Strategies To Design Selective Histone Deacetylase Inhibitors
Melesina, Jelena, Simoben, Conrad V., Praetorius, Lucas, Bülbül, Emre F., Robaa, Dina, Sippl, Wolfgang
Published in ChemMedChem (06.05.2021)
Published in ChemMedChem (06.05.2021)
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Journal Article
Development of Alkylated Hydrazides as Highly Potent and Selective Class I Histone Deacetylase Inhibitors with T cell Modulatory Properties
Sun, Ping, Wang, Jing, Khan, Khadija S., Yang, Weiqin, Ng, Billy Wai-Lung, Ilment, Nikita, Zessin, Matthes, Bülbül, Emre F., Robaa, Dina, Erdmann, Frank, Schmidt, Matthias, Romier, Christophe, Schutkowski, Mike, Cheng, Alfred Sze-Lok, Sippl, Wolfgang
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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Journal Article
Synthesis and biological evaluation of triazolyl-substituted benzyloxyacetohydroxamic acids as LpxC inhibitors
Hoff, Katharina, Mielniczuk, Sebastian, Agoglitta, Oriana, Iorio, Maria Teresa, Caldara, Manlio, Bülbül, Emre F., Melesina, Jelena, Sippl, Wolfgang, Holl, Ralph
Published in Bioorganic & medicinal chemistry (01.07.2020)
Published in Bioorganic & medicinal chemistry (01.07.2020)
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Journal Article
Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic Activity
Ibrahim, Hany S, Abdelsalam, Mohamed, Zeyn, Yanira, Zessin, Matthes, Mustafa, Al-Hassan M, Fischer, Marten A, Zeyen, Patrik, Sun, Ping, Bülbül, Emre F, Vecchio, Anita, Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Barinka, Cyril, Romier, Christophe, Schutkowski, Mike, Krämer, Oliver H, Sippl, Wolfgang
Published in International journal of molecular sciences (29.12.2021)
Published in International journal of molecular sciences (29.12.2021)
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Journal Article
Comparison of laparoscopic and open ureterolysis for retroperitoneal fibrosis: Results from a tertiary referral center
İlki, Fahri Yavuz, Bülbül, Emre, Gultekin, Mehmet Hamza, Citgez, Sinharib, Demirdag, Cetin, Ozden, Sami Berk, Onal, Bulent
Published in Journal of endourology (01.11.2022)
Published in Journal of endourology (01.11.2022)
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Journal Article
Small Changes Make the Difference for SIRT2: Two Different Binding Modes for 3‑Arylmercapto-Acylated Lysine Derivatives
Kalbas, Diana, Meleshin, Marat, Liebscher, Sandra, Zessin, Matthes, Melesina, Jelena, Schiene-Fischer, Cordelia, Bülbül, Emre Fatih, Bordusa, Frank, Sippl, Wolfgang, Schutkowski, Mike
Published in Biochemistry (Easton) (06.09.2022)
Published in Biochemistry (Easton) (06.09.2022)
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Journal Article
Thiazole‐substituted benzoylpiperazine derivatives as acetylcholinesterase inhibitors
Sahin, Zafer, Ertas, Merve, Bender, Ceysu, Bülbül, Emre F., Berk, Barkin, Biltekin, Sevde N., Yurttaş, Leyla, Demirayak, Şeref
Published in Drug development research (01.12.2018)
Published in Drug development research (01.12.2018)
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Journal Article
Application of Ligand- and Structure-Based Prediction Models for the Design of Alkylhydrazide-Based HDAC3 Inhibitors as Novel Anti-Cancer Compounds
Bülbül, Emre F, Robaa, Dina, Sun, Ping, Mahmoudi, Fereshteh, Melesina, Jelena, Zessin, Matthes, Schutkowski, Mike, Sippl, Wolfgang
