Discovery and Characterization of a Novel Inhibitor of Matrix Metalloprotease-13 That Reduces Cartilage Damage in Vivo without Joint Fibroplasia Side Effects
Johnson, Adam R., Pavlovsky, Alexander G., Ortwine, Daniel F., Prior, Faith, Man, Chiu-Fai, Bornemeier, Dirk A., Banotai, Craig A., Mueller, W. Thomas, McConnell, Patrick, Yan, Chunhong, Baragi, Vijay, Lesch, Charles, Roark, W. Howard, Wilson, Michael, Datta, Kaushik, Guzman, Roberto, Han, Hyo-Kyung, Dyer, Richard D.
Published in The Journal of biological chemistry (21.09.2007)
Published in The Journal of biological chemistry (21.09.2007)
Get full text
Journal Article
Structures of human MAP kinase kinase 1 (MEK1) and MEK2 describe novel noncompetitive kinase inhibition
Hasemann, Charles A, Ohren, Jeffrey F, Chen, Huifen, Pavlovsky, Alexander, Whitehead, Christopher, Zhang, Erli, Kuffa, Peter, Yan, Chunhong, McConnell, Patrick, Spessard, Cindy, Banotai, Craig, Mueller, W Thomas, Delaney, Amy, Omer, Charles, Sebolt-Leopold, Judith, Dudley, David T, Leung, Iris K, Flamme, Cathlin, Warmus, Joseph, Kaufman, Michael, Barrett, Stephen, Tecle, Haile
Published in Nature structural & molecular biology (01.12.2004)
Published in Nature structural & molecular biology (01.12.2004)
Get full text
Journal Article
class of selective antibacterials derived from a protein kinase inhibitor pharmacophore
Miller, J. Richard, Dunham, Steve, Mochalkin, Igor, Banotai, Craig, Bowman, Matthew, Buist, Susan, Dunkle, Bill, Hanna, Debra, Harwood, H. James, Huband, Michael D, Karnovsky, Alla, Kuhn, Michael, Limberakis, Chris, Liu, Jia Y, Mehrens, Shawn, Mueller, W. Thomas, Narasimhan, Lakshmi, Ogden, Adam, Ohren, Jeff, Prasad, J.V.N. Vara, Shelly, John A, Skerlos, Laura, Sulavik, Mark, Thomas, V. Hayden, VanderRoest, Steve, Wang, LiAnn, Wang, Zhigang, Whitton, Amy, Zhu, Tong, Stover, C. Kendall
Published in Proceedings of the National Academy of Sciences - PNAS (10.02.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (10.02.2009)
Get full text
Journal Article
Characterization of substrate binding and catalysis in the potential antibacterial target N‐acetylglucosamine‐1‐phosphate uridyltransferase (GlmU)
Mochalkin, Igor, Lightle, Sandra, Zhu, Yaqi, Ohren, Jeffrey F., Spessard, Cindy, Chirgadze, Nickolay Y., Banotai, Craig, Melnick, Michael, McDowell, Laura
Published in Protein science (01.12.2007)
Published in Protein science (01.12.2007)
Get full text
Journal Article
Stereoselective binding of an enantiomeric pair of stromelysin-1 inhibitors caused by conformational entropy factors
Parker, Matthew H, Ortwine, Daniel F, O'Brien, Patrick M, Lunney, Elizabeth A, Banotai, Craig A, Mueller, William T, McConnell, Patrick, Brouillette, Christie G
Published in Bioorganic & medicinal chemistry letters (06.11.2000)
Published in Bioorganic & medicinal chemistry letters (06.11.2000)
Get full text
Journal Article
Discovery of potent, selective, bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model, Part I: Transformation of selective pyrazolodiazepinone phosphodiesterase 4 (PDE4) inhibitors into selective PDE2 inhibitors
Plummer, Mark S., Cornicelli, Joseph, Roark, Howard, Skalitzky, Donald J., Stankovic, Charles J., Bove, Susan, Pandit, Jayvardhan, Goodman, Annise, Hicks, James, Shahripour, Aurash, Beidler, David, Lu, Xiao Kang, Sanchez, Brian, Whitehead, Christopher, Sarver, Ron, Braden, Timothy, Gowan, Richard, Shen, Xi Qiang, Welch, Katherine, Ogden, Adam, Sadagopan, Nalini, Baum, Heidi, Miller, Howard, Banotai, Craig, Spessard, Cindy, Lightle, Sandra
Published in Bioorganic & medicinal chemistry letters (01.06.2013)
Published in Bioorganic & medicinal chemistry letters (01.06.2013)
Get full text
Journal Article
Discovery of potent selective bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model. Part II: Optimization studies and demonstration of in vivo efficacy
Plummer, Mark S., Cornicelli, Joseph, Roark, Howard, Skalitzky, Donald J., Stankovic, Charles J., Bove, Susan, Pandit, Jayvardhan, Goodman, Annise, Hicks, James, Shahripour, Aurash, Beidler, David, Lu, Xiao Kang, Sanchez, Brian, Whitehead, Christopher, Sarver, Ron, Braden, Timothy, Gowan, Richard, Shen, Xi Qiang, Welch, Katherine, Ogden, Adam, Sadagopan, Nalini, Baum, Heidi, Miller, Howard, Banotai, Craig, Spessard, Cindy, Lightle, Sandra
Published in Bioorganic & medicinal chemistry letters (01.06.2013)
Published in Bioorganic & medicinal chemistry letters (01.06.2013)
Get full text
Journal Article
Application of electrospray ionization mass spectrometry for studying human immunodeficiency virus protein complexes
Loo, Joseph A., Holler, Tod P., Foltin, Susan K., McConnell, Patrick, Banotai, Craig A., Horne, Nicole M., Mueller, W. Tom, Stevenson, Tracy I., Mack, David P.
