Unexpected Intermolecular Pd-Catalyzed Cross-Coupling Reaction Employing Heteroaromatic Carboxylic Acids as Coupling Partners
Forgione, Pat, Brochu, Marie-Christine, St-Onge, Miguel, Thesen, Kris H, Bailey, Murray D, Bilodeau, François
Published in Journal of the American Chemical Society (06.09.2006)
Published in Journal of the American Chemical Society (06.09.2006)
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Journal Article
Preclinical Profile of BI 224436, a Novel HIV-1 Non-Catalytic-Site Integrase Inhibitor
FENWICK, Craig, AMAD, Ma'an, FADER, Lee D, FAUCHER, Anne-Marie, GARNEAU, Michel, JAKALIAN, Araz, KAWAI, Stephen, LAMORTE, Louie, LAPLANTE, Steven, LAIBIN LUO, MASON, Steve, POUPART, Marc-André, BAILEY, Murray D, RIOUX, Nathalie, SCHROEDER, Patricia, SIMONEAU, Bruno, TREMBLAY, Sonia, TSANTRIZOS, Youla, WITVROUW, Myriam, YOAKIM, Christiane, BETHELL, Richard, BÖS, Michael, BONNEAU, Pierre, CORDINGLEY, Michael, COULOMBE, René, DUAN, Jianmin, EDWARDS, Paul
Published in Antimicrobial agents and chemotherapy (01.06.2014)
Published in Antimicrobial agents and chemotherapy (01.06.2014)
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Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV‑1
Fader, Lee D, Malenfant, Eric, Parisien, Mathieu, Carson, Rebekah, Bilodeau, François, Landry, Serge, Pesant, Marc, Brochu, Christian, Morin, Sébastien, Chabot, Catherine, Halmos, Ted, Bousquet, Yves, Bailey, Murray D, Kawai, Stephen H, Coulombe, René, LaPlante, Steven, Jakalian, Araz, Bhardwaj, Punit K, Wernic, Dominik, Schroeder, Patricia, Amad, Ma’an, Edwards, Paul, Garneau, Michel, Duan, Jianmin, Cordingley, Michael, Bethell, Richard, Mason, Stephen W, Bös, Michael, Bonneau, Pierre, Poupart, Marc-André, Faucher, Anne-Marie, Simoneau, Bruno, Fenwick, Craig, Yoakim, Christiane, Tsantrizos, Youla
Published in ACS medicinal chemistry letters (10.04.2014)
Published in ACS medicinal chemistry letters (10.04.2014)
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Journal Article
Synthesis of (1R,2S)-1-Amino-2-vinylcyclopropanecarboxylic Acid Vinyl-ACCA) Derivatives: Key Intermediates for the Preparation of Inhibitors of the Hepatitis C Virus NS3 Protease
Beaulieu, Pierre L, Gillard, James, Bailey, Murray D, Boucher, Colette, Duceppe, Jean-Simon, Simoneau, Bruno, Wang, Xiao-Jun, Zhang, Li, Grozinger, Karl, Houpis, Ioannis, Farina, Vittorio, Heimroth, Heidi, Krueger, Thomas, Schnaubelt, Jürgen
Published in Journal of organic chemistry (22.07.2005)
Published in Journal of organic chemistry (22.07.2005)
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Minimizing the Contribution of Enterohepatic Recirculation to Clearance in Rat for the NCINI Class of Inhibitors of HIV
Fader, Lee D, Carson, Rebekah, Morin, Sébastien, Bilodeau, François, Chabot, Catherine, Halmos, Ted, Bailey, Murray D, Kawai, Stephen H, Coulombe, René, Laplante, Steven, Mekhssian, Kevork, Jakalian, Araz, Garneau, Michel, Duan, Jianmin, Mason, Stephen W, Simoneau, Bruno, Fenwick, Craig, Tsantrizos, Youla, Yoakim, Christiane
Published in ACS medicinal chemistry letters (12.06.2014)
Published in ACS medicinal chemistry letters (12.06.2014)
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Journal Article
The Use of Chemical Double-Mutant Cycles in Biomolecular Recognition Studies: Application to HCV NS3 Protease Inhibitors
Kawai, Stephen H., Bailey, Murray D., Halmos, Ted, Forgione, Pat, LaPlante, Steven R., Llinàs-Brunet, Montse, Naud, Julie, Goudreau, Natalie
Published in ChemMedChem (17.11.2008)
Published in ChemMedChem (17.11.2008)
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Journal Article
Discovery of a Potent and Selective Noncovalent Linear Inhibitor of the Hepatitis C Virus NS3 Protease (BI 201335)
Llinàs-Brunet, Montse, Bailey, Murray D, Goudreau, Nathalie, Bhardwaj, Punit K, Bordeleau, Josée, Bös, Michael, Bousquet, Yves, Cordingley, Michael G, Duan, Jiamin, Forgione, Pat, Garneau, Michel, Ghiro, Elise, Gorys, Vida, Goulet, Sylvie, Halmos, Ted, Kawai, Stephen H, Naud, Julie, Poupart, Marc-André, White, Peter W
Published in Journal of medicinal chemistry (09.09.2010)
Published in Journal of medicinal chemistry (09.09.2010)
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Journal Article
A Systematic Approach to the Optimization of Substrate-Based Inhibitors of the Hepatitis C Virus NS3 Protease: Discovery of Potent and Specific Tripeptide Inhibitors
