Discovery of BAY-390, a Selective CNS Penetrant Chemical Probe as Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonist
Mesch, Stefanie, Walter, Daryl, Laux-Biehlmann, Alexis, Basting, Daniel, Flanagan, Stuart, Miyatake Ondozabal, Hideki, Bäurle, Stefan, Pearson, Christopher, Jenkins, James, Elves, Philip, Hess, Stephen, Coelho, Anne-Marie, Rotgeri, Andrea, Bothe, Ulrich, Nawaz, Schanila, Zollner, Thomas M., Steinmeyer, Andreas
Published in Journal of medicinal chemistry (26.01.2023)
Published in Journal of medicinal chemistry (26.01.2023)
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Journal Article
Discovery and In Vitro Characterization of BAY 2686013, an Allosteric Small Molecule Antagonist of the Human Pituitary Adenylate Cyclase-Activating Polypeptide Receptor
Langer, Gernot, Scott, John, Lind, Christoffer, Otto, Christiane, Bothe, Ulrich, Laux-Biehlmann, Alexis, Müller, Jörg, le Roy, Beau, Irlbacher, Horst, Nowak-Reppel, Katrin, Schlüter, Anne, Davenport, Adam J, Slack, Mark, Bäurle, Stefan
Published in Molecular pharmacology (01.09.2023)
Published in Molecular pharmacology (01.09.2023)
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Discovery and Characterization of BAY 1214784, an Orally Available Spiroindoline Derivative Acting as a Potent and Selective Antagonist of the Human Gonadotropin-Releasing Hormone Receptor as Proven in a First-In-Human Study in Postmenopausal Women
Panknin, Olaf, Wagenfeld, Andrea, Bone, Wilhelm, Bender, Eckhard, Nowak-Reppel, Katrin, Fernández-Montalván, Amaury E, Nubbemeyer, Reinhard, Bäurle, Stefan, Ring, Sven, Schmees, Norbert, Prien, Olaf, Schäfer, Martina, Friedrich, Christian, Zollner, Thomas M, Steinmeyer, Andreas, Mueller, Thomas, Langer, Gernot
Published in Journal of medicinal chemistry (22.10.2020)
Published in Journal of medicinal chemistry (22.10.2020)
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Journal Article
Identification of a Benzimidazolecarboxylic Acid Derivative (BAY 1316957) as a Potent and Selective Human Prostaglandin E2 Receptor Subtype 4 (hEP4-R) Antagonist for the Treatment of Endometriosis
Bäurle, Stefan, Nagel, Jens, Peters, Olaf, Bräuer, Nico, ter Laak, Antonius, Preusse, Cornelia, Rottmann, Antje, Heldmann, Dieter, Bothe, Ulrich, Blume, Thorsten, Zorn, Ludwig, Walter, Daryl, Zollner, Thomas M, Steinmeyer, Andreas, Langer, Gernot
Published in Journal of medicinal chemistry (14.03.2019)
Published in Journal of medicinal chemistry (14.03.2019)
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특정 안구 장애를 치료하기 위한, P2X4 수용체 길항 활성을 갖는 N-페닐아세트아미드의 용도
CHEN MINJIE, FINIS DAVID, SEO STEFANIE, BAEURLE STEFAN, NAGEL JENS, YIU SAMUEL, TERJUNG CARSTEN, LIN HUI, SCHUBERT WILLIAM
Year of Publication 07.03.2023
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Year of Publication 07.03.2023
Patent
P2X4 수용체 길항 활성을 갖는 치환된 N-페닐아세트아미드
SCOTT ROBERT JOHN, BAEURLE STEFAN, RING SVEN, WALTER DARYL SIMON, LAUX BIEHLMANN ALEXIS, WITTROCK SVEN, NAGEL JENS, POOK ELISABETH, NUBBEMEYER REINHARD
Year of Publication 07.03.2023
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Year of Publication 07.03.2023
Patent
브라디키닌 B1 수용체의 길항제로서의 카르복실산 방향족 아미드
GROETICKE INA, ROTGERI ANDREA, BAEURLE STEFAN, NAGEL JENS, SCHMIDT NICOLE, DAVENPORT ADAM JAMES, DYRKS THOMAS, KLAR JUERGEN, STIMSON CHRISTOPHER, RAUSCH ALEXANDRA
Year of Publication 29.08.2019
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Year of Publication 29.08.2019
Patent
SPIROINDOLINE DERIVATIVES FOR USE AS GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS
PANKNIN OLAF, RING SVEN, BAEURLE STEFAN, WAGENFELD ANDREA, LANGER GERNOT, NUBBEMEYER REINHARD, NOWAK REPPEL KATRIN
Year of Publication 14.12.2015
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Year of Publication 14.12.2015
Patent
A CONTROLLER, AND A POWER SUPPLY
ZHANG GUANGCHAO DARSON, ODELL ARTHUR B, BAEURLE STEFAN, MAO MINGMING, ZHANG MICHAEL YUE, DENG EDWARD
Year of Publication 09.01.2014
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Year of Publication 09.01.2014
Patent