Therapy with a Selective Cannabinoid Receptor Type 2 Agonist Limits Albuminuria and Renal Injury in Mice with Type 2 Diabetic Nephropathy
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Aleglitazar, a new, potent, and balanced dual PPARα/γ agonist for the treatment of type II diabetes
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Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Effects of pioglitazone and fenofibrate co-administration on bone biomechanics and histomorphometry in ovariectomized rats
Smith, Susan Y., Samadfam, Rana, Chouinard, Luc, Awori, Malaika, Bénardeau, Agnes, Bauss, Frieder, Guldberg, Robert E., Sebokova, Elena, Wright, Matthew B.
Published in Journal of bone and mineral metabolism (01.11.2015)
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Effects of aleglitazar, a balanced dual peroxisome proliferator-activated receptor α/γ agonist on glycemic and lipid parameters in a primate model of the metabolic syndrome
Hansen, Barbara C, Tigno, Xenia T, Bénardeau, Agnes, Meyer, Markus, Sebokova, Elena, Mizrahi, Jacques
Published in Cardiovascular diabetology (20.01.2011)
Published in Cardiovascular diabetology (20.01.2011)
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The Impact of the Nitric Oxide (NO)/Soluble Guanylyl Cyclase (sGC) Signaling Cascade on Kidney Health and Disease: A Preclinical Perspective
Krishnan, Shalini M, Kraehling, Jan R, Eitner, Frank, Bénardeau, Agnès, Sandner, Peter
Published in International journal of molecular sciences (09.06.2018)
Published in International journal of molecular sciences (09.06.2018)
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Design and Biological Evaluation of Novel, Balanced Dual PPARα/γ Agonists
Grether, Uwe, Bénardeau, Agnes, Benz, Jörg, Binggeli, Alfred, Blum, Denise, Hilpert, Hans, Kuhn, Bernd, Märki, Hans Peter, Meyer, Markus, Mohr, Peter, Püntener, Kurt, Raab, Susanne, Ruf, Armin, Schlatter, Daniel
Published in ChemMedChem (08.06.2009)
Published in ChemMedChem (08.06.2009)
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Novel soluble guanylyl cyclase activators increase glomerular cGMP, induce vasodilation and improve blood flow in the murine kidney
Stehle, Daniel, Xu, Min Ze, Schomber, Tibor, Hahn, Michael G., Schweda, Frank, Feil, Susanne, Kraehling, Jan R., Eitner, Frank, Patzak, Andreas, Sandner, Peter, Feil, Robert, Bénardeau, Agnès
Published in British journal of pharmacology (01.06.2022)
Published in British journal of pharmacology (01.06.2022)
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Runcaciguat, a novel soluble guanylate cyclase activator, shows renoprotection in hypertensive, diabetic, and metabolic preclinical models of chronic kidney disease
Bénardeau, Agnès, Kahnert, Antje, Schomber, Tibor, Meyer, Jutta, Pavkovic, Mira, Kretschmer, Axel, Lawrenz, Bettina, Hartmann, Elke, Mathar, Ilka, Hueser, Joerg, Kraehling, Jan R., Eitner, Frank, Hahn, Michael G., Stasch, Johannes-Peter, Sandner, Peter
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.12.2021)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.12.2021)
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6‑Alkoxy-5-aryl-3-pyridinecarboxamides, a New Series of Bioavailable Cannabinoid Receptor Type 1 (CB1) Antagonists Including Peripherally Selective Compounds
Röver, Stephan, Andjelkovic, Mirjana, Bénardeau, Agnès, Chaput, Evelyne, Guba, Wolfgang, Hebeisen, Paul, Mohr, Susanne, Nettekoven, Matthias, Obst, Ulrike, Richter, Wolfgang F, Ullmer, Christoph, Waldmeier, Pius, Wright, Matthew B
Published in Journal of medicinal chemistry (27.12.2013)
Published in Journal of medicinal chemistry (27.12.2013)
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The sGC Activator Runcaciguat Has Kidney Protective Effects and Prevents a Decline of Kidney Function in ZSF1 Rats
Kraehling, Jan R, Benardeau, Agnes, Schomber, Tibor, Popp, Laura, Vienenkoetter, Julia, Ellinger-Ziegelbauer, Heidrun, Pavkovic, Mira, Hartmann, Elke, Siudak, Krystyna, Freyberger, Alexius, Hagelschuer, Ina, Mathar, Ilka, Hueser, Joerg, Hahn, Michael G, Geiss, Volker, Eitner, Frank, Sandner, Peter
