Design and Synthesis of Novel Aminoindazole-pyrrolo[2,3- b ]pyridine Inhibitors of IKKα That Selectively Perturb Cellular Non-Canonical NF-κB Signalling
Riley, Christopher, Ammar, Usama, Alsfouk, Aisha, Anthony, Nahoum G, Baiget, Jessica, Berretta, Giacomo, Breen, David, Huggan, Judith, Lawson, Christopher, McIntosh, Kathryn, Plevin, Robin, Suckling, Colin J, Young, Louise C, Paul, Andrew, Mackay, Simon P
Published in Molecules (Basel, Switzerland) (01.08.2024)
Published in Molecules (Basel, Switzerland) (01.08.2024)
Get full text
Journal Article
Easy-To-Synthesize Spirocyclic Compounds Possess Remarkable in Vivo Activity against Mycobacterium tuberculosis
Guardia, Ana, Baiget, Jessica, Cacho, Mónica, Pérez, Arancha, Ortega-Guerra, Montserrat, Nxumalo, Winston, Khanye, Setshaba D, Rullas, Joaquín, Ortega, Fátima, Jiménez, Elena, Pérez-Herrán, Esther, Fraile-Gabaldón, María Teresa, Esquivias, Jorge, Fernández, Raquel, Porras-De Francisco, Esther, Encinas, Lourdes, Alonso, Marta, Giordano, Ilaria, Rivero, Cristina, Miguel-Siles, Juan, Osende, Javier G, Badiola, Katrina A, Rutledge, Peter J, Todd, Matthew H, Remuiñán, Modesto, Alemparte, Carlos
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
Get full text
Journal Article
Manganese dioxide mediated one-pot synthesis of methyl 9H-pyrido[3,4-b]indole-1-carboxylate: Concise synthesis of alangiobussinine
Baiget, Jessica, Llona-Minguez, Sabin, Lang, Stuart, Mackay, Simon P, Suckling, Colin J, Sutcliffe, Oliver B
Published in Beilstein journal of organic chemistry (12.10.2011)
Published in Beilstein journal of organic chemistry (12.10.2011)
Get full text
Journal Article
Design and Synthesis of Novel Aminoindazole-pyrrolo2,3-bpyridine Inhibitors of IKKα That Selectively Perturb Cellular Non-Canonical NF-κB Signalling
Riley, Christopher, Ammar, Usama, Alsfouk, Aisha, Anthony, Nahoum G, Baiget, Jessica, Berretta, Giacomo, Breen, David, Huggan, Judith, Lawson, Christopher, McIntosh, Kathryn, Plevin, Robin, Suckling, Colin J, Young, Louise C, Paul, Andrew, Mackay, Simon P
Published in Molecules (Basel, Switzerland) (26.07.2024)
Published in Molecules (Basel, Switzerland) (26.07.2024)
Get full text
Journal Article
Topographical Mapping of Isoform-Selectivity Determinants for J‑Channel-Binding Inhibitors of Sphingosine Kinases 1 and 2
Adams, David R, Tawati, Salha, Berretta, Giacomo, Rivas, Paula Lopez, Baiget, Jessica, Jiang, Zhong, Alsfouk, Aisha, Mackay, Simon P, Pyne, Nigel J, Pyne, Susan
Published in Journal of medicinal chemistry (11.04.2019)
Published in Journal of medicinal chemistry (11.04.2019)
Get full text
Journal Article
Inhibitory Kappa B Kinase α (IKKα) Inhibitors That Recapitulate Their Selectivity in Cells against Isoform-Related Biomarkers
Anthony, Nahoum G, Baiget, Jessica, Berretta, Giacomo, Boyd, Marie, Breen, David, Edwards, Joanne, Gamble, Carly, Gray, Alexander I, Harvey, Alan L, Hatziieremia, Sophia, Ho, Ka Ho, Huggan, Judith K, Lang, Stuart, Llona-Minguez, Sabin, Luo, Jia Lin, McIntosh, Kathryn, Paul, Andrew, Plevin, Robin J, Robertson, Murray N, Scott, Rebecca, Suckling, Colin J, Sutcliffe, Oliver B, Young, Louise C, Mackay, Simon P
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
Get full text
Journal Article
Small-molecule inhibitors of IκB kinase (IKK) and IKK-related kinases
Llona-Minguez, Sabin, Baiget, Jessica, Mackay, Simon P
Published in Pharmaceutical patent analyst (01.07.2013)
Published in Pharmaceutical patent analyst (01.07.2013)
Get more information
Journal Article
Manganese dioxide mediated one-pot synthesis of methyl 9 H -pyrido[3,4- b ]indole-1-carboxylate: Concise synthesis of alangiobussinine
Baiget, Jessica, Llona-Minguez, Sabin, Lang, Stuart, MacKay, Simon P, Suckling, Colin J, Sutcliffe, Oliver B
Published in Beilstein journal of organic chemistry (12.10.2011)
Published in Beilstein journal of organic chemistry (12.10.2011)
Get full text
Journal Article
PRODRUGS OF OPICAPONE
BAIGET, Jessica, BELIAEV, Alexander, HOLENZ, Joerg, KISS, Laszlo, KAROLI, Tomislav, BARROCAS, Pedro, REVUNOV, Evgeny
Year of Publication 03.10.2024
Get full text
Year of Publication 03.10.2024
Patent
PRODRUGS OF OPICAPONE
BAIGET, Jessica, BELIAEV, Alexander, HOLENZ, Joerg, KISS, Laszlo, KAROLI, Tomislav, BARROCAS, Pedro, REVUNOV, Evgeny
Year of Publication 05.10.2023
Get full text
Year of Publication 05.10.2023
Patent
IKK INHIBITORS
BERRETTA, Giacomo, MASCI, Domiziana, BREEN, David, SUCKLING, Colin J, ALSFOUK, Aisha A, LLONA-MINGUEZ, Sabin, RILEY, Christopher, BAIGET, Jessica, LAWSON, Christopher, ANTHONY, Nahoum G, WEST, Christopher, AMMAR, Usama, HUGGAN, Judith, MACKAY, Simon P
Year of Publication 16.11.2023
Get full text
Year of Publication 16.11.2023
Patent
Prodrugs of OPICAPONE
KAROLI, TOMISLAV, BARROCAS, PEDRO, REVUNOV, EVGENY, BELIAEV, ALEXANDER, HOLENZ, JOERG, BAIGET, JESSICA, KISS, LASZLO
Year of Publication 01.02.2024
Get full text
Year of Publication 01.02.2024
Patent