ZY15557, a novel, long acting inhibitor of dipeptidyl peptidase‐4, for the treatment of Type 2 diabetes mellitus
Jain, Mukul R, Joharapurkar, Amit A, Kshirsagar, Samadhan G, Patel, Vishal J, Bahekar, Rajesh H, Patel, Harilal V, Jadav, Pradip A, Patel, Pankaj R, Desai, Ranjit C
Published in British journal of pharmacology (01.07.2017)
Published in British journal of pharmacology (01.07.2017)
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Journal Article
Synthesis and antidiabetic activity of 2,5-disubstituted-3-imidazol-2-yl-pyrrolo[2,3- b]pyridines and thieno[2,3- b]pyridines
Bahekar, Rajesh H., Jain, Mukul R., Jadav, Pradip A., Prajapati, Vijay M., Patel, Dipam N., Gupta, Arun A., Sharma, Ajay, Tom, Robby, Bandyopadhya, Debdutta, Modi, Honey, Patel, Pankaj R.
Published in Bioorganic & medicinal chemistry (01.11.2007)
Published in Bioorganic & medicinal chemistry (01.11.2007)
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Journal Article
Co-agonist of glucagon and GLP-1 reduces cholesterol and improves insulin sensitivity independent of its effect on appetite and body weight in diet-induced obese C57 mice
Patel, Vishal, Joharapurkar, Amit, Dhanesha, Nirav, Kshirsagar, Samadhan, Patel, Kartik, Bahekar, Rajesh, Shah, Gaurang, Jain, Mukul
Published in Canadian journal of physiology and pharmacology (01.12.2013)
Published in Canadian journal of physiology and pharmacology (01.12.2013)
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Journal Article
Coagonist of GLP-1 and Glucagon Receptor Ameliorates Development of Non-Alcoholic Fatty Liver Disease
Patel, Vishal, Joharapurkar, Amit, Kshirsagar, Samadhan, Sutariya, Brijesh, Patel, Maulik, Patel, Hiren, Pandey, Dheerendra, Patel, Dipam, Ranvir, Ramchandra, Kadam, Shekhar, Bahekar, Rajesh, Jain, Mukul
Published in Cardiovascular & hematological agents in medicinal chemistry (2018)
Published in Cardiovascular & hematological agents in medicinal chemistry (2018)
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Journal Article
Activation of GLP-1 and Glucagon Receptors Regulates Bile Homeostasis Independent of Thyroid Hormone
Patel, Vishal J, Joharapurkar, Amit A, Kshirsagar, Samadhan G, Sutariya, Brijesh K, Patel, Maulik S, Bahekar, Rajesh H, Jain, Mukul R
Published in Current molecular pharmacology (01.01.2019)
Published in Current molecular pharmacology (01.01.2019)
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Journal Article
Design, synthesis, and biological evaluation of substituted- N-(thieno[2,3- b]pyridin-3-yl)-guanidines, N-(1 H-pyrrolo[2,3- b]pyridin-3-yl)-guanidines, and N-(1 H-indol-3-yl)-guanidines
Bahekar, Rajesh H., Jain, Mukul R., Goel, Ashish, Patel, Dipam N., Prajapati, Vijay M., Gupta, Arun A., Jadav, Pradip A., Patel, Pankaj R.
Published in Bioorganic & medicinal chemistry (01.05.2007)
Published in Bioorganic & medicinal chemistry (01.05.2007)
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Journal Article
ZYBT1, a potent, irreversible Bruton’s Tyrosine Kinase (BTK) inhibitor that inhibits the C481S BTK with profound efficacy against arthritis and cancer
Ghoshdastidar, Krishnarup, Patel, Hoshang, Bhayani, Hitesh, Patel, Ankit, Thakkar, Kinjal, Patel, Dinesh, Sharma, Manoranjan, Singh, Jaideep, Mohapatra, Jogeswar, Chatterjee, Abhijit, Patel, Dipam, Bahekar, Rajesh, Sharma, Rajiv, Gupta, Lakshmikant, Patel, Nirmal, Giri, Poonam, Srinivas, Nuggehally R., Jain, Mukul, Bandyopadhyay, Debdutta, Patel, Pankaj R., Desai, Ranjit C.
