Potent nor-triterpenoid blockers of the voltage-gated potassium channel Kv1.3 from Spachea correae
Goetz, Michael A., Hensens, Otto D., Zink, Deborah L., Borris, Robert P., Morales, Francisco, Tamayo-Castillo, Giselle, Slaughter, Robert S., Felix, John, Ball, Richard G.
Published in Tetrahedron letters (01.05.1998)
Published in Tetrahedron letters (01.05.1998)
Get full text
Journal Article
Mitsunobu-like Processes with a Novel Triphenylphosphine-Cyclic Sulfamide Betaine
Castro, Jose L, Matassa, Victor G, Ball, Richard G
Published in Journal of organic chemistry (01.05.1994)
Published in Journal of organic chemistry (01.05.1994)
Get full text
Journal Article
1-(((7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo[2.2.1]heptan-1(S)-yl)methyl)sulfonyl)-4-(2-methylphenyl)piperazine (L-368,899): An Orally Bioavailable, Non-Peptide Oxytocin Antagonist with Potential Utility for Managing Preterm Labor
Williams, Peter D, Anderson, Paul S, Ball, Richard G, Bock, Mark G, Carroll, LeighAnne, Chiu, Shuet-Hing Lee, Clineschmidt, Bradley V, Culberson, J. Chris, Erb, Jill M
Published in Journal of medicinal chemistry (01.03.1994)
Published in Journal of medicinal chemistry (01.03.1994)
Get full text
Journal Article
Methoxylation of cocaine reduces binding affinity and produces compounds of differential binding and dopamine uptake inhibitory activity: discovery of a weak cocaine "antagonist"
Simoni, Daniele, Stoelwinder, Johannes, Kozikowski, Alan P, Johnson, Kenneth M, Bergmann, John S, Ball, Richard G
Published in Journal of medicinal chemistry (26.11.1993)
Published in Journal of medicinal chemistry (26.11.1993)
Get full text
Journal Article
Identification of 3,5-Dihydro-2-aryl-1H-pyrazolo[3,4-c]quinoline-1,4(2H)-diones as Novel High-Affinity Glycine Site N-Methyl-D-aspartate Antagonists
MacLeod, Angus M, Grimwood, Sarah, Barton, Cheryl, Bristow, Linda, Saywell, Kay L, Marshall, George R, Ball, Richard G
Published in Journal of medicinal chemistry (01.06.1995)
Published in Journal of medicinal chemistry (01.06.1995)
Get full text
Journal Article
Fusidienol A: A Novel Ras Farnesyl-Protein Transferase Inhibitor from Phoma sp
Singh, Sheo B, Ball, Richard G, Zink, Deborah L, Monaghan, Richard L, Polishook, Jon D, Sanchez, Manuel, Pelaez, Fernando, Silverman, Keith C, Lingham, Russell B
Published in Journal of organic chemistry (17.10.1997)
Published in Journal of organic chemistry (17.10.1997)
Get full text
Journal Article
5-(Piperidin-2-yl)- and 5-(Homopiperidin-2-yl)-1,4-benzodiazepines: High-Affinity, Basic Ligands for the Cholecystokinin-B Receptor
Castro, José L, Broughton, Howard B, Russell, Michael G. N, Rathbone, Denise, Watt, Alan P, Ball, Richard G, Chapman, Kerry L, Patel, Smita, Smith, Alison J, Marshall, George R, Matassa, Victor G
Published in Journal of medicinal chemistry (01.08.1997)
Published in Journal of medicinal chemistry (01.08.1997)
Get full text
Journal Article
Barceloneic Acid A, a New Farnesyl-Protein Transferase Inhibitor from a Phoma Species
Jayasuriya, Hiranthi, Ball, Richard G, Zink, Deborah L, Smith, Jack L, Goetz, Michael A, Jenkins, Rosalind G, Nallin-Omstead, Mary, Silverman, Keith C, Bills, Gerald F, Lingham, Russell B, Singh, Sheo B, Pelaez, Fernando, Cascales, Carmen
Published in Journal of natural products (Washington, D.C.) (01.07.1995)
Published in Journal of natural products (Washington, D.C.) (01.07.1995)
Get full text
Journal Article
HIV INTEGRASE INHIBITORS
SU DAI SHI, FISHER THORSTEN E, WAI JOHN S, CHOI ERIC J, WILLIAMS PETER D, DUBOST DAVID C, EMBREY MARK W, ISAACS RICHARD C. A, THOMPSON WAYNE J, PEI TAO, BALL RICHARD G, VENKATRAMAN SHANKAR, TRICE SARAH L
Year of Publication 16.06.2011
Get full text
Year of Publication 16.06.2011
Patent
Delineating the pharmacophoric elements of huperzine A: importance of the unsaturated three-carbon bridge to its AChE inhibitory activity
Kozikowski, Alan P, Miller, Chris P, Yamada, Fumio, Pang, Yuan Ping, Miller, Jacqueline H, McKinney, Michael, Ball, Richard G
Published in Journal of medicinal chemistry (01.12.1991)
Published in Journal of medicinal chemistry (01.12.1991)
Get full text
Journal Article
Highly potent, orally active diester macrocyclic human renin inhibitors
Weber, Ann E, Steiner, Mark G, Krieter, Philip A, Colletti, Adria E, Tata, James R, Halgren, Thomas A, Ball, Richard G, Doyle, John J, Schorn, Terry W
Published in Journal of medicinal chemistry (01.10.1992)
Published in Journal of medicinal chemistry (01.10.1992)
Get full text
Journal Article
Discovery of N -[(4 R )-6-(4-Chlorophenyl)-7-(2,4-dichlorophenyl)-2,2-dimethyl-3,4-dihydro-2 H -pyrano[2,3- b ]pyridin-4-yl]-5-methyl-1 H -pyrazole-3-carboxamide (MK-5596) as a Novel Cannabinoid-1 Receptor (CB1R) Inverse Agonist for the Treatment of Obesity
Yan, Lin, Huo, Pei, Debenham, John S., Madsen-Duggan, Christina B., Lao, Julie, Chen, Richard Z., Xiao, Jing Chen, Shen, Chun-Pyn, Stribling, D. Sloan, Shearman, Lauren P., Strack, Alison M., Tsou, Nancy, Ball, Richard G., Wang, Junying, Tong, Xinchun, Bateman, Thomas J., Reddy, Vijay B. G., Fong, Tung M., Hale, Jeffrey J.
Published in Journal of medicinal chemistry (27.05.2010)
Published in Journal of medicinal chemistry (27.05.2010)
Get full text
Journal Article
2-[(3a R ,4 R ,5 S ,7a S )-5-{(1 S )-1-[3,5-Bis(trifluoromethyl)phenyl]-2-hydroxyethoxy}-4-(2-methylphenyl)octahydro-2 H -isoindol-2-yl]-1,3-oxazol-4(5 H )-one: A Potent Human NK 1 Receptor Antagonist with Multiple Clearance Pathways
Kassick, Andrew J., Jiang, Jinlong, Bunda, Jaime, Wilson, David, Bao, Jianming, Lu, Huagang, Lin, Peter, Ball, Richard G., Doss, George A., Tong, Xinchun, Tsao, Kwei-Lan C., Wang, Hong, Chicchi, Gary, Karanam, Bindhu, Tschirret-Guth, Richard, Samuel, Koppara, Hora, Donald F., Kumar, Sanjeev, Madeira, Maria, Eng, Waisi, Hargreaves, Richard, Purcell, Mona, Gantert, Liza, Cook, Jacquelyn, DeVita, Robert J., Mills, Sander G.
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
Get full text
Journal Article