - PNAS (15.09.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (15.09.1998)
Get full text
Journal Article
Dinucleotide Analogues as Novel Inhibitors of RNA-Dependent RNA Polymerase of Hepatitis C Virus
Zhong, Weidong, An, Haoyun, Barawkar, Dinesh, Hong, Zhi
Published in Antimicrobial Agents and Chemotherapy (01.08.2003)
Published in Antimicrobial Agents and Chemotherapy (01.08.2003)
Get full text
Journal Article