Published in Pharmaceuticals (Basel, Switzerland) (01.07.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.07.2023)
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Journal Article
Docking, Binding Free Energy Calculations and In Vitro Characterization of Pyrazine Linked 2-Aminobenzamides as Novel Class I Histone Deacetylase (HDAC) Inhibitors
Bülbül, Emre F, Melesina, Jelena, Ibrahim, Hany S, Abdelsalam, Mohamed, Vecchio, Anita, Robaa, Dina, Zessin, Matthes, Schutkowski, Mike, Sippl, Wolfgang
Published in Molecules (Basel, Switzerland) (14.04.2022)
Published in Molecules (Basel, Switzerland) (14.04.2022)
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Journal Article
Synthesis, biological evaluation, and molecular docking studies of deoxygenated C-glycosides as LpxC inhibitors
Dreger, Alexander, Hoff, Katharina, Agoglitta, Oriana, Bülbül, Emre F., Melesina, Jelena, Sippl, Wolfgang, Holl, Ralph
Published in Bioorganic chemistry (01.12.2021)
Published in Bioorganic chemistry (01.12.2021)
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Journal Article
Ureteral wall thickness at the stone site: A critical predictor of success and complications in children undergoing semi-rigid ureteroscopy
Kırlı, Elif Altınay, Bülbül, Emre, Kaygısız, Onur, Yeni, Sezgin, Can, Günay, Tutar, Onur, Onal, Bulent
Published in Journal of pediatric urology (01.12.2021)
Published in Journal of pediatric urology (01.12.2021)
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Journal Article
Does prolonged QTc predict pulmonary involvement in COVID-19 patients?
SARIHAN, Aydın, RAHMAN, Ömer Faruk, KORAN, Serhat, AYTEMİZ, Fatih, CAN, Çağdaş, RAHMAN, Fatih, BULBUL, Emre
Published in The European research journal (04.11.2023)
Published in The European research journal (04.11.2023)
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Journal Article
Novel thiazole‐piperazine derivatives as potential cholinesterase inhibitors
Demirayak, Şeref, Şahin, Zafer, Ertaş, Merve, Bülbül, Emre Fatih, Bender, Ceysu, Biltekin, Sevde Nur, Berk, Barkin, Sağlık, Begüm Nurpelin, Levent, Serkan, Yurttaş, Leyla
Published in Journal of heterocyclic chemistry (01.12.2019)
Published in Journal of heterocyclic chemistry (01.12.2019)
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Journal Article
Synthesis, biological evaluation, and molecular docking studies of aldotetronic acid-based LpxC inhibitors
Wimmer, Stefan, Hoff, Katharina, Martin, Benedikt, Grewer, Martin, Denni, Laura, Lascorz Massanet, Raquel, Raimondi, Maria Valeria, Bülbül, Emre F., Melesina, Jelena, Hotop, Sven-Kevin, Haupenthal, Jörg, Rohde, Holger, Heisig, Peter, Hirsch, Anna K.H., Brönstrup, Mark, Sippl, Wolfgang, Holl, Ralph
Published in Bioorganic chemistry (01.02.2023)
Published in Bioorganic chemistry (01.02.2023)
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Journal Article
Rarely Observed Sports Injuries: Two Case Reports
Uzun, Erdal, Kizkapan, Turan Bilge, Bulbul, Emre
Published in Akademik acil tıp olgu sunumları dergisi (01.01.2016)
Published in Akademik acil tıp olgu sunumları dergisi (01.01.2016)
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Journal Article
Kayseri İlinde Halkın 112 Acil Yardım Hizmetleri Hakkında Bilgi, Düşünce ve Memnuniyet Düzeyleri
DOĞAN, Mehmet, ŞENOL, Vesile, ÇETİNKAYA, Fevziye, NAÇAR, Melis, BÜLBÜL, Emre
Published in Çağdaş tıp dergisi (30.09.2020)
Published in Çağdaş tıp dergisi (30.09.2020)
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