Targeting PIM2 by JP11646 results in significant antitumor effects in solid tumors
Katsuta, Eriko, Gil-Moore, Malgorzata, Moore, Justine, Yousif, Mohamed, Adjei, Alex A, Ding, Yi, Caserta, Justin, Baldino, Carmen M, Lee, Kelvin P, Gelman, Irwin H, Takabe, Kazuaki, Opyrchal, Mateusz
Published in International journal of oncology (01.10.2022)
Published in International journal of oncology (01.10.2022)
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Journal Article
Three-Component One-Pot Total Syntheses of Glyantrypine, Fumiquinazoline F, and Fiscalin B Promoted by Microwave Irradiation
Liu, Ji-Feng, Ye, Ping, Zhang, Bailin, Bi, Grace, Sargent, Katie, Yu, Libing, Yohannes, Daniel, Baldino, Carmen M
Published in Journal of organic chemistry (05.08.2005)
Published in Journal of organic chemistry (05.08.2005)
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Journal Article
Microwave-Promoted Suzuki Reactions of Aryl Chlorides in Aqueous Media
Miao, Guobin, Ye, Ping, Yu, Libing, Baldino, Carmen M.
Published in Journal of organic chemistry (18.03.2005)
Published in Journal of organic chemistry (18.03.2005)
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Journal Article
Novel One-Pot Total Syntheses of Deoxyvasicinone, Mackinazolinone, Isaindigotone, and Their Derivatives Promoted by Microwave Irradiation
Liu, Ji-Feng, Ye, Ping, Sprague, Kevin, Sargent, Katie, Yohannes, Daniel, Baldino, Carmen M, Wilson, Christopher J, Ng, Shi-Chung
Published in Organic letters (21.07.2005)
Published in Organic letters (21.07.2005)
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Journal Article
Microwave-Assisted Concise Total Syntheses of Quinazolinobenzodiazepine Alkaloids
Liu, Ji-Feng, Kaselj, Mira, Isome, Yuko, Chapnick, Jennifer, Zhang, Bailin, Bi, Grace, Yohannes, Daniel, Yu, Libing, Baldino, Carmen M
Published in Journal of organic chemistry (09.12.2005)
Published in Journal of organic chemistry (09.12.2005)
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Journal Article
Development of α-keto-based inhibitors of cruzain, a cysteine protease implicated in Chagas disease
Choe, Youngchool, Brinen, Linda S., Price, Mark S., Engel, Juan C., Lange, Meinolf, Grisostomi, Corinna, Weston, Scott G., Pallai, Peter V., Cheng, Hong, Hardy, Larry W., Hartsough, David S., McMakin, Marsha, Tilton, Robert F., Baldino, Carmen M., Craik, Charles S.
Published in Bioorganic & medicinal chemistry (15.03.2005)
Published in Bioorganic & medicinal chemistry (15.03.2005)
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Journal Article
The accelerated development of an optimized synthesis of 1,2,4-oxadiazoles: application of microwave irradiation and statistical design of experiments
Evans, Marc D, Ring, Jessica, Schoen, Adam, Bell, Andrew, Edwards, Paul, Berthelot, Didier, Nicewonger, Robb, Baldino, Carmen M
Published in Tetrahedron letters (22.12.2003)
Published in Tetrahedron letters (22.12.2003)
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Journal Article
Microwave-assisted one-pot synthesis of 2,3-disubstituted 3H-quinazolin-4-ones
Liu, JF, Lee, JY, Dalton, AM, Bi, G, Yu, LB, Baldino, CM, McElory, E, Brown, M
Published in Tetrahedron letters (21.02.2005)
Published in Tetrahedron letters (21.02.2005)
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Journal Article
Regioselective synthesis of [1,2,3]-triazoles catalyzed by Cu(I) generated in situ from Cu(0) nanosize activated powder and amine hydrochloride salts
Orgueira, Hernán A., Fokas, Demosthenes, Isome, Yuko, Chan, Philip C.-M., Baldino, Carmen M.
Published in Tetrahedron letters (18.04.2005)
Published in Tetrahedron letters (18.04.2005)
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Journal Article
Indoloprodigiosins from the C-10 bipyrrolic precursor: New antiproliferative prodigiosin analogs
Baldino, Carmen M., Parr, Jonathan, Wilson, Christopher J., Ng, Shi-Chung, Yohannes, Daniel, Wasserman, Harry H.
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Journal Article
Novel inhibition of PIM2 kinase has significant anti-tumor efficacy in multiple myeloma
Nair, J R, Caserta, J, Belko, K, Howell, T, Fetterly, G, Baldino, C, Lee, K P
Published in Leukemia (01.08.2017)
Published in Leukemia (01.08.2017)
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Journal Article
Abstract 5056: PIM-1 kinase regulates vitamin D receptor signaling in human renal carcinoma cells
Luo, Wei, Ma, Yingyu, Baldino, Carmen, Caserta, Justin, Ramakrishnan, Swathi, Roberto, Pili, Johnson, Candace, Trump, Donald
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Journal Article
A versatile synthesis of novel pan-PIM kinase inhibitors with initial SAR study
Flanders, Yvonne, Dumas, Stephane, Caserta, Justin, Nicewonger, Robb, Baldino, Michael, Lee, Chee-Seng, Baldino, Carmen M.
Published in Tetrahedron letters (03.06.2015)
Published in Tetrahedron letters (03.06.2015)
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Journal Article
Surviving the odds: targeting PIM2 in plasma cell survival (TUM10P.1051)
Nair, Jayakumar, Baldino, Carmen, Caserta, Justin, Carlson, Louise, Fetterly, Gerald, Lee, Kelvin
Published in The Journal of immunology (1950) (01.05.2015)
Published in The Journal of immunology (1950) (01.05.2015)
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Journal Article
Targeting the Serine-Threonine Kinase PIM2: Implications in IL-6 Mediated Survival in Myeloma
Nair, Jayakumar R, Howell, Tyger L, Caserta, Justin, Baldino, Carmen M, Fetterly, Gerald, Lee, Kelvin P
Published in Blood (06.12.2014)
Published in Blood (06.12.2014)
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Journal Article