Piperidine-based heterocyclic oxalyl amides as potent p38α MAP kinase inhibitors
Mavunkel, Babu J., Perumattam, John J., Tan, Xuefei, Luedtke, Gregory R., Lu, Qing, Lim, Don, Kizer, Darin, Dugar, Sundeep, Chakravarty, Sarvajit, Xu, Yong-jin, Jung, Joon, Liclican, Albert, Levy, Daniel E., Tabora, Jocelyn
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Design and synthesis of piperazine-indole p38α MAP kinase inhibitors with improved pharmacokinetic profiles
Tan, Xuefei, Tester, Richland W., Luedtke, Gregory R., Chakravarty, Sarvajit, Mavunkel, Babu J., Perumattam, John J., Lu, Qing, Nashashibi, Imad, Jung, Joon, Hu, Jie, Liclican, Albert, Almirez, Ramona, Tabora, Jocelyn, Tran, Vinh, Laney, Maureen, Levy, Daniel E., Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Indole-based heterocyclic inhibitors of p38α MAP kinase: designing a conformationally restricted analogue
Mavunkel, Babu J, Chakravarty, Sarvajit, Perumattam, John J, Luedtke, Gregory R, Liang, Xi, Lim, Don, Xu, Yong-jin, Laney, Maureen, Liu, David Y, Schreiner, George F, Lewicki, John A, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (2003)
Published in Bioorganic & medicinal chemistry letters (2003)
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Journal Article
Pharmacological Properties of SD-282 – An α-Isoform Selective Inhibitor for p38 MAP Kinase
Koppelman, Bruce, Webb, Heather K., Medicherla, Satyanarayana, Almirez, Ramona, Feng, Ying, Chavez, Jose Carlos, Mao, Cheng Ping, Nguyen, Aaron, Liu, Yu-Wang, Kapoun, Ann M., Muiru, Gladys, Huang, Yuanying Anne, Dugar, Sundeep, Mavunkel, Babu J., Lim, Don W., Chakravarty, Sarvajit, Luedtke, Gregory, Protter, Andrew A., Higgins, Linda S.
Published in Pharmacology (01.01.2008)
Published in Pharmacology (01.01.2008)
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Journal Article
Synthesis and Characterization of Pseudopeptide Bradykinin B2 Receptor Antagonists Containing the 1,3,8-Triazaspiro[4.5]decan-4-one Ring System
Mavunkel, Babu J, Lu, Zhijian, Goehring, R. Richard, Lu, Songfeng, Chakravarty, Sarvajit, Perumattam, John, Novotny, Elizabeth A, Connolly, Maureen, Valentine, Heather, Kyle, Donald J
Published in Journal of medicinal chemistry (02.08.1996)
Published in Journal of medicinal chemistry (02.08.1996)
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Journal Article
Piperidine-based heterocyclic oxalyl amides as potent p38a MAP kinase inhibitors
Mavunkel, Babu J, Perumattam, John J, Tan, Xuefei, Luedtke, Gregory R, Lu, Qing, Lim, Don, Kizer, Darin, Dugar, Sundeep, Chakravarty, Sarvajit, Xu, Yong-Jin, Jung, Joon, Liclican, Albert, Levy, Daniel E, Tabora, Jocelyn
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Design and synthesis of piperazine-indole p38a MAP kinase inhibitors with improved pharmacokinetic profiles
Tan, Xuefei, Tester, Richland W, Luedtke, Gregory R, Chakravarty, Sarvajit, Mavunkel, Babu J, Perumattam, John J, Lu, Qing, Nashashibi, Imad, Jung, Joon, Hu, Jie, Liclican, Albert, Almirez, Ramona, Tabora, Jocelyn, Tran, Vinh, Laney, Maureen, Levy, Daniel E, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Aryl–indolyl maleimides as inhibitors of CaMKIIδ. Part 1: SAR of the aryl region
Levy, Daniel E., Wang, Dan-Xiong, Lu, Qing, Chen, Zheng, Perumattam, John, Xu, Yong-jin, Liclican, Albert, Higaki, Jeffrey, Dong, Hanmin, Laney, Maureen, Mavunkel, Babu, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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Journal Article
Pyrimidine-based inhibitors of CaMKIIδ
Mavunkel, Babu, Xu, Yong-jin, Goyal, Bindu, Lim, Don, Lu, Qing, Chen, Zheng, Wang, Dan-Xiong, Higaki, Jeffrey, Chakraborty, Indrani, Liclican, Albert, Sideris, Steve, Laney, Maureen, Delling, Ulrike, Catalano, Rosanne, Higgins, Linda S., Wang, Hui, Wang, Jing, Feng, Ying, Dugar, Sundeep, Levy, Daniel E.