Published in Proteins, structure, function, and bioinformatics (1998)
Published in Proteins, structure, function, and bioinformatics (1998)
Get full text
Journal Article
Rational protein engineering in action: The first crystal structure of a phenylalanine tRNA synthetase from Staphylococcus haemolyticus
Evdokimov, Artem G., Mekel, Marlene, Hutchings, Kim, Narasimhan, Lakshmi, Holler, Tod, McGrath, Teresa, Beattie, Bryan, Fauman, Eric, Yan, Chunhong, Heaslet, Holly, Walter, Richard, Finzel, Barry, Ohren, Jeffrey, McConnell, Patrick, Braden, Timothy, Sun, Fang, Spessard, Cindy, Banotai, Craig, Al-Kassim, Loola, Ma, Weijun, Wengender, Paul, Kole, Denis, Garceau, Norman, Toogood, Peter, Liu, Jia
Published in Journal of structural biology (01.04.2008)
Published in Journal of structural biology (01.04.2008)
Get full text
Journal Article
Corrigendum: Structures of human MAP kinase kinase 1 (MEK1) and MEK2 describe novel noncompetitive kinase inhibition
Ohren, Jeffrey F, Chen, Huifen, Pavlovsky, Alexander, Whitehead, Christopher, Zhang, Erli, Kuffa, Peter, Yan, Chunhong, McConnell, Patrick, Spessard, Cindy, Banotai, Craig, Mueller, W Thomas, Delaney, Amy, Omer, Charles, Sebolt-Leopold, Judith, Dudley, David T, Leung, Iris K, Flamme, Cathlin, Warmus, Joseph, Kaufman, Michael, Barrett, Stephen, Tecle, Haile, Hasemann, Charles A
Published in Nature structural & molecular biology (01.03.2005)
Published in Nature structural & molecular biology (01.03.2005)
Get full text
Journal Article
Erratum: Corrigendum: Structures of human MAP kinase kinase 1 (MEK1) and MEK2 describe novel noncompetitive kinase inhibition
Ohren, Jeffrey F, Chen, Huifen, Pavlovsky, Alexander, Whitehead, Christopher, Zhang, Erli, Kuffa, Peter, Yan, Chunhong, McConnell, Patrick, Spessard, Cindy, Banotai, Craig, Mueller, W Thomas, Delaney, Amy, Omer, Charles, Sebolt-Leopold, Judith, Dudley, David T, Leung, Iris K, Flamme, Cathlin, Warmus, Joseph, Kaufman, Michael, Barrett, Stephen, Tecle, Haile, Hasemann, Charles A
Published in Nature structural & molecular biology (01.03.2005)
Published in Nature structural & molecular biology (01.03.2005)
Get full text
Journal Article
PHLOROGLUCINOL SYNTHASES AND METHODS OF MAKING AND USING THE SAME
JANCAUSKAS, JUSTAS, LAU, MAN KIT, BANOTAI, CRAIG, LEHNER, BETSY, FROST, JOHN
Year of Publication 03.05.2012
Get full text
Year of Publication 03.05.2012
Patent
PHLOROGLUCINOL SYNTHASES AND METHODS OF MAKING AND USING THE SAME
JANCAUSKAS, JUSTAS, LAU, MAN KIT, BANOTAI, CRAIG, LEHNER, BETSY, FROST, JOHN
Year of Publication 05.01.2012
Get full text
Year of Publication 05.01.2012
Patent