Transient receptor potential ankyrin receptor 1 is a novel target for pro‐tussive agents
Andrè, E, Gatti, R, Trevisani, M, Preti, D, Baraldi, PG, Patacchini, R, Geppetti, P
Published in British journal of pharmacology (01.11.2009)
Published in British journal of pharmacology (01.11.2009)
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Journal Article
DNA minor groove binders as potential antitumor and antimicrobial agents
Baraldi, Pier Giovanni, Bovero, Andrea, Fruttarolo, Francesca, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Pavani, Maria Giovanna, Romagnoli, Romeo
Published in Medicinal research reviews (01.07.2004)
Published in Medicinal research reviews (01.07.2004)
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Journal Article
A glance at adenosine receptors: novel target for antitumor therapy
Merighi, Stefania, Mirandola, Prisco, Varani, Katia, Gessi, Stefania, Leung, Edward, Baraldi, Pier Giovanni, Tabrizi, Mojgan Aghazadeh, Borea, Pier Andrea
Published in Pharmacology & therapeutics (Oxford) (01.10.2003)
Published in Pharmacology & therapeutics (Oxford) (01.10.2003)
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Journal Article
7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility
Baraldi, PG, Cacciari, B, Romagnoli, R, Spalluto, G, Monopoli, A, Ongini, E, Varani, K, Borea, PA
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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Journal Article
Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A(2B) adenosine receptor antagonists
Baraldi, PG, Tabrizi, MA, Preti, D, Bovero, A, Romagnoli, R, Fruttarolo, F, Zaid, NA, Moorman, AR, Varani, K, Gessi, S, Merighi, S, Borea, PA
Published in Journal of medicinal chemistry (11.03.2004)
Published in Journal of medicinal chemistry (11.03.2004)
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Journal Article
Combined target-based and ligand-based drug design approach as a tool to define a novel 3D-pharmacophore model of human A(3) adenosine receptor antagonists: Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as a key study
Moro, S, Braiuca, P, Deflorian, F, Ferrari, C, Pastorin, G, Cacciari, B, Baraldi, PG, Varani, K, Borea, PA, Spalluto, G
Published in Journal of medicinal chemistry (13.01.2005)
Published in Journal of medicinal chemistry (13.01.2005)
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Journal Article
New 2-arylpyrazolo[4,3-c]quinoline derivatives as potent and selective human A(3) adenosine receptor antagonists
Baraldi, PG, Tabrizi, MA, Preti, D, Bovero, A, Fruttarolo, F, Romagnoli, R, Zaid, NA, Moorman, AR, Varani, K, Borea, PA
Published in Journal of medicinal chemistry (28.07.2005)
Published in Journal of medicinal chemistry (28.07.2005)
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Journal Article
Synthesis and biological activity of N-arylpiperazine-modified analogues of KN-62, a potent antagonist of the purinergic P2X(7) receptor
Baraldi, PG, Nunez, MD, Morelli, A, Falzoni, S, Di Virgilio, F, Romagnoli, R
Published in Journal of medicinal chemistry (10.04.2003)
Published in Journal of medicinal chemistry (10.04.2003)
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Journal Article
Antimicrobial and antitumor activity of n-heteroimmine-1,2,3-dithiazoles and their transformation in triazolo-, imidazo-, and pyrazolopirimidines
Baraldi, Pier Giovanni, Pavani, Maria Giovanna, Nuñez, Maria del Carmen, Brigidi, Patrizia, Vitali, Beatrice, Gambari, Roberto, Romagnoli, Romeo
Published in Bioorganic & medicinal chemistry (01.02.2002)
Published in Bioorganic & medicinal chemistry (01.02.2002)
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Journal Article
Adenosine Receptors as Mediators of Both Cell Proliferation and Cell Death of Cultured Human Melanoma Cells
Merighi, Stefania, Mirandola, Prisco, Milani, Daniela, Varani, Katia, Gessi, Stefania, Klotz, Karl-Norbert, Leung, Edward, Baraldi, Pier Giovanni, Borea, Pier Andrea
Published in Journal of investigative dermatology (01.10.2002)
Published in Journal of investigative dermatology (01.10.2002)
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Journal Article
Design, Synthesis, and Biological Evaluation of Hybrid Molecules Containing α-Methylene-γ-butyrolactones and Polypyrrole Minor Groove Binders
Baraldi, Pier Giovanni, del Carmen Nunez, Maria, Tabrizi, Mojgan Aghazadeh, De Clercq, Erik, Balzarini, Jan, Bermejo, Jaime, Estévez, Francisco, Romagnoli, Romeo
Published in Journal of medicinal chemistry (20.05.2004)
Published in Journal of medicinal chemistry (20.05.2004)
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Journal Article
A(3) adenosine receptors in human neutrophils and promyelocytic HL60 cells: a pharmacological and biochemical study
Gessi, Stefania, Varani, Katia, Merighi, Stefania, Cattabriga, Elena, Iannotta, Valeria, Leung, Edward, Baraldi, Pier Giovanni, Borea, Pier Andrea
Published in Molecular pharmacology (01.02.2002)
Published in Molecular pharmacology (01.02.2002)
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Journal Article
[(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors
Varani, K, Merighi, S, Gessi, S, Klotz, K N, Leung, E, Baraldi, P G, Cacciari, B, Romagnoli, R, Spalluto, G, Borea, P A
Published in Molecular pharmacology (01.05.2000)
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Published in Molecular pharmacology (01.05.2000)
Journal Article
Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor antagonists. Influence of the N5 substituent on the affinity at the human A(3) and A(2B) adenosine receptor subtypes: A molecular modeling investigation
Pastorin, G, Da Ros, T, Spalluto, G, Deflorian, F, Moro, S, Cacciari, B, Baraldi, PG, Gessi, S, Varani, K, Borea, PA
Published in Journal of medicinal chemistry (25.09.2003)
Published in Journal of medicinal chemistry (25.09.2003)
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Journal Article
Design, synthesis, and biological evaluation of C-9- and C-2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c] pyrimidines as new A(2A) and A(3) adenosine receptors antagonists
Baraldi, PG, Fruttarolo, F, Tabrizi, MA, Preti, D, Romagnoli, R, El-Kashef, H, Moorman, A, Varani, K, Gessi, S, Merighi, S, Borea, PA
Published in Journal of medicinal chemistry (27.03.2003)
Published in Journal of medicinal chemistry (27.03.2003)
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Journal Article
New pyrrolo[2,1-f]purine-2,4-dione and imidazo[2,1-f]purine-2,4-dione derivatives as potent and selective human A(3) adenosine receptor antagonists
Baraldi, PG, Preti, D, Tabrizi, MA, Fruttarolo, F, Romagnoli, R, Zaid, NA, Moorman, AR, Merighi, S, Varani, K, Borea, PA
Published in Journal of medicinal chemistry (14.07.2005)
Published in Journal of medicinal chemistry (14.07.2005)
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Journal Article
A(3) adenosine receptor ligands: history and perspectives
Baraldi, P G, Cacciari, B, Romagnoli, R, Merighi, S, Varani, K, Borea, P A, Spalluto, G
Published in Medicinal research reviews (01.03.2000)
Published in Medicinal research reviews (01.03.2000)
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Journal Article