Llinàs-Brunet, Montse, Bailey, Murray D, Ghiro, Elise, Gorys, Vida, Halmos, Ted, Poirier, Martin, Rancourt, Jean, Goudreau, Nathalie
Published in Journal of medicinal chemistry (16.12.2004)
Published in Journal of medicinal chemistry (16.12.2004)
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Journal Article
Structure−Activity Study on a Novel Series of Macrocyclic Inhibitors of the Hepatitis C Virus NS3 Protease Leading to the Discovery of BILN 2061
Llinàs-Brunet, Montse, Bailey, Murray D, Bolger, Gordon, Brochu, Christian, Faucher, Anne-Marie, Ferland, Jean Marie, Garneau, Michel, Ghiro, Elise, Gorys, Vida, Grand-Maître, Chantal, Halmos, Ted, Lapeyre-Paquette, Nicole, Liard, Francine, Poirier, Martin, Rhéaume, Manon, Tsantrizos, Youla S, Lamarre, Daniel
Published in Journal of medicinal chemistry (25.03.2004)
Published in Journal of medicinal chemistry (25.03.2004)
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Journal Article
Synthesis of BILN 2061, an HCV NS3 Protease Inhibitor with Proven Antiviral Effect in Humans
Faucher, Anne-Marie, Bailey, Murray D, Beaulieu, Pierre L, Brochu, Christian, Duceppe, Jean-Simon, Ferland, Jean-Marie, Ghiro, Elise, Gorys, Vida, Halmos, Ted, Kawai, Stephen H, Poirier, Martin, Simoneau, Bruno, Tsantrizos, Youla S, Llinàs-Brunet, Montse
Published in Organic letters (19.08.2004)
Published in Organic letters (19.08.2004)
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Journal Article
Synthesis and optimization of a novel series of HCV NS3 protease inhibitors: 4-Arylproline analogs
Bilodeau, François, Bailey, Murray D., Bhardwaj, Punit K., Bordeleau, Josée, Forgione, Pat, Garneau, Michel, Ghiro, Elise, Gorys, Vida, Halmos, Ted, Jolicoeur, Eric S., Leblanc, Mélissa, Lemke, Christopher T., Naud, Julie, O’Meara, Jeff, White, Peter W., Llinàs-Brunet, Montse
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
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Journal Article
Peptide backbone replacement of hepatitis C virus NS3 serine protease C-terminal cleavage product analogs: Discovery of potent succinamide inhibitors
Bailey, Murray D., Bordeleau, Josée, Garneau, Michel, Leblanc, Mélissa, Lemke, Christopher T., O’Meara, Jeff, White, Peter W., Llinàs-Brunet, Montse
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
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Journal Article
Novel Azapeptide Inhibitors of Hepatitis C Virus Serine Protease
Bailey, Murray D, Halmos, Ted, Goudreau, Nathalie, Lescop, Ewen, Llinàs-Brunet, Montse
Published in Journal of medicinal chemistry (15.07.2004)
Published in Journal of medicinal chemistry (15.07.2004)
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Journal Article
INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION
FADER LEE, SURPRENANT SIMON, MORIN SEBASTIEN, TSANTRIZOS YOULA S, KAWAI STEPHEN, BILODEAU FRANCOIS, SIMONEAU BRUNO, THIBEAULT CARL, BAILEY MURRAY D, CARSON REBEKAH J, YOAKIM CHRISTIANE, LAPLANTE STEVEN
Year of Publication 06.02.2014
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Year of Publication 06.02.2014
Patent
INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION
FADER LEE, HALMOS TEDDY, POUPART MARC ANDRE, BILODEAU FRANCOIS, SIMONEAU BRUNO, LANDRY SERGE, MORIN SEBASTIEN, TSANTRIZOS YOULA S, KAWAI STEPHEN, COULOMBE RENE, PARISIEN MATHIEU, BAILEY MURRAY D, CARSON REBEKAH J, LAPLANTE STEVEN
Year of Publication 02.09.2010
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Year of Publication 02.09.2010
Patent
Nitro-olefin bicycloannulation: one-step synthesis of tricyclo[3.2.1.02,7]octan-6-ones from cyclohexenones and of tricyclo[2.2.1.02,6]heptan-3-ones from cyclopentenones
Cory, Robert M, Anderson, Paul C, Bailey, Murray D, McLaren, Fred R, Renneboog, Richard M, Yamamoto, Brian R
Published in Canadian journal of chemistry (01.10.1985)
Published in Canadian journal of chemistry (01.10.1985)
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Journal Article
Chemo-enzymatic synthesis of chiral 2-substituted succinic acid derivatives
Bailey, Murray D., Halmos, Ted, Adamson, Dan, Bordeleau, Josée, Grand-Maı̂tre, Chantal
Published in Tetrahedron: asymmetry (27.08.1999)
Published in Tetrahedron: asymmetry (27.08.1999)
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