Published in Pharmacology research & perspectives (01.08.2020)
Published in Pharmacology research & perspectives (01.08.2020)
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Journal Article
Synthesis and preliminary evaluation of some N-[5-(2-furanyl)-2-methyl-4-oxo-4H-thieno[2,3-d]pyrimidin-3-yl]-carboxamide and 3-substituted-5-(2-furanyl)-2-methyl-3H-thieno[2,3-d]pyrimidin-4-ones as antimicrobial agents
Chambhare, RV, Khadse, BG, Bobde, AS, Bahekar, RH
Published in European journal of medicinal chemistry (01.01.2003)
Published in European journal of medicinal chemistry (01.01.2003)
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Journal Article
Coagonist of glucagon-like peptide-1 and glucagon receptors ameliorates kidney injury in murine models of obesity and diabetes mellitus
Patel, Vishal J, Joharapurkar, Amit A, Kshirsagar, Samadhan G, Sutariya, Brijesh K, Patel, Maulik S, Patel, Hiren M, Pandey, Dheerendra K, Bahekar, Rajesh H, Jain, Mukul R
Published in World journal of diabetes (15.06.2018)
Published in World journal of diabetes (15.06.2018)
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Journal Article
Omeprazole improves the anti-obesity and antidiabetic effects of exendin-4 in db/db mice (奥美拉唑改善唾液素-4 对db/db小鼠的减肥与降糖作用)
Patel, Vishal, Joharapurkar, Amit, Gandhi, Tejal, Patel, Kirti, Dhanesha, Nirav, Kshirsagar, Samadhan, Dhote, Vipin, Detroja, Jaysukh, Bahekar, Rajesh, Jain, Mukul
Published in Journal of diabetes (01.06.2013)
Published in Journal of diabetes (01.06.2013)
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Journal Article
Pharmacological characterization of ZYDPLA1, a novel long-acting dipeptidyl peptidase-4 inhibitor
Jain, Mukul R., Joharapurkar, Amit A., Bahekar, Rajesh H., Patel, Harilal, Jadav, Pradip, Kshirsagar, Samadhan G., Patel, Vishal J., Patel, Kartikkumar N., Ramanathan, Vikram K., Patel, Pankaj R., Desai, Ranjit C.
Published in Journal of diabetes (01.09.2015)
Published in Journal of diabetes (01.09.2015)
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Journal Article
Discovery of Orally Active, Potent, and Selective Benzotriazole-Based PTP1B Inhibitors
Patel, Dipam, Jain, Mukul, Shah, Shailesh R., Bahekar, Rajesh, Jadav, Pradip, Darji, Brijesh, Siriki, Yernaidu, Bandyopadhyay, Debdutta, Joharapurkar, Amit, Kshirsagar, Samadhan, Patel, Harilal, Shaikh, Mubeen, Sairam, Kalapatapu V. V. M., Patel, Pankaj
Published in ChemMedChem (06.06.2011)
Published in ChemMedChem (06.06.2011)
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Journal Article
Synthesis of 3,8,9-trisubstituted-1,7,9-triaza-fluorene-6-carboxylic acid derivatives as a new class of insulin secretagogues
Bahekar, Rajesh H., Jain, Mukul R., Jadav, Pradip A., Goel, Ashish, Patel, Dipam N., Prajapati, Vijay M., Gupta, Arun A., Modi, Honey, Patel, Pankaj R.
Published in Bioorganic & medicinal chemistry (01.09.2007)
Published in Bioorganic & medicinal chemistry (01.09.2007)
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Journal Article
Peptidomimetics as potent and selective PTP1B inhibitors
Patel, Dipam, Jain, Mukul, Shah, Shailesh R, Bahekar, Rajesh, Jadav, Pradip, Shah, Kiran, Joharapurkar, Amit, Shaikh, Mubeen, Sairam, Kalapatapu V V M
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.08.2013)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.08.2013)
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Journal Article
Synthesis and Antidiabetic Activity of 3,6,7-Trisubstituted-2-(1H-imidazol-2-ylsulfanyl)quinoxalines and Quinoxalin-2-yl isothioureas
Bahekar, Rajesh H., Jain, Mukul R., Gupta, Arun A., Goel, Ashish, Jadav, Pradip A., Patel, Dipam N., Prajapati, Vijay M., Patel, Pankaj R.
Published in Archiv der Pharmazie (Weinheim) (01.07.2007)
Published in Archiv der Pharmazie (Weinheim) (01.07.2007)
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Journal Article
Evaluation of Cardioprotective Effect of 3,5,3'-Tri-iodo-L-thyronine in Isoproterenol-Induced Cardiotoxicity
Mishra, Vinay, Ghumatkar, Priya, Patel, Maulik V., Devada, Shilpesh, Ranvir, Ramchandra, Swain, Prabodha, Sundar, Rajesh, Bahekar, Rajesh, Jain, Mukul R.
Published in International Journal of Endocrinology (01.01.2011)
Published in International Journal of Endocrinology (01.01.2011)
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Journal Article
신규한 오토택신 억제제
BAHEKAR RAJESH, PRAJAPATI VIJAY, DAVE KAMAL, JOSHI DARSHAN, SHARMA RAJIV
Year of Publication 05.09.2023
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Year of Publication 05.09.2023
Patent
ZYKR1, a novel, potent, and peripherally selective kappa opioid receptor agonist reduces visceral pain and pruritus in animal models
Jain, Mukul R., Patel, Rakesh B., Prajapati, Kanaiyalal D., Vyas, Purvi, Bandyopadhyay, Debdutta, Prajapati, Vijay, Bahekar, Rajesh, Patel, Prakash N., Kawade, Harish M., Kokare, Dadasaheb M., Pawar, Vishwanath, Desai, Ranjit
Published in European journal of pharmacology (05.06.2022)
Published in European journal of pharmacology (05.06.2022)
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