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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Journal Article
Aryl-indolyl maleimides as inhibitors of CaMKIIδ. Part 2: SAR of the amine tether
Levy, Daniel E., Wang, Dan-Xiong, Lu, Qing, Chen, Zheng, Perumattam, John, Xu, Yong-jin, Higaki, Jeffrey, Dong, Hanmin, Liclican, Albert, Laney, Maureen, Mavunkel, Babu, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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Journal Article
Preventive and therapeutic potential of p38 alpha-selective mitogen-activated protein kinase inhibitor in nonobese diabetic mice with type 1 diabetes
Medicherla, Satyanarayana, Protter, Andrew A, Ma, Jing Ying, Mangadu, Ruban, Almirez, Ramona, Koppelman, Bruce, Kerr, Irene, Navas, Tony A, Movius, Fabiola, Reddy, Mamatha, Liu, Yu-Wang, Luedtke, Gregory, Perumattam, John, Mavunkel, Babu, Dugar, Sundeep, Schreiner, George F
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
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Journal Article
Preventive and Therapeutic Potential of p38α-Selective Mitogen-Activated Protein Kinase Inhibitor in Nonobese Diabetic Mice with Type 1 Diabetes
Satyanarayana Medicherla, Andrew A. Protter, Jing Ying Ma, Ruban Mangadu, Ramona Almirez, Bruce Koppelman, Irene Kerr, Tony A. Navas, Fabiola Movius, Mamatha Reddy, Yu-Wang Liu, Gregory Luedtke, John Perumattam, Babu Mavunkel, Sundeep Dugar, George F. Schreiner
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2006)
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Journal Article
A Combinatorial Approach to the Identification of Dipeptide Aldehyde Inhibitors of β-Amyloid Production
Higaki, Jeffrey N, Chakravarty, Sarvajit, Bryant, Carmen M, Cowart, Lisa R, Harden, Paul, Scardina, Jan Marian, Mavunkel, Babu, Luedtke, Gregory R, Cordell, Barbara
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Journal Article
Pharmacological Properties of SD-282 - An [alpha]-Isoform Selective Inhibitor for p38 MAP Kinase
Koppelman, Bruce, Webb, Heather K, Medicherla, Satyanarayana, Almirez, Ramona, Feng, Ying, Chavez, Jose Carlos, Mao, Cheng Ping, Nguyen, Aaron, Liu, Yu-wang, Kapoun, Ann M, Muiru, Gladys, Huang, Yuanying Anne, Dugar, Sundeep, Mavunkel, Babu J, Lim, Don W, Chakravarty, Sarvajit, Luedtke, Gregory, Protter, Andrew A, Higgins, Linda S
Published in Pharmacology (01.03.2008)
Published in Pharmacology (01.03.2008)
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Journal Article
Aryl-indolyl maleimides as inhibitors of CaMKIIdelta. Part 1: SAR of the aryl region
Levy, Daniel E, Wang, Dan-Xiong, Lu, Qing, Chen, Zheng, Perumattam, John, Xu, Yong-Jin, Liclican, Albert, Higaki, Jeffrey, Dong, Hanmin, Laney, Maureen, Mavunkel, Babu, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (01.04.2008)
Published in Bioorganic & medicinal chemistry letters (01.04.2008)
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Journal Article
Aryl-indolyl maleimides as inhibitors of CaMKIIdelta. Part 2: SAR of the amine tether
Levy, Daniel E, Wang, Dan-Xiong, Lu, Qing, Chen, Zheng, Perumattam, John, Xu, Yong-Jin, Higaki, Jeffrey, Dong, Hanmin, Liclican, Albert, Laney, Maureen, Mavunkel, Babu, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (01.04.2008)
Published in Bioorganic & medicinal chemistry letters (01.04.2008)
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Journal Article
Indole-based heterocyclic inhibitors of p38alpha MAP kinase: designing a conformationally restricted analogue
Mavunkel, Babu J, Chakravarty, Sarvajit, Perumattam, John J, Luedtke, Gregory R, Liang, Xi, Lim, Don, Xu, Yong-jin, Laney, Maureen, Liu, David Y, Schreiner, George F, Lewicki, John A, Dugar, Sundeep
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Journal Article
Antioedematogenic and antinociceptive actions of NPC 18521, a novel bradykinin B 2 receptor antagonist
De Campos, Rafael O.P., Alves, Ricardo V., Kyle, Donald J., Chakravarty, Sarvajit, Mavunkel, Babu J., Calixto, João B.
Published in European journal of pharmacology (05.12.1996)
Published in European journal of pharmacology (05.12.1996)
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