Published in International journal of molecular sciences (01.09.2023)
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Mechanisms underlying off-target effects of the cholesteryl ester transfer protein inhibitor torcetrapib involve L-type calcium channels
Clerc, Roger G, Stauffer, Andrea, Weibel, Franziska, Hainaut, Emmanuelle, Perez, Anne, Hoflack, Jean-Christophe, Bénardeau, Agnès, Pflieger, Philippe, Garriz, Jose Mr, Funder, John W, Capponi, Alessandro M, Niesor, Eric J
Published in Journal of hypertension (01.08.2010)
Published in Journal of hypertension (01.08.2010)
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Nitric oxide regulates the calcium current in isolated human atrial myocytes
Kirstein, M, Rivet-Bastide, M, Hatem, S, Bénardeau, A, Mercadier, J J, Fischmeister, R
Published in The Journal of clinical investigation (01.02.1995)
Published in The Journal of clinical investigation (01.02.1995)
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Animal Models of Diabetic Macrovascular Complications: Key Players in the Development of New Therapeutic Approaches
Gomez, Maria F., Jönsson-Rylander, Ann-Cathrine, Benardeau, Agnes, Hiss, Katrin, Åkesson, Lina, Hübschle, Thomas, Bengtsson, Eva, Genové, Guillem, Heinonen, Suvi E., Ylä-Herttuala, Seppo
Published in Journal of Diabetes Research (01.01.2015)
Published in Journal of Diabetes Research (01.01.2015)
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Different Compartments of Sarcoplasmic Reticulum Participate in the Excitation-Contraction Coupling Process in Human Atrial Myocytes
Hatem, Stephane N, Benardeau, Agnes, Rucker-Martin, Catherine, Marty, Isabelle, de Chamisso, Patricia, Villaz, Michel, Mercadier, Jean-Jacques
Published in Circulation research (01.03.1997)
Published in Circulation research (01.03.1997)
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The Renoprotective Effects of the Soluble Guanylate Cyclase (sGC) Activator Runcaciguat Are Associated with Distinct Changes in Renal Gene Expression Profiles: PO0708
Kraehling, Jan R., Ellinger-Ziegelbauer, Heidrun C., Benardeau, Agnes M., Pavkovic, Mira, Mathar, Ilka, Vienenkoetter, Julia, Eitner, Frank, Sandner, Peter
Published in Journal of the American Society of Nephrology (01.10.2021)
Published in Journal of the American Society of Nephrology (01.10.2021)
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Assessment of Candidate Renal Protective Drug-Induced Biomarkers in Diabetic Kidney Disease Using Targeted Proteomic Profiling: PO0721
Goea, Laura, Benardeau, Agnes M., Liu, Shuya, Lu, Shun, Ju, Wenjun, Eitner, Frank, Huber, Tobias B., Schomber, Tibor
Published in Journal of the American Society of Nephrology (01.10.2021)
Published in Journal of the American Society of Nephrology (01.10.2021)
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ACE Inhibition and GLP1 Receptor Agonism Have Direct Effects on the Glomerular Capillary Wall to Reduce Glomerular Albumin Permeability in Diabetes: TH-PO193
Crompton, Michael, Butler, Matthew J., Welsh, Gavin I., Bhayana, Sagar, Foster, Rebecca R., Benardeau, Agnes M., Satchell, Simon C., Renal, Bristol
Published in Journal of the American Society of Nephrology (01.11.2022)
Published in Journal of the American Society of Nephrology (01.11.2022)
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Discovery of the Soluble Guanylate Cyclase Activator Runcaciguat (BAY 1101042)
Hahn, Michael G, Lampe, Thomas, El Sheikh, Sherif, Griebenow, Nils, Woltering, Elisabeth, Schlemmer, Karl-Heinz, Dietz, Lisa, Gerisch, Michael, Wunder, Frank, Becker-Pelster, Eva-Maria, Mondritzki, Thomas, Tinel, Hanna, Knorr, Andreas, Kern, Armin, Lang, Dieter, Hueser, Joerg, Schomber, Tibor, Benardeau, Agnes, Eitner, Frank, Truebel, Hubert, Mittendorf, Joachim, Kumar, Vijay, van den Akker, Focco, Schaefer, Martina, Geiss, Volker, Sandner, Peter, Stasch, Johannes-Peter
Published in Journal of medicinal chemistry (13.05.2021)
Published in Journal of medicinal chemistry (13.05.2021)
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