An Efficient Synthesis of Enamides from Ketones
Zhao, Hang, Vandenbossche, Charles P, Koenig, Stefan G, Singh, Surendra P, Bakale, Roger P
Published in Organic letters (07.02.2008)
Published in Organic letters (07.02.2008)
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Journal Article
Development of a Process Route to the FAK/ALK Dual Inhibitor TEV-37440
Allwein, Shawn P, Mowrey, Dale R, Petrillo, Daniel E, Reif, James J, Purohit, Vikram C, Milkiewicz, Karen L, Bakale, Roger P, Christie, Michael A, Olsen, Mark A, Neville, Christopher J, Gilmartin, Gregory J
Published in Organic process research & development (19.05.2017)
Published in Organic process research & development (19.05.2017)
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Discovery and Process Synthesis of Novel 2,7-Pyrrolo[2,1-f][1,2,4]triazines
Thieu, Tho, Sclafani, Joseph A, Levy, Daniel V, McLean, Andrew, Breslin, Henry J, Ott, Gregory R, Bakale, Roger P, Dorsey, Bruce D
Published in Organic letters (19.08.2011)
Published in Organic letters (19.08.2011)
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Journal Article
The First Asymmetric Pilot-Scale Synthesis of TV-45070
Sclafani, Joseph A, Chen, Jian, Levy, Daniel V, Reese, Harlan, Dimitri, Mina, Mudipalli, Partha, Christie, Michael, Neville, Christopher J, Olsen, Mark, Bakale, Roger P
Published in Organic process research & development (20.10.2017)
Published in Organic process research & development (20.10.2017)
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Journal Article
A General Preparation of Protected Phosphoamino Acids
Petrillo, Daniel E, Mowrey, Dale R, Allwein, Shawn P, Bakale, Roger P
Published in Organic letters (02.03.2012)
Published in Organic letters (02.03.2012)
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Journal Article
A Facile Deprotection of Secondary Acetamides
Koenig, Stefan G, Vandenbossche, Charles P, Zhao, Hang, Mousaw, Patrick, Singh, Surendra P, Bakale, Roger P
Published in Organic letters (15.01.2009)
Published in Organic letters (15.01.2009)
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Journal Article
Development and Scale-Up of an Optimized Route to the ALK Inhibitor CEP-28122
Allwein, Shawn P, Roemmele, Renee C, Haley, James J, Mowrey, Dale R, Petrillo, Daniel E, Reif, James J, Gingrich, Diane E, Bakale, Roger P
Published in Organic process research & development (20.01.2012)
Published in Organic process research & development (20.01.2012)
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Journal Article
Development of a Large-Scale Stereoselective Process for (1R,4S)-4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-1-amine Hydrochloride
Han, Zhengxu, Koenig, Stefan G, Zhao, Hang, Su, Xiping, Singh, Surendra P, Bakale, Roger P
Published in Organic process research & development (01.07.2007)
Published in Organic process research & development (01.07.2007)
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Journal Article
Demonstration of a Scalable One-Pot Synthesis of Fmoc‑O‑Benzylphospho‑l‑serine
Mowrey, Dale R, Petrillo, Daniel E, Allwein, Shawn P, Graf, Stéphanie, Bakale, Roger P
Published in Organic process research & development (16.11.2012)
Published in Organic process research & development (16.11.2012)
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Journal Article
Formation of (S)-5-Cyclohexyl-5-phenyl-1,3-dioxolane-2,4-dione: A Key Intermediate in the Synthesis of (S)-Oxybutynin Hydrochloride
Vandenbossche, Charles P, de Croos, Philomen, Singh, Surendra P, Bakale, Roger P, Wagler, Thomas R
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
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Journal Article
Control of Diastereoselectivity by Solvent Effects in the Addition of Grignard Reagents to Enantiopure t-Butylsulfinimine: Syntheses of the Stereoisomers of the Hydroxyl Derivatives of Sibutramine
Lu, Bruce Z, Senanayake, Chris, Li, Nansheng, Han, Zhengxu, Bakale, Roger P, Wald, Stephen A
Published in Organic letters (23.06.2005)
Published in Organic letters (23.06.2005)
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Journal Article
Remarkably selective palladium-catalyzed amination process: Rapid assembly of multiamino based structures
Hong, Yaping, Senanayake, Chris H., Xiang, Tingjian, Vandenbossche, Charles P., Tanoury, Gerald J., Bakale, Roger P., Wald, Stephen A.
Published in Tetrahedron letters (14.05.1998)
Published in Tetrahedron letters (14.05.1998)
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Journal Article
Palladium catalyzed amination of 2-chloro-1,3-azole derivatives: Mild entry to potent H1- antihistaminic norastemizole
Hong, Yaping, Tanoury, Gerald J., Wilkinson, H.Scott, Bakale, Roger P., Wald, Stephen A., Senanayake, Chris H.
Published in Tetrahedron letters (01.08.1997)
Published in Tetrahedron letters (01.08.1997)
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Journal Article
A large-scale asymmetric synthesis of ( S)-cyclohexylphenyl glycolic acid
Su, Xiping, Bhongle, Nandkumar N, Pflum, Derek, Butler, Hal, Wald, Stephen A, Bakale, Roger P, Senanayake, Chris H
Published in Tetrahedron: asymmetry (14.11.2003)
Published in Tetrahedron: asymmetry (14.11.2003)
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