BCX4430, a novel nucleoside analog, effectively treats yellow fever in a Hamster model
Julander, Justin G, Bantia, Shanta, Taubenheim, Brian R, Minning, Dena M, Kotian, Pravin, Morrey, John D, Smee, Donald F, Sheridan, William P, Babu, Yarlagadda S
Published in Antimicrobial agents and chemotherapy (01.11.2014)
Published in Antimicrobial agents and chemotherapy (01.11.2014)
Get full text
Journal Article
Activity of Galidesivir in a Hamster Model of SARS-CoV-2
Taylor, Ray, Bowen, Richard, Demarest, James F, DeSpirito, Michael, Hartwig, Airn, Bielefeldt-Ohmann, Helle, Walling, Dennis M, Mathis, Amanda, Babu, Yarlagadda S
Published in Viruses (21.12.2021)
Published in Viruses (21.12.2021)
Get full text
Journal Article
Plasmodium falciparum parasites are killed by a transition state analogue of purine nucleoside phosphorylase in a primate animal model
Cassera, María B, Hazleton, Keith Z, Merino, Emilio F, Obaldia, 3rd, Nicanor, Ho, Meng-Chiao, Murkin, Andrew S, DePinto, Richard, Gutierrez, Jemy A, Almo, Steven C, Evans, Gary B, Babu, Yarlagadda S, Schramm, Vern L
Published in PloS one (11.11.2011)
Published in PloS one (11.11.2011)
Get full text
Journal Article
Protection against filovirus diseases by a novel broad-spectrum nucleoside analogue BCX4430
Warren, Travis K, Wells, Jay, Panchal, Rekha G, Stuthman, Kelly S, Garza, Nicole L, Van Tongeren, Sean A, Dong, Lian, Retterer, Cary J, Eaton, Brett P, Pegoraro, Gianluca, Honnold, Shelley, Bantia, Shanta, Kotian, Pravin, Chen, Xilin, Taubenheim, Brian R, Welch, Lisa S, Minning, Dena M, Babu, Yarlagadda S, Sheridan, William P, Bavari, Sina
Published in Nature (London) (17.04.2014)
Published in Nature (London) (17.04.2014)
Get full text
Journal Article
Berotralstat (BCX7353): Structure-Guided Design of a Potent, Selective, and Oral Plasma Kallikrein Inhibitor to Prevent Attacks of Hereditary Angioedema (HAE)
Kotian, Pravin L, Wu, Minwan, Vadlakonda, Satish, Chintareddy, Venkat, Lu, Pengcheng, Juarez, Luis, Kellogg-Yelder, Debra, Chen, Xilin, Muppa, Saritha, Chambers-Wilson, Ramanda, Davis Parker, Cynthia, Williams, Jason, Polach, Kevin J, Zhang, Weihe, Raman, Krishnan, Babu, Yarlagadda S
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
Get full text
Journal Article
A direct-acting antiviral drug abrogates viremia in Zika virus-infected rhesus macaques
Lim, So-Yon, Osuna, Christa E, Best, Katharine, Taylor, Ray, Chen, Elsa, Yoon, Gyeol, Kublin, Jessica L, Schalk, Dane, Schultz-Darken, Nancy, Capuano, Saverio, Safronetz, David, Luo, Ma, MacLennan, Steve, Mathis, Amanda, Babu, Yarlagadda S, Sheridan, William P, Perelson, Alan S, Whitney, James B
Published in Science translational medicine (10.06.2020)
Published in Science translational medicine (10.06.2020)
Get more information
Journal Article
Synthesis of novel azasugar-containing 2'β-C-Me 9-deaza nucleosides as potential anti-hepatitis C virus agents
Kotian, Pravin L., Wu, Minwan, Ghosh, Ajit, Polach, Kevin J., El-Kattan, Yahya, Kumar, V. Satish, Lin, Tsu-Hsing, Cheng, Xiaogang, Bantia, Shanta, Raman, Krishnan, Chand, Pooran, Babu, Yarlagadda S.
Published in Nucleosides, nucleotides & nucleic acids (2023)
Published in Nucleosides, nucleotides & nucleic acids (2023)
Get full text
Journal Article
Oral Administration of Cyclopentane Neuraminidase Inhibitors Protects Ferrets against Influenza Virus Infection
SWEET, Clive, JAKEMAN, Kenneth J, BUSH, Karen, WAGAMAN, Pamela C, MCKOWN, Linda A, STREETER, Anthony J, DESAI-KRIEGER, Daksha, CHAND, Pooran, BABU, Yarlagadda S
Published in Antimicrobial Agents and Chemotherapy (01.04.2002)
Published in Antimicrobial Agents and Chemotherapy (01.04.2002)
Get full text
Journal Article
Design and Synthesis of Benzoic Acid Derivatives as Influenza Neuraminidase Inhibitors Using Structure-Based Drug Design
Chand, Pooran, Babu, Yarlagadda S, Bantia, Shanta, Chu, Naiming, Cole, L. Brent, Kotian, Pravin L, Laver, W. Graeme, Montgomery, John A, Pathak, Ved P, Petty, Sandra L, Shrout, David P, Walsh, David A, Walsh, Gerald M
Published in Journal of medicinal chemistry (05.12.1997)
Published in Journal of medicinal chemistry (05.12.1997)
Get full text
Journal Article
Potent orally bioavailable purine nucleoside phosphorylase inhibitor BCX-4208 induces apoptosis in B- and T-lymphocytes—A novel treatment approach for autoimmune diseases, organ transplantation and hematologic malignancies
Bantia, Shanta, Parker, Cynthia, Upshaw, Ramanda, Cunningham, Amanda, Kotian, Pravin, Kilpatrick, J. Michael, Morris, Philip, Chand, Pooran, Babu, Yarlagadda S.
Published in International immunopharmacology (01.07.2010)
Published in International immunopharmacology (01.07.2010)
Get full text
Journal Article
Comparison of the anti-influenza virus activity of cyclopentane derivatives with oseltamivir and zanamivir in vivo
Chand, Pooran, Bantia, Shanta, Kotian, Pravin L., El-Kattan, Yahya, Lin, Tsu-Hsing, Babu, Yarlagadda S.
Published in Bioorganic & medicinal chemistry (02.06.2005)
Published in Bioorganic & medicinal chemistry (02.06.2005)
Get full text
Journal Article
ALK2 - IMIDAZOLE-CONTAINING INHIBITORS OF ALK2 KINASE
KUMAR V. SATISH, ZHANG WEIHE, LU PENG CHENG, KOTIAN PRAVIN L, RAMAN KRISHNAN, BABU YARLAGADDA S
Year of Publication 10.05.2024
Get full text
Year of Publication 10.05.2024
Patent
KLK5의 이환식 헤테로방향족 저해제
DANG ZHAO, ZHANG WEIHE, LU PENG CHENG, KOTIAN PRAVIN L, RAMAN KRISHNAN, BABU YARLAGADDA S
Year of Publication 20.12.2023
Get full text
Year of Publication 20.12.2023
Patent
HUMAN PLASMA KALLIKREIN INHIBITORS
WU MINWAN, KUMAR V. SATISH, ZHANG WEIHE, KOTIAN PRAVIN L, BABU YARLAGADDA S, CHINTAREDDY VENKAT R
Year of Publication 28.03.2023
Get full text
Year of Publication 28.03.2023
Patent