Design, Synthesis, In Vitro Anti-cancer Activity, ADMET Profile and Molecular Docking of Novel Triazolo[3,4-a]phthalazine Derivatives Targeting VEGFR-2 Enzyme
El-Helby, Abdel-Ghany A, Sakr, Helmy, Ayyad, Rezk R A, El-Adl, Khaled, Ali, Mamdouh M, Khedr, Fathalla
Published in Anti-cancer agents in medicinal chemistry (01.01.2018)
Published in Anti-cancer agents in medicinal chemistry (01.01.2018)
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Phthalazine-1,4-dione derivatives as non-competitive AMPA receptor antagonists: design, synthesis, anticonvulsant evaluation, ADMET profile and molecular docking
El-Helby, Abdel-Ghany A., Ayyad, Rezk R. A., El-Adl, Khaled, Elkady, Hazem
Published in Molecular diversity (01.05.2019)
Published in Molecular diversity (01.05.2019)
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Design, synthesis, in silico ADMET profile and GABA‐A docking of novel phthalazines as potent anticonvulsants
El‐Helby, Abdel‐Ghany A., Ayyad, Rezk R. A., Zayed, Mohamed F., Abulkhair, Hamada S., Elkady, Hazem, El‐Adl, Khaled
Published in Archiv der Pharmazie (Weinheim) (01.05.2019)
Published in Archiv der Pharmazie (Weinheim) (01.05.2019)
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Design, Synthesis, Molecular Docking, and Anticancer Activity of Phthalazine Derivatives as VEGFR‐2 Inhibitors
El‐Helby, Abdel‐Ghany A., Ayyad, Rezk R. A., Sakr, Helmy, El‐Adl, Khaled, Ali, Mamdouh M., Khedr, Fathalla
Published in Archiv der Pharmazie (Weinheim) (01.12.2017)
Published in Archiv der Pharmazie (Weinheim) (01.12.2017)
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Design, molecular docking and synthesis of some novel 4-acetyl-1-substituted-3,4-dihydroquinoxalin-2(1H)-one derivatives for anticonvulsant evaluation as AMPA-receptor antagonists
El-Helby, Abdel-Ghany A., Ayyad, Rezk R. A., El-Adl, Khaled, Sakr, Helmy, Abd-Elrahman, Ashraf A., Eissa, Ibrahim H., Elwan, Alaa
Published in Medicinal chemistry research (01.12.2016)
Published in Medicinal chemistry research (01.12.2016)
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